Facile Novel Synthesis and Reactions of Thiazolidin-4-one Derivatives for Antimicrobial Agents

REFERENCES

• Küçükgüzel , G. ; Kocatepe , A. ; De Clercq , E. ; Şahin , F. ; Güllüce , M. Synthesis and biological activity of 4-thiazolidinones, thiosemicarbazides derived from diflunisal hydrazide . Eur. J. Med. Chem. 2006 , 41 , 353 – 359 .
   PubMed Web of Science ®Google Scholar
• Chen , H. ; Bai , J. ; Jiao , L. ; Guo , Z. ; Yin , Q. ; Li , X. Design, microwave-assisted synthesis, and HIV-RT inhibitory activity of 2-(2,6-dihalophenyl)-3-(4,6-dimethyl-5-(un)substituted-pyrimidin-2-yl) thiazolidin-4-ones . Bioorg Med. Chem. Lett. 2009 , 17 ( 11 ), 3980 – 3986 .
   Web of Science ®Google Scholar
• Rao , A. ; Balzarini , J. ; Carbone , A. ; Chimirri , A. ; De Clercq , E. ; Monforte , A. M. ; Monforte , P. ; Pannecouque , C. ; Zappalà , M. 2-(2,6-Dihalophenyl)-3-(pyrimidin-2-yl)-1,3-thiazolidin-4-ones as non-nucleoside HIV-1 reverse transcriptase inhibitors . Antiviral Res. 2004 , 63 ( 2 ), 79 – 84 .
   PubMed Web of Science ®Google Scholar
• Srivastava , T. ; Haq , W. ; Katti , S. B. Carbodiimide-mediated synthesis of 4-thiazolidinones by one-pot, three-component condensation . Tetrahedron 2002 , 58 , 7619 – 7624 .
   Web of Science ®Google Scholar
• Colombo , A. ; Fernàndez , J. C. ; Fernández-Forner , D. ; de la Figuera , N. ; Albericio , F. ; Forns , P. Stereomeric studies on the oxidation and alkylation of 4-thiazolidinones . Tetrahedron Lett. 2008 , 49 ( 10 ), 1569 – 1572 .
   Web of Science ®Google Scholar
• Barreca , M. L. ; Chimirri , A. ; De Luca , L. ; Monforte , A. M. ; Monforte , P. ; Rao , A. ; Zappalà , M. ; Balzarini , J. ; De Clercq , E. ; Pannecouque , C. ; Witvrouw , M. Discovery of 2,3-diaryl-1,3-thiazolidin-4-ones as potent anti-HIV-1 agents . Bioorg Med. Chem. Lett. 2001 , 11 ( 13 ), 1793 – 1796 .
   PubMed Web of Science ®Google Scholar
• Jain , S. C. ; Sinha , J. ; Bhagat , S. ; Errington , W. ; Olsen , C. E. A facile synthesis of novel spiro-[indole-pyrazolinyl-thiazolidine]-2,4′-dione . Synth. Commun. 2003 , 33 , 563 – 577 .
   Web of Science ®Google Scholar
• Lewis , A. F. ; Drach , J. C. ; Fennewald , S. M. ; Huffman , J. H. ; Ptak , R. G. ; Sommadossi , J. P. ; Revankar , G. R. ; Rando , R. F. Inhibition of human cytomegalo virus in culture by alkenyl guanine analogs of the thiazolo[4,5-d]pyrimidine ring system. J. Antimicrob. Agents Chemother. 1994, 38(12), 2889–2895.
   PubMed Web of Science ®Google Scholar
• Binnun , E. ; Connolty , P. J. ; Johnson , S. G. ; Lin , R. ; Middleton , S. A. ; Moreno , S. J. ; Pandey , N. B. ; Water , S. Thiazolopyrimidine modulators of TRRVI. U.S. Patent 514,260,100, 2007.
