Convenient, One-Step Syntheses of 2-Fluoroveratrole And 2-Fluoroveratraldehyde

References

• March , J. 1985 . Advanced Organic Chemistry , Third Ed. , 479 593 602 – 603 . New York, NY : John Wiley and Sons . For methods of introducing fluorine into aromatic rings, see
   Google Scholar
• Kollonitsch , J. 1978 . Isr. J. Chem. , 17 : 53 “Biomedicinal Aspects of Fluorine Chemistry,” R. Filler, Y. Kobayashi, Eds., Elsevier Biomedical Press, New York, NY, 1982
   Google Scholar
• Goldberg , L. I. , Kohli , J. D. , Cantacuzene , D. , Kirk , K. L. and Creveling , C. R. 1980 . J. Pharm. Exp. Ther. , 213 : 509
   PubMedGoogle Scholar
• Daly , J. W. , Padgett , W. , Nimitkitpaisan , Y. , Creveling , C. R. , Cantacuzene , D. and Kirk , K. L. 1953 . J. Pharm. Exp. Ther. , 108 : 177 Kirk, K. L., Cantacuzene, D., Nimitkitpaisan, Y., McCulloh, D., Padgett, W. L., Daly, J. W. and Creveling, C. R., J. Med. Chem., 1979, 22, 1493
   PubMedGoogle Scholar
• Kirk , K. L. 1976 . J. Org. Chem. , 41 : 2373
   PubMed Web of Science ®Google Scholar
• Ladd , D. L. and Weinstock , J. 1981 . J. Org. Chem. , 46 : 203
   Web of Science ®Google Scholar
• Ladd , D. L. , Gaitanopoulos , D. and Weinstock , J. 1985 . Synth. Commun. , 15 : 61
   Web of Science ®Google Scholar
• Clark , M. D. and Miller , D. D. 1985 . Tetrahedron Lett. , 26 : 4299
   Web of Science ®Google Scholar
• Peet , J. H. J. and Rocket , B. W. 1974 . J. Organometal. Chem. , 82 : C57 Perchloryl fluoride (Pennwalt) is a reactive, toxic gas which should be handled with caution. We have had no adverse incidents with this reagent, sparging it into reaction solutions at 0°C. Others, however, under different conditions, have encountered violent explosions with this reagent. See Adcock, W. and Khor, T. C., J. Organometal. Chem., 1975, 91, C20; Wang, C.‐L. J., Grieco, P. A. and Okuniewicz, F. J., J. Chem. Soc., Chem. Commun., 1976, 468; and Schroepfer, G. J., Parish, E. J., Tsuda, M. and Kandutsch, A. A., Biochem. Biophys. Res. Comm., 1979, 91, 606
   Web of Science ®Google Scholar
• Comins , D. L. and Brown , J. D. 1984 . J. Org. Chem. , 49 : 1078
   Google Scholar
• Schuetz , R. D. , Taft , D. D. , O'Brien , J. P. , Shea , J. L. and Mork , H. M. 1963 . J. Org. Chem. , 28 : 1420
   Google Scholar
• Gronowitz , S. and Rosen , U. 1968 . Acta Chem. Scand. , 22 : 907 Christiansen, H., Gronowitz, S., Rodmar, B., Rodmar, S., Rosen, U. and Sharma, M. K., Arkiv KemiM, 1969, 30, 561
   Google Scholar
• LeTourneau , M. E. and McCarthy , J. R. 1984 . Tetrahedron Lett. , 25 : 5227
   Google Scholar
• McCarthy , J. R. , Peet , N. P. , LeTourneau , M. E. and Inbasekaran , M. 1985 . J. Am. Chem. Soc. , 107 : 735
   Web of Science ®Google Scholar
• Inbasekaran , M. , Peet , N. P. , McCarthy , J. R. and LeTourneau , M. E. 1985 . J. Chem. Soc., Chem. Commun. , 678
   Google Scholar
• Sharts , C. M. and Sheppard , W. A. 1974 . Org. Reactions , 21 : 225 – 236 .
   Google Scholar