Efficient Synthesis of Substances Related to Cinacalcet Hydrochloride via Heck Coupling

REFERENCES

• (a) Hebert , S. C. Annu. Rev. Med. 2006 , 57 , 349 – 364 ; (b) Nagano , N. Pharmacol. Ther. 2006 , 109 , 339 – 365 ; (c) Franceschini , N. ; Joy , M. S. ; Kshirsagar , A. Expert Opin. Invest. Drugs 2003 , 12 , 1413 – 1421 .
   PubMed Web of Science ®Google Scholar
• Nemeth , E. F. ; Van , W. B. C. ; Balandrin , M. F. ; Del Mar , E. G. ; Moe , S. T. U. S. Patent 6011068, January 4, 2000 .
   Google Scholar
• Thiel , O. R. ; Bernard , C. ; Tormos , W. ; Brewin , A. ; Hirotani , S. ; Murakami , K. ; Saito , K. ; Larsen , R. D. ; Martinelli , M. J. ; Reider , P. J. Tetrahedron Lett. 2008 , 49 , 13 – 15 .
   Web of Science ®Google Scholar
• Bijukumar , G. ; Maloyesh , B. ; Bhaskar , B. S. ; Rajendra , A. Synth. Commun. 2008 , 38 , 1512 – 1517 .
   Web of Science ®Google Scholar
• (a) ICH Guidelines, Q3A (R): Impurities in New Drug Substances. International Conference of Harmonisation, Geneva, Switzerland, February 2002; (b) ICH Guidelines, Q3B (R): Impurities in New Drug Products. International Conference of Harmonisation, Geneva, Switzerland, February 2002; (c) Impurities Guidelines for Residual Solvents, Q3(c). International Conference on Harmonisation, Geneva, Switzerland, 1997 .
   Google Scholar
• Wang , X. ; Chen , Y. ; Crockett , R. ; Briones , J. ; Yan , T. ; Orihuela , C. ; Zhi , B. ; Ng , J. Tetrahedron Lett. 2004 , 45 , 8355 – 8358 .
   Web of Science ®Google Scholar
• Mariappan , P. ; Muniappan , T. J. Organometal. Chem. 2000 , 609 , 137 – 151 .
   Web of Science ®Google Scholar
• Pendrak , I. ; Chambers , P. A. J. Org. Chem. 1995 , 60 , 3249 – 3251 .
   Web of Science ®Google Scholar
• Sonny , S. ; Sarma , P. S. R. ; Katikireddy , R. WO Patent 2010067204, June 17, 2010 .
   Google Scholar