A Facile Synthesis of 5-Arylidene-2-imino-4-thiazolidinones Under Microwave Irradiation

REFERENCES

• Blanchet , J. ; Zhu , J. Reeves synthesis of 2-imino-4-thiazolidinone from alkyl (aryl) trichloromethylcarbinol revisited: A three-component process from aldehyde, chloroform, and thiourea . Tetrahedron Lett. 2004 , 45 , 4449 – 4452 .
   Web of Science ®Google Scholar
• Troutman , H. D. ; Long , L. M. The synthesis of 2,3-disubstituted-4-thiazolidinones . J. Am. Chem. Soc. 1948 , 70 , 3436 – 3439 .
   PubMed Web of Science ®Google Scholar
• Vicini , P. ; Geronikaki , A. ; Anastasia , K. ; Incerti , M. ; Zani , F. Synthesis and antimicrobial activity of novel 2-thiazolylimino-5-arylidene-thiazolidinones . Bioorg. Med. Chem. 2006 , 14 , 3859 – 3864 .
   PubMed Web of Science ®Google Scholar
• El-Gendy , Z. ; Abdel-Rahman , R. M. ; Fawzy , M. M. ; Mahmoud , M. B. Biologically active thiazolidinone, part II: Synthesis and fungitoxicities of isolated and fused thiazolidinones derived from thiosemicarbazones . J. Indian Chem. Soc. 1990 , 67 , 927 – 929 .
   Web of Science ®Google Scholar
• Zervosen , A. ; Lu , W. P. ; Chen , Z. ; White , R. E. ; Demuth Jr. , T. P. ; Frère , J. M. Interaction between penicillin-binding proteins (PBPs) and two novel classes of PBP inhibitors, arylalkylidene rhodanines and arylalkylidene iminothiazolidin-4-ones. Antimicrob. Agents Chemother. 2004, 48, 961–969.
   PubMed Web of Science ®Google Scholar
• Diurno , M. V. ; Mazzoni , O. ; Piscopo , E. ; Calignano , A. ; Giordano , F. ; Bolognese , A. Synthesis and antihistaminic activity of some thiazolidin-4-ones . J. Med. Chem. 1992 , 35 , 2910 – 2912 .
   PubMed Web of Science ®Google Scholar
• Bhargava , P. N. ; Prakash , S. ; Lakhan , R. Synthesis of 2-(4′,5′-disubstituted thiazol-2′-ylimino)-3-(methylphenyl)-5-methyl(or H)-thiazolidin-4-ones and their fungicidal activity . Indian J. Chem. 1981 , 20B , 927 – 929 .
   Google Scholar
• Liu , H.-L. ; Li , Z. ; Anthonsen , T. Synthesis and fungicidal activity of 2-imino-3-(4-aryl-thiazol-2-yl)-thiazolidin-4-ones and their 5-arylidene derivatives . Molecules 2000 , 5 , 1055 – 1061 .
   Web of Science ®Google Scholar
• Zhou , J.-F. ; Song , Y.-Z. ; Yang , Y.-L. ; Zhu , Y.-L. ; Tu , S.-J. One-step synthesis of 2-aryl-4,5-diphenylimidazoles under microwave irradiation . Syn. Commun. 2005 , 35 , 1369 – 1373 .
   Web of Science ®Google Scholar
• Ottana , R. ; Maccari , R. ; Barreca , M. L. ; Bruno , G. ; Rotondo , A. ; Rossi , A. ; Chiricosta , G. ; Di-Paola , R. ; Sautebin , L. ; Cuzzocrea , S. ; Vigorita , M. G. 5-Arylidene-2-imino-4-thiazolidinones: Design and synthesis of novel antiinflammatory agents . Bioorg. Med. Chem. 2005 , 13 , 4243 – 4252 .
   PubMed Web of Science ®Google Scholar
• Andreanil , A. ; Rambaldil , M. ; Leonil , A. ; Locatellil , A. ; Bossa , R. ; Chiericozzi , M. ; Galatulasz , I. ; Salvatore , G. Synthesis and cardiotonic activity of imidazo[2,1 = b]thiazoles bearing a lactam ring . Eur. J. Med. Chem. 1996 , 31 , 383 – 387 .
   Google Scholar
• Lakhan , R. ; Singh , R. L. Synthesis and evaluation of 2-imino-3-(4-arylthiazol-2-yl)-4-thiazolidinones and their 5-arylidene derivatives as potential fungicides . J. Agric. Food Chem. 1991 , 39 , 580 – 583 .
   Web of Science ®Google Scholar