References
- Wild, S.; Roglic, G.; Green, A.; Sicree, R.; King, H. Global Prevalence of Diabetes: Estimates for the Year 2000 and Projections for 2030. Diabetes Care. 2004, 27, 1047–1053. DOI: https://doi.org/10.2337/diacare.27.5.1047.
- Roglic, G.; Unwin, N.; Bennett, P. H.; Mathers, C.; Tuomilehto, J.; Nag, S.; Connolly, V.; King, H. The Burden of Mortality Attributable to Diabetes: Realistic Estimates for The Year 2000. Diabetes Care. 2005, 28, 2130–2135. DOI: https://doi.org/10.2337/diacare.28.9.2130.
- Fujisawa, T.; Ikegami, H.; Inoue, K.; Kawabata, Y.; Ogihara, T. Effect of Two Alpha-Glucosidase Inhibitors, Voglibose and Acarbose, on Postprandial Hyperglycemia Correlates with Subjective Abdominal Symptoms. Metabolism. 2005, 54, 387–390. DOI: https://doi.org/10.1016/j.metabol.2004.10.004.
- Singh, S. K.; Rai, P. K.; Jaiswal, D.; Watal, G. Evidence-Based Critical Evaluation of Glycemic Potential of Cynodon Dactylon. Evid. Based Complement. Altern. Med. 2008, 5, 415–420. DOI: https://doi.org/10.1093/ecam/nem044.
- Gachons, CPd.; Breslin, P. A. S. Salivary Amylase: digestion and Metabolic Syndrome. Curr. Diabetes Rep. 2016, 16, 1–7. DOI: https://doi.org/10.1007/s11892-016-0794-7.
- Sales, P. M.; Souza, P. M.; Simeoni, L. A.; Silveira, D. Alpha-Amylase Inhibitors: A Review of Raw Material and Isolated Compounds from Plant Source. J. Pharm. Pharmaceut. Sci. 2012, 15, 141–183. DOI: https://doi.org/10.18433/j35s3k.
- Subramanian, R.; Asmawi, M. Z.; Sadikun, A. In Vitro Alpha-Glucosidase and Alpha Amylase Enzyme Inhibitory Effects of Andrographis paniculata Extract and Andrographolide. Acta Biochim. Pol. 2008, 55, 391–398.
- Eduardo, B. D. M.; Adriane, D. S. Gomes, I. C. α- and β-Glucosidase Inhibitors: Chemical Structure and Biological Activity. Tetrahedron. 2006, 62, 10277–10302. DOI: https://doi.org/10.1016/j.tet.2006.08.055.
- Vorathavorn, V. I.; Sykes, J. E.; Feldman, D. G.; Vet, J. Cryptococcosis as an Emerging Systemic Mycosis in Dogs. J. Vet. Emerg. Crit. Care. 2013, 23, 489–497. DOI: https://doi.org/10.1111/vec.12087.
- Shiro, T.; Fukaya, T.; Tobe, M. The Chemistry and Biological Activity of Heterocycle-Fused Quinolinone Derivatives: A Review. Eur. J. Med. Chem. 2015, 97, 397–408. DOI: https://doi.org/10.1016/j.ejmech.2014.12.004.
- Bozdağ-Dündar, O.; Verspohl, E. J.; Daş-Evcimen, N.; Kaup, R. M.; Bauer, K.; Sarikaya, M.; Evranos, B.; Ertan, R. Synthesis and Biological Activity of Some New Flavonyl-2,4-Thiazolidinediones. Bioorg. Med. Chem. 2008, 16, 6747–6751. DOI: https://doi.org/10.1016/j.bmc.2008.05.059.
- Mori, M.; Takagi, M.; Noritake, C.; Kagabu, S. 2,4-Dioxo-1,3-Thiazolidine Derivatives as a Lead for New Fungicides. J. Pestic. Sci. 2008, 33, 357–363. DOI: https://doi.org/10.1584/jpestics.G08-15.
- Visentini, P. Antituberculosis Chemotherapeutic Action of Derivatives of 2-4 Thiazolidinedione. I. Action in Vitro of the 2-Phenylhydrazone of 2,4-Thiazolidinedione. Farmaco. Sci. 1954, 9, 274–277. PMID: 13191358.
- Marshall, P. G.; Vallance, D. K. Anticonvulsant Activity; Derivatives of Succinimide, Glutarimide, Thiazolidinedione and Methanol, and Some Miscellaneous Compounds. J. Pharm. Pharmacol. 1954, 6, 740–746. DOI: https://doi.org/10.1111/j.2042-7158.1954.tb11011.x.