   Google Scholar
• Amr , A. E. ; Maigali , S. S. ; Abdulla , M. M. Synthesis and analgesic and antiparkinsonian activities of thiopyrimidine, pyrane, pyrazoline, and thiazolopyrimidine derivatives from 2-chloro-6-ethoxy-4-acetylpyridine . Monatsch. Chem. 2008 , 139 , 1409 – 1415 .
   Web of Science ®Google Scholar
• Diego , M. J. ; Antonio , M. ; Yolanda , R. ; Andres , R. G. ; Ether , P. C. ; Manuel , M. A. ; Arat , N. V. ; Squella , L. J. ; Juan , A. ; Jorge , E. F. ; Arturo , S. O. Trypanosoma cruzi inhibition of parasite growth and respiration by oxazolo(thiazolo)pyridine derivatives and its relationship to redox potential and lipoplicity . J. Exper. Parasit. 2001 , 99 ( 1 ), 1 – 6 .
   PubMed Web of Science ®Google Scholar
• Sayed , H. H. ; Shamroukh , A. H. ; Rashad , A. E. Synthesis and biological evaluation of some pyrimidine, pyrimido[2,1-b][1,3]thiazine, and thiazolo[3,2-a]pyrimidine derivatives . Acta Pharm. 2006 , 56 , 231 – 244 .
   PubMedGoogle Scholar
• Amr , A. E. ; Sayed , H. H. ; Abdulla , M. A. Synthesis and reactions of some new substituted pyridine and pyrimidine derivatives as analgesic, anticonvulsant, and antiparkinsonian agents . Arch. Pharm. Chem. Life Sci. 2005 , 338 , 433 – 440 .
   PubMed Web of Science ®Google Scholar
• Sayed , H. H. Reactions of α,β-spiro alkanones, part VI: Reactions of spirononanones with amine and thiourea . Indian J. Chem. 1998 , 37B , 1045 – 1058 .
   Google Scholar
• Sayed , H. H. Synthesis and reactions of 3-aryloxiran-2-yl-pyridin-2-yl methanone: A novel synthesis of triazolopyrimidine for biological evaluation . Egypt. J. Chem. 2005 , 48 ( 2 ), 223 – 234 .
   Google Scholar
• Sayed , H. H. ; Moustafa , A. H. ; Yousif , N. M. ; Assy , M. G. ; Abd El-Halim , M. A. Synthesis and reactions of some novel mercaptopyrimidine derivatives for biological evaluation . Phosphorus, Sulfur Silicon Relat. Elem. 2008 , 183 , 2318 – 2329 .
   Web of Science ®Google Scholar
• Sayed , H. H. ; Ali , M. A. Synthesis of 3-[(4-chloro-phenyl) oxiranyl]thiophen-2-yl-propanone and their reactions with some nucleophilles for antiviral evaluations . Phosphorus, Sulfur Silicon Relat. Elem. 2008 , 183 , 156 – 167 .
   Web of Science ®Google Scholar
• Shamroukh , A. H. ; Zaki , M. E. A. ; Morsy , E. M. H. ; Abdel-Motti , F. M. ; Abdel-Megeid , F. M. E. Synthesis of pyrazolo[4',3':5,6]pyrano[2,3-d]pyrimidine derivatives for antiviral evaluation . Arch. Pharm. 2007 , 340 , 236 – 243 .
   PubMed Web of Science ®Google Scholar
• Shamroukh , A. H. ; Zaki , M. E. A. ; Morsy , E. M. H. ; Abdel-Motti , F. M. ; Abdel-Megeid , F. M. E. Anti-HAV activity of some newly synthesized triazolo[4,3-b]pyridazines . Arch. Pharm. 2007 , 340 , 345 – 351 .
   PubMed Web of Science ®Google Scholar
• Bauer , A. W. ; Kirby , M. M. ; Sherris , J. C. ; Turck , M. Antibiotic susceptibility testing by a standardized single disc method . Am. J. Clin. Pathol. 1996 , 45 , 493 – 496 .
   Google Scholar