Microwave-Assisted Synthesis of Propesticides 1,3,4-Thiadiazole Aminophosphonates

REFERENCES

• Schenone , S. ; Brullo , C. ; Bruno , O. ; Bondavalli , F. ; Ranise , A. ; Filippelli , W. ; Rinaldi , B. ; Capuano , A. ; Falcone , G. New 1,3,4-thiadiazole derivatives endowed with analgesic and anti-inflammatory activities . Bioorg. Med. Chem. 2006 , 14 , 1698 – 1705 .
   PubMed Web of Science ®Google Scholar
• Matysiak , J. Evaluation of antiproliferative effect in vitro of some 2-amino-5-(2,4-dihydroxyphenyl)-1,3,4-thiadiazole derivatives. Chem. Pharm. Bull. 2006, 54, 988–991.
   PubMed Web of Science ®Google Scholar
• Foroumadi , A. ; Emami , S. ; Hassanzadeh , A. ; Rajaee , M. ; Sokhanvar , K. ; Moshafi , M. ; Shafiee , A. Synthesis and antibacterial activity of N-(5-benzylthio-1,3,4-thiadiazol-2-yl) and N-(5-benzylsulfonyl-1,3,4-thiadiazol-2-yl) piperazinyl quinolone derivatives . Bioorg. Med. Chem. Lett. 2005 , 15 , 4488 – 4492 .
   PubMed Web of Science ®Google Scholar
• Tehranchian , S. ; Akbarzadeh , T. ; Fazeli , M. R. ; Jamalifar , H. ; Shafiee , A. Synthesis and antibacterial activity of 1-[1,2,4-triazol-3-yl] and 1-[1,3,4-thiadiazol-2-yl]-3-methylthio-6,7-dihydrobenzo[c]thiophen-4(5H)ones . Bioorg. Med. Chem. Lett. 2005 , 15 , 1023 – 1025 .
   PubMed Web of Science ®Google Scholar
• Thomasco , L. M. ; Gadwood , R. C. ; Weaver , E. A. ; Ochoada , J. M. ; Ford , C. W. ; Zurenko , G. E. ; Hamel , J. C. ; Stapert , D. ; Moerman , J. K. ; Schaadt , R. D. ; Yagi , B. H. The synthesis and antibacterial activity of 1,3,4-Thiadiazole phenyl oxazolidinone analogues . Bioorg. Med. Chem. Lett. 2003 , 13 , 4193 – 4196 .
   PubMed Web of Science ®Google Scholar
• Kafarski , P. ; Lejczak , B. Aminophosphonic acids of potential medical importance . Curr. Med. Chem. Anti-Cancer Agents 2001 , 1 , 301 – 312 .
   PubMedGoogle Scholar
• De Lombaert , S. ; Blanchard , L. ; Tan , J. ; Sakane , Y. ; Berry , C. ; Ghai , R. D. Nonpeptidic inhibitors of neutral endopeptidase 24.11, 1: Discovery and optimization of potency . Bioorg. Med. Chem. Lett. 1995 , 5 , 145 – 150 .
   Web of Science ®Google Scholar
• Kafarski , P. ; Lejczak , B. Biological activity of aminophosphonic acids . Phosphorus Sulfur Relat. Elem. 1991 , 63 , 193 – 215 .
   Web of Science ®Google Scholar
• Kafarski , P. ; Lejczak , B. ; Tyka , R. ; Koba , L. ; Pliszczak , E. ; Wieczorek , P. Herbicidal activity of phosphonic, phosphinic, and phosphonous acid analogues of phenylglycine and phenylalanine . J. Plant. Growth Regul. 1995 , 14 , 199 – 203 .
   Web of Science ®Google Scholar
• Perreux , L. ; Loupy , A. A tentative rationalization of microwave effects in organic synthesis according to the reaction medium and mechanistic considerations . Tetrahedron 2001 , 57 , 9199 – 9223 .
   Web of Science ®Google Scholar
• Kappe , C. O. ; Stadler , A. Microwaves in Organic and Medicinal Chemistry ; Wiley-VCH : Weinheim , 2005 .
   Google Scholar
• Wu , F. Study on the Synthesis and Biological Activity of 1,3,4-Thiadiazole Derivatives ; PhD thesis , Nanjing University of Technology : Nanjing , 2006 .
   Google Scholar