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Synthetic Communications
An International Journal for Rapid Communication of Synthetic Organic Chemistry
Volume 20, 1990 - Issue 3
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Original Articles

Synthesis of 5-Aryluridines and 5-Aryl-2′-deoxyuridines

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Pages 413-422 | Received 02 Oct 1989, Published online: 24 Oct 2006

References

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  • Hawthorne , M. F. 1958 . J. Am. Chem. Soc. , 80 : 4291 The required arylboronic acids are readily prepared by reaction of aryllithium or aryl Grignard reagents with tributylborate followed by mild acid hydrolysis. For example see:
  • Miyaura , N. , Yanagi , T. and Suzuki , A. 1981 . Synth. Commun. , 11 : 513
  • Eaborn , C. and Waters , J. A. 1962 . J. Chem. Soc. , : 1131 Aryltrimethylstannanes were conveniently prepared by reaction of chlorotrimethylstannane with the appropriate aryllithium or aryl Grignard reagent. For example see:

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