- Ceriello, A. Thiazolidinediones as Anti-Inflammatory and Anti-Atherogenic Agents. Diabetes. Metab. Res. Rev. 2008, 24, 14–26. DOI: https://doi.org/10.1002/dmrr.790.
- Eun, J. S.; Kim, K. S.; Kim, H. N.; Park, S. A.; Ma, T.-Z.; Lee, K. A.; Kim, D. K.; Kim, H. K.; Kim, I. S.; Jung, Y. H.; et al. Synthesis of Psoralen Derivatives and Their Blocking Effect of hKv1.5 Channel. Arch. Pharm. Res. 2007, 30, 155–160. DOI: https://doi.org/10.1007/BF02977688.
- Sahu, S. K.; Banerjee, M.; Mishra, S. K.; Mohanta, R. K.; Panda, P. K.; Misro, P. K. Synthesis, Partition Coefficients and Antibacterial Activity of 3′-Phenyl (Substituted)-6′ Aryl-2′ (1H)-Cis-3′,3‘a-Dihydrospiro [3-H-Indole-3,5’-Pyrazolo (3′,4′-d)-Thiazolo-2-(1H) Ones]. Acta Pol. Pharm. 2007, 64, 121–126. PMID: 17665861
- Angajala, G.; Subashini, R. In Diabetes Mellitus and Human Health Care; Sebastian, M., Ed.; Chapter 5, Florida USA: Apple Academic Press, Inc., 2014; pp. 229–246.
- Yoshioka, T.; Fujita, T.; Kanai, T.; Aizawa, Y.; Kurumada, T.; Hasegawa, K.; Horikoshi, H. Studies on Hindered Phenols and Analogues.1-Hypolipidemic and Hypoglycemic Agents with Ability to Inhibit Lipid Peroxidation. J. Med. Chem. 1989, 32, 421–428. DOI: https://doi.org/10.1021/jm00122a022.
- Gotoda, S.; Takahashi, N.; Nakagawa, H.; Murakami, M.; Takechi, T.; Komura, T.; Uchida, T.; Takagi, Y. Synthesis and Fungicidal Activity against Pyricularia Oryzae of 6-(1,2,4-Triazol-4-yl)Chromone and -1-Thiochromone Derivatives. Pestic. Sci. 1998, 52, 309–320. DOI: https://doi.org/10.1002/(SICI)1096-9063(199804)52:4<309::AID-PS727>3.0.CO;2-J.
- Singh, B. K.; Walker, A. Microbial Degradation of Organophosphorus Compounds. FEMS Microbiol. Rev. 2006, 30, 428–471. DOI: https://doi.org/10.1111/j.1574-6976.2006.00018.x.
- Marklund, A.; Andersson, B.; Haglund, P. Screening of Organophosphorus Compounds and Their Distribution in Various Indoor Environments. Chemosphere. 2003, 53, 1137–1146. DOI: https://doi.org/10.1016/S0045-6535(03)00666-0.
- Hudson, H. R.; Wardle, N. J.; Bligh, S. W.; Greiner, I.; Grun, A.; Keglevich, G. N-Heterocyclic Dronic Acids: Applications and Synthesis. Mini-Rev. Med. Chem 2012, 12, 313–325. DOI: https://doi.org/10.2174/138955712799829285.
- De. Clercq, E. Antivirals: Past, Present and Future. Biochem. Pharmacol. 2013, 85, 727–744. DOI: https://doi.org/10.1016/j.bcp.2012.12.011.
- McKellar, Q. A.; Jackson, F. Veterinary Anthelmintics: Old and New. Trends Parasitol. 2004, 20, 456–461. DOI: https://doi.org/10.1016/j.pt.2004.08.002.
- Derbalah, A.; Chidya, R.; Jadoon, W.; Sakugawa, H. Temporal Trends in Organophosphorus Pesticides Use and Concentrations in River Water in Japan, and Risk Assessment. J. Environ. Sci. 2019, 79, 135–152. DOI: https://doi.org/10.1016/j.jes.2018.11.019.
- Cycoń, M.; Wójcik, M.; Piotrowska-Seget, Z. Biodegradation of the Organophosphorus Insecticide Diazinon by Serratia sp. and Pseudomonas sp. and Their Use in Bioremediation of Contaminated Soil. Chemosphere. 2009, 76, 494–501. DOI: https://doi.org/10.1016/j.chemosphere.2009.03.023.
