Concise and Efficient Synthesis of 1H-Pyrazoles: Reaction of [Hydroxy(tosyloxy)iodo]benzene with Ethyl 2,3-Dioxobutanoate-2-arylhydrazones

References

• Goodman , L. S. and Gilman , A. 1980 . The Pharmacological Basis of Therapeutics , New York : Macmillan .
   Google Scholar
• Wachter , M. and Ferro , M. U. S. Patent 4826868 . 1989 .
   Google Scholar
• 1988 . Chem. Abstr. , 108 : 186735v
   Google Scholar
• Argentieri , D. , Ritchie , D. , Tolman , E. , Ferro , M. , Wachter , M. , Mezick , J. and Capetola , R. 1988 . The FASEB Journal Antiinflammatory agents , 2 : A369 Vol. 4
   Google Scholar
• Secor , H. V. and De Bardelaben , J. F. 1971 . J. Med. Chem. , 14 : 997
   PubMed Web of Science ®Google Scholar
• Bauer , V. J. , Fanshawe , W. J. , Dalalian , H. P. , Safir , S. R. , Tocus , E. C. and Boshart , C. R. 1968 . J. Med. Chem. , 11 : 981
   PubMed Web of Science ®Google Scholar
• Corsi , G. , Germani , C. , Palazzo , G. , Silvestrini , B. and Barcellona , P. S. 1976 . J. Med. Chem. , 19 : 778
   PubMed Web of Science ®Google Scholar
• Durham , N. N. , Chesnut , R. W. , Hashem , M. M. and Berlin , K. D. 1976 . J. Med. Chem. , 19 : 229
   PubMed Web of Science ®Google Scholar
• Wiley , R. H. 1967 . Pyrazoles, Pyrazolines, Pyrazolidines, Indazoles and Condensed Rings; , New York : Wiley . For general reviews on synthesis of pyrazoles see:
   Google Scholar
• Kost , A. N. and Grandberg , I. I. 1966 . Advances in Heterocyclic Chemistry , Edited by: Katritzky , A. R. and Boulton , A. J. Vol. 6 , 347 New York : Academic .
   Google Scholar
• Jacobs , T. L. 1957 . Heterocyclic Compounds; , Edited by: Elderfield , R. C. Vol. 5 , 45 New York : Wiley .
   Google Scholar
• Volkov , A. N. and Nikol'skaya , A. N. 1977 . Russ. Chem. Rev. , 46 : 374
   Google Scholar
• Friestone , R. A. 1977 . Tetrahedron , 33 : 3009
   Google Scholar
• Wagner-Jauregg , T. 1976 . Synthesis , : 349
   Google Scholar
• Coispeau , G. and Elguero , J. 1970 . Bull. Soc. Chim. Fr. , : 2711
   Google Scholar
• Sokolvo , S. D. 1979 . Russ. Chem. Rev. , 48 : 289
   Google Scholar
• Elguero , J. 1984 . Comprehensive Heterocyclic Chemistry , Edited by: Potts , K. T. Vol. 5 , 167 New York : Pergamon .
   Google Scholar
• