REFERENCES
- Michael , A. Ueber die addition von natriumacetessig- und natriummalonsäureäthern zu den aethern ungesättigter Säuren . J. Prakt. Chem. 1887 , 35 , 349 – 356 .
- Wabnitz , T. C. ; Yu , J. Q. ; Spencer , J. B. Evidence that protons can be the active catalysts in Lewis acid–mediated hetero-Michael addition reactions . Chem. Eur. J. 2004 , 10 , 484 – 493 .
- Chamakh , A. ; Amri , H. A one-pot synthesis of (E)-4-alkylidene-2-cyclohexen-1-ones . Tetrahedron Lett. 1998 , 39 , 375 – 378 .
- Lee , K. Y. ; Gowrisankar , S. ; Kim , J. N. Baylis–Hillman reaction and chemical transformations . Bull. Korean Chem. Soc. 2005 , 26 , 1481 – 1490 .
- Ren , L. ; Piers , E. First total synthesis of (+)-pentandranoic acid A. Tetrahedron Lett. 2012, 53, 3329–3332.
- Cho , C. S. ; Patel , D. B. ; Shim , S. C. Palladium-catalyzed aromatization of β-bromovinyl aldehydes with alkenes . Tetrahedron 2005 , 61 , 9490 – 9494 .
- Schultz , A. G. ; Godfrey , J. D. An annelation approach to the synthesis of eudesmane and elemane sesquiterpene lactones: Total synthesis of dl-dihydrocallitrisin, dl-7,8-epialantolactone, dl-7,8-epiisoalantolactone, and dl-atractylon . J. Am. Chem. Soc. 1980 , 102 , 2414 – 2428 .
- Lahmar , N. ; Ben Ayed , T. ; Bellassoued , M. ; Amri , H. A convenient synthesis of γ-functionalized cyclopentenones . Beilstein J. Org. Chem. 2005 , 1 , 11 – 13 .
- Ben Ayed , T. ; El Gaïed , M. M. ; Amri , H. Conjugate addition of Grignard reagents to α-functional enone promoted by LiCuBr2 . J. Soc. Tunis. 1997 , 4 , 13 – 19 .
- Ben Ayed , T. ; Amri , H. A convenient synthesis of α-functional alkyl vinyl ketones . Synth. Commun. 1995 , 25 , 3813 – 3819 .
- (a) Belaud , C. ; Roussakis , C. ; Letourneux , Y. ; Alami , N. ; Villiéras , J. Synthèse des potentiels cytotoxiques α-méthylène γ-lactames . Synth. Commun. 1985 , 15 , 1233 – 1243 ; (b) Kornet , M. J. Synthèse des α-méthylène butyrolactams comme agents antitumoraux potentiels . J. Pharm. Sci. 1979 , 68 , 350 – 353 ; (c) Ikuta , H. ; Shirota , S. ; Kobayashi , Y. ; Yamagishi , K. ; Yamada , K. ; Yamatsu , I. ; Katayama , K. Synthesis and antiinflammatory activities of 3-(3,5-di-tert-butyl-4-hydroxybenzylidene)pyrrolidin-2-ones . J. Med. Chem. 1987 , 30 , 1995 – 1998 .
- Arfaoui , A. ; Beji , F. ; Amri , H. Effective synthesis of polysubstituted pyrroles from (E)-dimethyl 2-(bromomethyl)-3-(diethoxyphosphoryl)fumarate . Synth. Commun. 2010 , 40 , 766 – 771 .
- Krawczyk , H. ; Albrecht , L. ; Wojciechowski , J. ; Wolf , W. M. ; Krajewska , U. ; Rózalski , M. A convenient synthesis and cytotoxic evaluation of N-unsubstituted α-methylene-γ-lactams . Tetrahedron 2008 , 64 , 6307 – 6314 .
- Ballini , R. ; Gabrielli , S. ; Palmieri , A. Chemoselective SN2′ reaction of nitroalkanes to dialkyl 2-(bromomethyl)fumarates under cetyltrimethylammonium hydroxide (CTAOH) catalysis . Tetrahedron Lett. 2010 , 51 , 1233 – 1235 .
- Inguimbert , N. ; Dhôtel , H. ; Coric , Roques , B. Unexpected formation of new chiral 3-amino-5-alkyl-2,5-dihydro-1H-pyrrolin-2-ones from N-Boc-α-amino esters . Tetrahedron Lett. 2005 , 46 , 3517 – 3520 .
- Beji , F. ; Lebreton , J. ; Villiéras , J. ; Amri , H. A total stereospecific route to α-alkylidene-γ-lactams . Tetrahedron 2001 , 57 , 9959 – 9962 .
- Lee , K. Y. ; Lee , Y. J. ; Kim , J. N. Synthesis of β,γ-disubstituted α-methylene-γ-butyrolactams starting from the Baylis–Hillman adducts . Bull. Chem. Soc. 2007 , 28 , 143 – 146 .
- Basavaiah , D. ; Rao , J. S. Applications of Baylis–Hillman acetates: One-pot, facile, and convenient synthesis of substituted γ-lactams . Tetrahedron Lett. 2004 , 45 , 1621 – 1625 .
- Wu , X. M. ; Funkoshi , K. ; Sakai , K. Highly diastereoselective, enantioselective cyclization of symmetrical 3,4-disubstituted 4-pentenal using chiral rhodium(I)-complex . Tetrahedron Lett. 1993 , 34 , 5927 – 5930 .
- Ono , N. ; Yoshimura , T. ; Saito , T. ; Tamura , R. ; Tanikaga , R. ; Kaji , A. Alkylation and acylation of active methylene compounds using 1,8-diazabicyclo[5.4.0]undec-7-ene as base . Bull. Chem. Soc. Jpn. 1979 , 52 , 1716 – 1719 .
- Demir , A. S. ; Emrullahoglu , M. An effective new synthesis of 2-aminopyrrole-4-carboxylates . Tetrahedron 2005 , 61 , 10482 – 10489 .
- Robin , D. C. ; Leland , G. K. ; Clayton , H. H. Alkylation of diethyl 2-oxoalkanephosphonates . Synthesis 1975 , 635 – 636 .
- Villiéras , J. ; Rambaud , M. Wittig–Horner reaction in heterogeneous media: An efficient synthesis of α-methylenecarboxylic esters and α-methyleneketones under mild conditions . Synthesis 1984 , 406 – 408 .
- Kimura , Y. ; Atarashi , S. ; Takahashi , M. ; Hayakawa , I. Synthesis and structure–activity of 7-[3-(1-aminoalkyl)pyrrolidinyl]- and 7-[3-(1-aminocycloalkyl)pyrrolidinyl]-quinolone antibacterials. Chem. Pharm. Bull. 1994, 42, 1442–1454.
- Beltaief , I. ; Besbes , R. ; Ben Amor , F. ; Villiéras , M. ; Villiéras , J. ; Amri , H. (Z)-Dimethyl α-(bromomethyl)fumarate, an efficient intermediate for the selective synthesis of dimethyl 3-alkyl itaconates and 2-alkyl 3-carbomethoxy-γ-lactams . Tetrahedron 1999 , 55 , 3949 – 3958 .
- Baldwin , J. E. ; Thomas , R. C. ; Kruse , L. I. ; Silberman , L. Rules for ring closure: Ring formation by conjugate addition of oxygen nucleophiles . J. Org. Chem. 1977 , 42 , 3846 – 3852 .