- Zenneck, U.; Hofmann, M. 2.20 - Four-Membered Rings with Two Heteroatoms Including Phosphorus to Bismuth, Comprehensive Heterocyclic Chemistry III. 2008, 2, 875–905. DOI: https://doi.org/10.1016/B978-008044992-0.00220-0.
- Făgădar-Cosma, E.; Laichici, M.; Făgădar-Cosma, G.; Vlascici, D. Synthesis, Characterization and Correlative Biological Effects in Wheat of a Benzoxaza- and a Diaza-Phosphorus(V) heterocycles. J. Serb. Chem. Soc. 2006, 71, 1031–1038. DOI: https://doi.org/10.2298/JSC0610031F.
- Abdel-Aziz, S. A.-G.; Ali, T. E.-S.; El-Mahdy, K. M.; Abdel-Karim, S. M. Synthesis and Antimicrobial Activities of Some Novel Bis-Pyrazole Derivatives Containing a Hydrophosphoryl Unit. Eur. J. Chem. 2011, 2, 25–35. DOI: https://doi.org/10.5155/eurjchem.2.1.25-35.208.
- Haribabu, Y.; Srinivasulu, K.; Reddy, C. S.; Reddy, C. D. Synthesis of Novel Fused Heterocyclic System: 5-(Substituted)-5-Oxo-5H-6,12-Dioxa-5λ5-Phosphabenzo (a) Anthracene-7-Ones. Arkivoc. 2006, 15, 95–103. DOI: https://doi.org/10.3998/ark.5550190.0007.f12.
- Pettersen, E. F.; Goddard, T. D.; Huang, C. C.; Couch, G. S.; Greenblatt, D. M.; Meng, E. C.; Ferrin, T. E. UCSF Chimera – A Visualization System for Exploratory Research and Analysis. J. Comput. Chem. 2004, 25, 1605–1612. DOI: https://doi.org/10.1002/jcc.20084.
- Sujatha, B.; Subramanyam, C.; Venkataramaiah, C.; Rajendra, W.; Prasada Rao, K. Synthesis and anti-Diabetic Activity Evaluation of Phosphonates Containing Thiazolidinedione Moiety. Phos. Sulf. Silicon Relat. Elem. 2020, 195, 1–6. DOI: https://doi.org/10.1080/10426507.2020.1737061.
- Altaff, S. K.; Md, Raja Rajeswari, T.; Subramanyam, C. Synthesis, α-Amylase Inhibitory Activity Evaluation and in Silico Molecular Docking Study of Some New Phosphoramidates Containing Heterocyclic Ring. Phos. Sulf. Silicon Relat. Elem. 2021, 196, 389–397. DOI: https://doi.org/10.1080/10426507.2020.1845679.
- Quin, L. D.; Verkade, J. G. Phosphorus-31 NMR Spectral Properties Compound Characterization and Structural Analysis; VCH Publishers: New York, 1994.
- Hay, M.; Thomas, D. W.; Craighead, J. L.; Economides, C.; Rosenthal, J. Clinical Development Success Rates for Investigational Drugs. Nat. Biotechnol. 2014, 32, 40–51. DOI: https://doi.org/10.1038/nbt.2786.
- Daina, A.; Zoete, V. A Boiled-Egg to Predict Gastrointestinal Absorption and Brain Penetration of Small Molecules. Chem. Med. Chem. 2016, 11, 1117–1121. DOI: https://doi.org/10.1002/cmdc.201600182.
- Montanari, F.; Ecker, G. F. Prediction of drug-ABC-Transporter Interaction – Recent Advances and Future Challenges. Adv. Drug Deliv. Rev. 2015, 86, 17–26. DOI: https://doi.org/10.1016/j.addr.2015.03.001.
- Hollenberg, P. F. Characteristics and Common Properties of Inhibitors, Inducers, and Activators of CYP Enzymes. Drug Metab. Rev. 2002, 34, 17–35. DOI: https://doi.org/10.1081/dmr-120001387.
- Huang, S.-M.; Strong, J. M.; Zhang, L.; Reynolds, K. S.; Nallani, S.; Temple, R.; Abraham, S.; Habet, S. A.; Baweja, R. K.; Burckart, G. J.; et al. New Era in Drug Interaction Evaluation: US Food and Drug Administration Update on CYP Enzymes, Transporters, and the Guidance Process. J. Clin. Pharmacol. 2008, 48, 662–670. DOI: https://doi.org/10.1177/0091270007312153.
