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Synthetic Communications
An International Journal for Rapid Communication of Synthetic Organic Chemistry
Volume 43, 2013 - Issue 3
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Original Articles

2-Keto-3-mercaptocinchoninic Acids as Precursors for Novel Thiazino[6,5-c]quinoline-1,5-dione Derivatives

Pages 398-405 | Received 17 Mar 2011, Published online: 02 Nov 2012

REFERENCES

  • Benaed , C. ; Zouhir , Z. ; Bayle , M. N. ; Danet , M. , Desmale , D. Liker-modified quinoline derivatives targeting HIV-1 integrase synthesis and biological activity . Biorg. Med. Chem. Lett. 2004 , 14 , 2473 – 2476 .
  • Agrawal , V. K. ; Sinha , S. ; Khadikar , P. QSAR studies on series of 4-quinoliecabinol-amine, antimalarials . Indian J. Heterocycl. Chem. 2000 , 39B , 462 – 474 .
  • Aghera , V. K. ; Patel , J. P. ; Parsania , P. H. Synthesis, spectral, and microbial studies of some novel quinoline derivatives via Vilsmeier–Haack reagent . Arkivoc 2008 , 12 , 195 – 204 .
  • Kumar , S. ; Bawa , S. ; Gupta , H. Biological activities of quinoline derivatives . Mini Rev. Med. Chem. 2009 , 9 , 1648 – 1654 .
  • Korrichi , L. ; Dalila , B. ; Dalila , S. Quinoline antioxidant activity–structure relationship . Eur. J. Biolog. Sci. 2009 , 1 , 32 – 36 .
  • Eswaran , S. ; Adhikari , A. V. ; Kumar , R. A. New 1,3-oxazolo[4,5-c]quinoline derivatives: Synthesis and evolution of antibacterial and antitiuberculosis properties . Eur. J. Med. Chem. 2010 , 45 , 957 – 966 .
  • Liyang , C. ; Tseng , H. C. ; Chen , Y. L. ; Lu , C. M. ; Kao , C. L. ; Wu , M. H. ; Tzeng , C. C. Identification of benzofuro[2,3-b]quinoline derivatives as a new class of antituberculosis agents . Eur. J. Med. Chem. 2010 , 45 , 602 – 607 .
  • Fujimura , K. I. ; Fujita , M. ; Suhara , H. ; Kawashima , Y. Conformational study of 2-phenylbenzothiazine part of SA2995, a Ca2+ antagonist having a benzothiazine skeleton, and structure–activity relationships . Bioorg. Med. Chem. 1994 , 2 , 235 – 242 .
  • Brown , C. ; Davidson , R. M. 1,4-Benzothiazinesdihydro-1,4-benzothiazines and related compounds . Adv. Heterocycl. Chem. 1985 , 38 , 135 – 176 .
  • Singh , D. N. ; Verma , N. ; Pathak , L. P. Synthesis and antiviral activity of some novel N-substituted benzimidazolyl annulated pyrimidines . J. Ind. Council Chem. 2008 , 25 , 19 – 22 .
  • Koketsu , M. ; Tanaka , K. ; Takenaka , Y. ; Kwong , C. D. ; Ishihara , H. Synthesis of 1,3-thiazine derivatives and their evaluation as potential antimycobacterial agents. Eur. J. Pharm. Sci. 2002, 15, 307–310.
  • Gupta , S. ; Ajmera , N. ; Meena , P. ; Gautam , N. ; Kumar , A. ; Gautan , D. C. Jordan J. Chem. 2009 , 4 , 209 – 221 .
  • Parai , M. K. ; Panda , G. A convenient synthesis of chiral amino acid–derived 3,4-dihydro-2H-benzo[b][1,4]thiazines and antibiotic levofloxacin . Tetrahedron Lett. 2009 , 50 , 4703 – 4705 .
  • Pandey , V. K. ; Saxena , S. K. ; Joshi , M. N. ; Bajpai , S. K. Synthesis and antiviral activity of some novel substituted phenothiazines . Indian J. Chem. 2004 , 43B , 1015 – 1017 .
  • Sundari , V. ; Nagarajan , G. ; Valliappan , P. Synthesis and biological activities of some N-hydroxymethylene and N-methoxymethylene thiazines . Med. Chem. Res. 2007 , 16 , 402 – 407 .
  • Ead , H. A. ; Abdallah , S. O. ; Kassab , N. A. ; Metwally , N. H. Synthesis of the novel thiazolo[5,4-e][1,2,3]thiadiazines and their biological activities . Sulfur Lett. 1989 , 9 , 23 – 32 .
  • Ead , H. A. ; Metwally , N. H. Cleavage reactions of 4-thiazolidinone-2-thiones: Synthesis and reactions of new 1,2,4-triazoles and their biological activities . Arch. Pharm. (Weinheim) 1990 , 323 , 57 – 58 .
  • Ead , H. A. ; Metwally , N. H. ; Morsy , N. M. Cycloaddition reactions of 5-(2-thienyl)methylene derivatives of thiazolidinone-4-thiones and their antimicrobial activities . Arch. Pharm (Weinheim) 1990 , 13 , 5 – 8 .
  • Ead , H. A. ; Abdelaziz , M. A. ; Metwally , N. H. A new route for synthesis of 1,3-oxathiolanes and their biological activities . Polish J. Chem. 1991 , 65 , 1291 .
  • Elgemeie , G. E. H. ; Mansour , O. A. ; Metwally , N. H. Synthesis and anti-HIV activity of different novel nonclassical nucleosides . Nucleosides Nucleotides 1999 , 18 , 113 – 123 .
  • Metwally , N. H. A new route for synthesis of some substiuted thiazoles and thiadiazolidin-4-one and thiadiazolo[2,3-a]triazole derivatives . Indian J. Chem. 2000 , 39B , 757 – 763 .
  • Metwally , N. H. Efficient synthesis of highly substituted furan, thiophene, pyrrole and 2-aminothiazole derivatives . Synth. Commun. 2007 , 37 , 4227 – 4237 .
  • Metwally , N. H. A facile one-pot synthesis of some new spiro-thiazolidin-4-ones and benzimidazole of biological interest . Phosphorus, Sulfur Silicon Relat Elem. 2008 , 183 , 34 – 43 .
  • Metwally , N. H. ; Abdalla , M. A. ; Mosselhi , M. A. ; El-Desoky , E. A. Synthesis and antimicrobial activity of some new N-glycosides of 2-thioxo-4-thiazolidinone derivatives . Carbohydr. Res. 2010 , 345 , 1135 – 1141 .
  • Shawali , A. S. ; Harb , N. M. S. ; Badhdah , K. O. J. Heterocycl. Chem. 1985 , 22 , 1397 – 1403 .
  • Jones , R. ; Ryan , A. J. ; Sternhell , S. ; Wright , S. E. The structures of some 5-pyrazol-ones and derived 4-arylazo-5-pyrazolones . Tetrahedron 1963 , 19 , 1497 – 1507 .
  • Wright , G. E. Hydrazine-hydrazone tautomerism in phenylhydrazino pyrimidines . J. Heterocycl. Chem. 1983 , 20 , 1037 .
  • Shawali , A. S. ; Albar , A. H. Kinetics and mechanism of dehydrochlorination of N-aryl-C-ethoxycarbonylformohydrazidoyl chlorides . Can. J. Chem. 1986 , 64 , 871 – 875 .
  • Jones , R. V. ; Henze , H. R. The synthesis from rhodanine-oxindoles of keto and mercapto derivatives of cinchoninic acid . J. Am. Chem. Soc. 1942 , 64 , 1669 – 1671 .

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