REFERENCES
- Sheehan , D. J. ; Hitchcock , C. A. ; Sibley , C. M. Current and emerging azole antifungal agents . Clin. Microbiol. Rev. 1999 , 12 ( 1 ), 40 – 79 .
- Saji , I. ; Tamoto , K. ; Tanaka , Y. ; Miyauchi , H. ; Fujimoto , K. ; Ohashi , N. Stereoselective synthesis of antifungal agents threo-2-(2,4-difluorophenyl)-3-methylsulfonyl-1-(1H-1,2,4-triazol-1-yl)-2-butanol (SM-8668). Bull. Chem. Soc. Jpn. 1994, 67, 1427–1433.
- Tasaka , A. ; Tamura , N. ; Matsushita , Y. ; Kitazaki , T. ; Hayashi , R. ; Okonogi , K. ; Itoh , K. Optically active antifungal azoles, IV: Synthesis and antifungal activity of (2 R,3 R)-3-azoyl-2-(substituted phenyl)-1-(1H-1,2,4-triazol-1-yl)-2-butanols . Chem. Pharm. Bull. 1995 , 43 ( 3 ), 432 – 440 .
- Gala , D. ; DiBenedetto , D. J. ; Mergelsberg , I. ; Kugelman , M. Total chiral synthesis of azole antifungals via α-hydroxylation of ketones . Tetrahedron Lett. 1996 , 37 ( 43 ), 8117 – 8120 .
- Kaku , Y. ; Tsuruoka , A. ; Kakinuma , H. ; Tsukuda , I. ; Yanagisawa , M. ; Naito , T. A novel route for chiral synthesis of triazole antifungal ER-30346 . Chem. Pharm. Bull. 1998 , 46 ( 7 ), 1125 – 1129 .
- Bennet , F. ; Ganguly , A. K. ; Girijavallabhan , V. M. ; Pinto , P. A an enantioselective synthesis of the antifungal agent (2 R,3 R)-(2,4-difluorophenyl)-3-methylsulfonyl-1-(1H-1,2,4-triazol-1-yl)-2-butanol (Sch 42427; SM-8668) . Synlett. 1995 , 1110 – 1113 .
- Soukup , M. Intermediate halophenyl derivatives and their use in a process for preparing azole derivatives. Patent PTC WO03/002498A1 , 2003 .
- Tamaru , Y. ; Tanaka , A. ; Yasui , K. ; Goto , S. ; Tanaka , S. Highly stereoselective allylation of benzaldehyde: Generation of a stereochemically defined allylzinc species from a π-allypalladium intermediate and diethylzinc . Angew. Chem., Int. Ed. Engl. 1995 , 34 , 787 .
- Marshall , J. A. , Adams , N. D. Synthesis of Chiral Enantioenriched Homopropargylic Mesylates Via Chiral Allylzinc Intermediates . J. Org. Chem. 1998 , 63 , 3812 – 3813 .
- Marshall , J. A. ; Wolf , M. A. ; Wallace , E. M. Synthetic routes to allenic acids and esters and their stereospecific conversion to butenolides . J. Org. Chem. 1997 , 62 , 367 .
- Sato , F. ; An , D. K. ; Okamoto , S. Synthetic routes to allyltitaniums having axial chirality by the reaction of optically active propargylic compounds with Ti(O-i-Pr)4/2-i-PrMgCl reagent . Tetrahedron Lett. 1998 , 39 , 4555 – 4558 .