- Lipinski, C. A.; Lombardo, F.; Dominy, B. W.; Feeney, P. J. Experimental and Computational Approaches to Estimate Solubility and Permeability in Drug Discovery and Development Settings. Adv. Drug Del. Rev. 2001, 46, 3–26. DOI: https://doi.org/10.1016/s0169-409x(00)00129-0.
- Ghose, A. K.; Viswanadhan, V. N.; Wendoloski, J. J. Prediction of Hydrophobic (Lipophilic) Properties of Small Organic Molecules Using Fragmental Methods: An Analysis of ALOGP and CLOGP Methods. J. Phys. Chem. A. 1998, 102, 3762–3772. DOI: https://doi.org/10.1021/jp980230o.
- Veber, D. F.; Johnson, S. R.; Cheng, H. Y.; Smith, B. R.; Ward, K. W.; Kopple, K. D. Molecular Properties That Influence the Oral Bioavailability of Drug Candidates. J. Med. Chem. 2002, 45, 2615–2623. DOI: https://doi.org/10.1021/jm020017n.
- Egan, W. J.; Lauri, G. Prediction of Intestinal Permeability. Adv. Drug Del. Rev. 2002, 54, 273–289. DOI: https://doi.org/10.1016/s0169-409x(02)00004-2.
- Muegge, I.; Heald, S. L.; Brittelli, D. Simple Selection Criteria for Drug-like Chemical Matter. J. Med. Chem. 2001, 44, 1841–1846. DOI: https://doi.org/10.1021/jm015507e.
- Trott, O.; Olson, A. J. Auto Dock Vina: improving the Speed and Accuracy of Docking with a New Scoring Function, Efficient Optimization and Multithreading. J. Comput. Chem. 2010, 31, 455–461. DOI: https://doi.org/10.1002/jcc.21334.
- Nickavar, B.; Amin, G. Enzyme Assay Guided Isolation of an Alpha-Amylase Inhibitor Flavonoid from Vaccinium Arctostaphylos Leaves. Iran J. Pharm. Res. 2011, 10, 849–853.
- Patil, V. S.; Nandre, K. P.; Ghosh, S.; Rao, V. J.; Chopade, B. A.; Sridhar, B.; Bhosale, S. V.; Bhosale, S. V. Synthesis, Crystal Structure and anti-Diabetic Activity of Substituted (E)-3-(Benzo[d]Thiazol-2-Ylamino)Phenylprop-2-en-1-One. Eur. J. Med. Chem. 2013, 59, 304–309. DOI: https://doi.org/10.1016/j.ejmech.2012.11.020.
- Kumar, P.; Soni, B. R.; Kumar, M.; Singh, S. S.; Patil, K.; Baig, M.; Laxmi, R. B. N. A. Synthesis, Glucose Uptake Activity and Structure-Activity Relationships of Some Novel Glitazones Incorporated with Glycine, Aromatic and Alicyclic Amine Moieties via Two Carbon Acyl Linker. Eur. J. Med. Chem. 2011, 46, 835–844. DOI: https://doi.org/10.1016/j.ejmech.2010.12.019.
- Young, M. H.; Yun Jung, P.; Jin-Ah, K.; Daeui, P.; Ji Young, P.; Hye Jin, L. Design and Synthesis of 5-(Substituted Benzylidene)Thiazolidine-2,4-Dione Derivatives as Novel Tyrosinase Inhibitors. Eur. J. Med. Chem. 2012, 49, 245–252. PMID 22301213.
- Kawade, D.; Nitin, J.; Jadhav, V.; Girish, K. Design Synthesis and Evaluation of Novel Thiazolidinedione Derivatives as Antidiabetic Agents. Pharma Innovat. J. 2017, 6, 390–398.
- Chandra Sekhar, K.; Venkataramaiah, Ch.; Naga Raju, C. In Silico, in Ovo and in Vitro Antiviral Efficacy of Phosphorylated Derivatives of Abacavir: An Experimental Approach. J. Recept. Signal Transduct. 2020, 40, 426–435. DOI: https://doi.org/10.1080/10799893.2020.
- Madhu Kumar Reddy, K.; Peddanna, K.; Varalakshmi, M.; Bakthavatchala Reddy, N.; Sravya, G.; Grigory, V. Z.; Suresh Reddy, C. Ceric Ammonium Nitrate (CAN) Catalyzed Synthesis and α -Glucosidase Activity of Some Novel Tetrahydropyridine Phosphonate Derivatives. Phos. Sulf. Silicon Relat. Elem. 2019, 194, 812–819. DOI: https://doi.org/10.1080/10426507.2018.1550641.