Publication Cover
Synthetic Communications
An International Journal for Rapid Communication of Synthetic Organic Chemistry
Volume 17, 1987 - Issue 4
38
Views
11
CrossRef citations to date
0
Altmetric
Original Articles

Facile Formation of Quaternary Azetidinium Compounds During Triflation of Dialkylaminopropanols

&
Pages 469-475 | Published online: 05 Dec 2006

References

  • Durant , G. J. , Ganellin , C. R. and Parsons , M. E. 1977 . Agents and Actions , 7 : 39
  • For subsequent conversion of 2 to 4 in general it is still likely that 3 is formed in situ as a reaction intermediate since more vigorous reaction conditions were employed
  • As determined by TLC during reaction and work-up with confirmation after purification and NMR characterization of products
  • Moore , J. A. 1983 . “Azetidines” . In Heterocyclic Compounds , Edited by: Hassner , A. Vol. 42 , New York : John Wiley and Sons . Part 2
  • Moore , J. A. 1964 . “Trimethyleneimines” . In Heterocyclic Compounds with Three and Four Membered Rings , Edited by: Weissberger , A. New York : John Wiley and Sons .
  • Crist , D. R. , Leonard and Agnew , N. J. 1969 . Chem. Int. Ed. , 8 : 962
  • Cromwell , N. H. and Phillips , B. 1979 . Chem. Rev. , 79 : 331
  • Stang , P. J. , White and Aldrichim , M. R. 1983 . Acta , 16 : 15
  • Vaughan , W. R. , Klonowski , R. S. , McElhinney , R. S. and Millward , B. B. 1961 . J. Org. Chem. , 26 : 138
  • Hanack , M. , Kang , S. , Haeffner , J. and Goerler , K. 1965 . Ann. Chem. , 690 : 98 Prepared by treating cyclopropylphenylcarbinol with concentrated hydrochloric acid according to
  • Erhardt , P. W. 1983 . Synth. Comm. , 13 : 103 Prepared by treating benzylmethylamine with 3-chloropropanol followed by hydrogenolysis according to general methodology described previously: Boiling point was identical to that reported by: Searles, S., Gregory, V. P. J. Am. Chem. Soc., 1954, 76, 2789

Reprints and Corporate Permissions

Please note: Selecting permissions does not provide access to the full text of the article, please see our help page How do I view content?

To request a reprint or corporate permissions for this article, please click on the relevant link below:

Academic Permissions

Please note: Selecting permissions does not provide access to the full text of the article, please see our help page How do I view content?

Obtain permissions instantly via Rightslink by clicking on the button below:

If you are unable to obtain permissions via Rightslink, please complete and submit this Permissions form. For more information, please visit our Permissions help page.