Publication Cover
Synthetic Communications
An International Journal for Rapid Communication of Synthetic Organic Chemistry
Volume 40, 2010 - Issue 4
93
Views
4
CrossRef citations to date
0
Altmetric
Original Articles

Green Synthesis of Some New (Substituted Fluorobenzoylimino)-3-aryl-4-methyl-1,3-thiazolines

&
Pages 564-569 | Received 26 Feb 2009, Published online: 03 Feb 2010

REFERENCES

  • Klijin , J. E. ; Engberts , J. B. F. N. Fast reactions “on water” . Nature 2005 , 435 , 746 .
  • Narayan , S. ; Muldoon , J. ; Finn , M. G. ; Fokin , V. V. ; Kolb , H. C. ; Sharpless , K. B. “On Water”: Unique reactivity of organic compounds in aqueous suspension . Angew. Chem. Int. Ed. 2005 , 44 , 3275 .
  • Breslow , R. ; Rizzo , C. J. Chaotropic salt effects in a hydrophobically accelerated Diels–Alder reaction . J. Am. Chem. Soc. 1991 , 113 , 4340 – 4341 .
  • Jacobson , G. B. ; Lee Jr. , T. C. ; da Rocha , S. R. P. ; Johnston , K. P. Organic synthesis in water/carbon dioxide emulsions . J. Org. Chem. 1999 , 64 ( 4 ), 1207 .
  • Vicini , P. ; Geronikaki , A. ; Anastasia , K. ; Incerti , M. ; Zani , F. Synthesis and antimicrobial activity of novel 2-thiazolylimino-5-arylidene-4-thiazolidinones . Bioorg. Med. Chem. 2006 , 14 , 3859 .
  • (a) Zhang , A. ; Kaiser , H. ; Maienfisch , P. ; Casida , J. E. Insect nicotinic acetylcholine receptor: Conserved neonicotinoid specificity of [3H]imidacloprid binding site . J. Neurochem. 2000 , 75 , 1294 ; (b) Maienfisch , P. ; Haettenschwiler , J. ; Rindlisbacher , A. ; Decock , A. ; Wellmann , H. ; Kayser , H. Azido-neonicotinoids as candidate photoaffinity probes for insect nicotinic acetylcholine receptors . Chimia 2003 , 57 , 710 .
  • (a) Hosseinimehr , S. J. ; Shafiee , A. ; Mozdarani , H. ; Akhlagpour , S. Radioprotective effects of 2-iminothiazolidine derivatives against lethal doses of gamma radiation in mice . J. Radiat. Res. 2001 , 42 , 401 ; (b) Hosseinimehr , S. J. ; Shafiee , A. ; Mozdarani , H. ; Akhlagpour , S. ; Froughizadeh , M. Radioprotective effects of 2-imino-3-[(chromone-2-yl)carbonyl]thiazolidines against γ-irradiation in mice . J. Radiat. Res. 2002 , 43 , 293 .
  • Bae , S. ; Hahn , H.-G. ; Nam , K. D. Solid-phase synthesis of fungitoxic 2-imino-1,3-thiazolines . J. Comb. Chem. 2005 , 7 , 7 .
  • Kim , D.-S. ; Jeong , Y.-M. ; Park , I.-K. ; Hahn , H.-G. ; Lee , H.-K. ; Kwon , S.-B. ; Yang , S. J. ; Sohn , U. D. ; Park , K.-C. A new 2-imino-1,3-thiazoline derivative, KHG22394, inhibits melanin synthesis in mouse B16 melanoma cells . Biol. Pharm. Bull. 2007 , 30 , 180 .
  • Pietrancosta , N. ; Moumen , A. ; Dono , R. ; Lingor , P. ; Planchamp , V. ; Lamballe , F. ; Bähr , M. ; Kraus , J.-L. ; Maina , F. Imino-tetrahydro-benzothiazole deriatives as p53 inhibitors: Discovery of a highly potent in vivo inhibitor and its action mechanism . J. Med. Chem. 2006 , 49 , 3645 .
  • Sondhi , S. M. ; Singh , S. ; Kumar , A. ; Jamal , H. ; Gupta , P. P. Synthesis of amidine and amide derivatives and their evaluation for anti-inflammatory and analgesic activities . Eur. J. Med. Chem. 2008 , 30 , 1 .
  • Manaka , A. ; Sato , M. ; Aoki , M. ; Tanaka , M. ; Ikeda , T. ; Toda , Y. ; Yamanane , Y. ; Nakaike , S. 2-Acylimino-3H-thiazoline derivatives: A novel template for platelet GPIIb/IIIa receptor antagonists . Bioorg. Med. Chem. Lett. 2001 , 11 , 1031 .
  • Sondhi , S. M. ; Singh , N. ; Lahoti , A. M. ; Bajaj , K. ; Kumar , A. ; Lozach , O. ; Meijer , L. Synthesis of acridinyl-thiazoline derivatives and their evaluation for anti-inflammatory, analgesic, and kinase inhibition activities . Bioorg. Med. Chem. 2005 , 13 , 4291 .
  • Shih , M.-H. ; Ke , F.-Y. Synthesis and evaluation of antioxidant activity of sydnonyl substituted thiazolidinone and thiazoline derivatives. J. Bioorg. Med. Chem. 2004, 12, 4633.
  • Sanemitsu , Y. ; Kawamura , S. ; Satoh , J. ; Katayama , T. ; Hashimoto , S. Synthesis and herbicidal activity of 2-acylimino-3-phenyl-1,3-thiazolines—A new family of bleaching herbicides . J. Pestic. Sci. 2006 , 31 , 305 .
  • Zeng , R.-S. ; Zou , J.-P. ; Zhi , S.-J. ; Chen , J. ; Shen , Q. Novel synthesis of 1-aroyl-3-aryl-4-substituted imidazole-2-thiones . Org. Lett. 2003 , 5 , 1657 .
  • Singh , C. B. ; Murru , S. ; Kavala , V. ; Patel , B. K. It is “thiazolidene-2-imine” and not imidazole-2-thione as the reaction product of 1-benzoyl-3-phenylthiourea with Br2/enolizable ketone . Org. Lett. 2006 , 8 , 5397 .
  • Germanas , J. P. ; Wang , S. ; Miner , A. ; Hao , W. ; Ready , J. M. Discovery of small-molecule inhibitors of tyrosinase . Bioorg. Med. Chem. Lett. 2007 , 17 , 6871 .
  • Saeed , A. ; Zaman , S. ; Bolte , M. Synthesis and crystal structure of some novel 2-aroylimino-3-aryl-4-phenyl-1,3-thiazolines . Synth. Commun. 2008 , 38 , 2185 .
  • Saeed , A. ; Parvez , M. The crystal structure of 1-(4-chlorophenyl)-3-(4-methylbenzoyl)thiourea . Cent. Eur. J. Chem. 2005 , 3 , 780 .

Reprints and Corporate Permissions

Please note: Selecting permissions does not provide access to the full text of the article, please see our help page How do I view content?

To request a reprint or corporate permissions for this article, please click on the relevant link below:

Academic Permissions

Please note: Selecting permissions does not provide access to the full text of the article, please see our help page How do I view content?

Obtain permissions instantly via Rightslink by clicking on the button below:

If you are unable to obtain permissions via Rightslink, please complete and submit this Permissions form. For more information, please visit our Permissions help page.