Heterocyclic Synthesis Using Nitrilimines, Part 12: Synthesis and Bioactivity of 5-Carboxymethylthio-1,2,4-triazoles

REFERENCES

• Dalloul , H. M. ; Al-Abadla , N. S. ; El-Nwairy , K. A. Heterocyclic synthesis using nitrilimines part 6: Synthesis of some new substituted 4,5-dihydro-1H-1,2,4-triazoles . Chem. Heterocycl. Compd. 2007 , 3 , 392 – 397 .
   Google Scholar
• Padwa , A. 1,3-Dipolar Cycloaddition Chemistry ; A. Padwa (Ed.); Wiley Interscience : New York , 1984 ; vol. 2 , chap 12 .
   Google Scholar
• Padwa , A. ; Schoffsttall , A. M. Advances in Cycloaddition ; D. P. Curran (Ed.); JAI : London , 1990 ; Vol. 2 , pp. 1 – 89 .
   Google Scholar
• Awadallah , A. M. ; Ferwanah , A. S. ; Elsawi , E. A. ; Dalloul , H. M. 1,2,4-Triazoles from 1,3-dipolar cycloaddition reaction of nitrilimines with aliphatic ketohydrazones carrying electron withdrawing groups . Asian J. Chem. 2002 , 14 , 1230 – 1234 .
   Google Scholar
• Dalloul , H. M. Heterocyclic synthesis using nitrilimines, part 4: Synthesis of 3-substituted 1-aryl-1,2,4-triazaspiroalk-2-nes . Chem. Heterocycl. Compd. 2004 , 40 , 1402 – 1407 .
   Google Scholar
• Dalloul , H. M. ; Boyle , P. H. Heterocyclic synthesis using nitrilimines, part 7: Synthesis of some new 3-substituted 1-aryl-1,2,4,8-tetraazaspiro[4.5]dec-2-enes . Heterocycl. Commun. 2007 , 13 , 155 – 160 .
   Web of Science ®Google Scholar
• (a) Hegarty , A. F. Stereospecific reactions of nitrilium ions and analogous 1,3-dipoles . Acc. Chem. Res. 1980 , 13 , 448 – 454 ; (b) Shawali , A. S. ; Hassaneen , H. M. ; Shetta , A. ; Osman , A. ; Abdel-Galil , F. Regioselectivity of reactions of furoyl-N-aryl nitrile imine with some dipolarophiles . Heterocycles 1982 , 19 , 57 – 62 .
   Google Scholar
• Dalloul , H. H. Synthesis of spiroheterocycles with the triazole and thiazolidinone moieties from nitrilimines . J. Chin. Chem. Soc. 2009 , 56 , 196 – 201 .
   Web of Science ®Google Scholar
• Ye , X. X. ; Chen , Z. F. ; Zhang , A. J. ; Zhang , L. X. Synthesis and biological evaluation of some novel schiff's bases from 1,2,4-triazoles . Molecules 2007 , 12 , 1202 – 1209 .
   PubMedGoogle Scholar
• Zhou , S. N. ; Zhang , L. X. ; Jin , J. Y. ; Zhang , A. J. ; Lei , X. X. ; Lin , J. S. ; Zhang , H. L. Synthesis and biological activities of some novel triazolothiadiazines and schiff bases derived from 1,2,4-triazole . Phosphorus, Sulfur Silicon Relat. Elem. 2007 , 182 , 419 – 432 .
   Web of Science ®Google Scholar
• Nadkarni , B. A. ; Kamat , V. R. ; Khadse , B. G. Synthesis and anthelmintic activity of 3,6-disubstituted-7H-s-triazolo[3,4-b]-1,3,4-thiadiazin . Arzeim. Forsch. 2001 , 51 , 569 – 573 .
   PubMed Web of Science ®Google Scholar
• Holla , B. S. ; Akberali , P. M. ; Shivananda , M. K. Studies on nitrophenylfuran derivatives, part XII: Synthesis, characterization, antibacterial and antiviral of some nitrophenyl-furfurylidene-1,2,4-triazolo[3,4-b]-1,3,4-thiadiazine . Farmaco 2001 , 56 , 919 – 927 .
   PubMedGoogle Scholar
• Hui , X. P. ; Zhang , Y. ; Xu , P. F. ; Wang , Q. ; Zhang , Q. ; Zhang , Z. Y. Syntheses and antibacterial activities of novel 3-substituted-6-(4-chlorophenyl)-7-(1H-1,2,4-triazole-1-yl)-1,2,4′-triazolo[3,4-b]-1,3,4-thiadiazine . Chin. J. Org. Chem. 2005 , 25 , 700 – 704 .
   Web of Science ®Google Scholar
• Holla , B. S. ; Rao , B. S. ; Sarojini , B. K. ; Akberali , P. M. ; Kumari , N. S. ; Synthesis and studies on some new fluorine containing triazolothiadiazines as possible antibacterial, antifungal, and anticancer agents . Eur. J. Med. Chem. 2006 , 41 , 657 – 663 .
   PubMed Web of Science ®Google Scholar
• Dalloul , H. M. Heterocyclic synthesis using nitrilimines, part 8: Synthesis of aromatic triazoles. J. Islamic Univ. Gaza (Ser. Nat. Stud. Eng.) 2008, 16, 112–120.
   Google Scholar
• Collins , C. H. Microbiological Methods ; Butterworths : London , 1967 ; p. 364 .
   Google Scholar
• El-Adadelah , M. M. ; Hussein , A. Q. ; Thaher , B. A. Heterocycles from nitrile imines, part IV: Chiral 4,5-dihydro-1,2,4-triazin-ones . Heterocycles 1991 , 32 , 1887 – 1995 .
   Google Scholar
• Farag , A. M. ; Algharib , M. S. Synthesis and reactions of C-(2-thenoyl)-N-aryl-formhydrazidoyl bromides . Org. Prep. Proced. Int. 1988 , 20 , 521 – 526 .
   Web of Science ®Google Scholar
• Frohberg , P. ; Drutkowski , G. ; Wagner , C. Synthesis and structural assignment of oxanilo-N-arylhydrazonoyl chlorides . Eur. J. Org. Chem. 2002 , 1654 – 1663 .
   Google Scholar
• Hassaneen , H. M. ; Shawali , A. S. ; Elwan , N. M. ; Abounada , N. M. Synthesis of pyrazolo[3,4-d]pyridazine, pyrazolo[3,4-d]pyrimidine, and imidazolo[1,2-a]pyridine derivatives using hydrazonyl bromides . Org. Prep. Proced. Int. 1992 , 24 , 171 – 175 .
   Web of Science ®Google Scholar
• Hassaneen , H. M. ; Shawali , A. S. ; Elwan , M. ; Abunada , N. M. Reaction of 1-(2-naphthoyl)methyl-2-dimethylsulfonium bromide with N-nitroso-N-arylacetamides and reactions of the products with some nucleophiles . Sulfur Lett. 1992 , 13 , 273 – 285 .
   Google Scholar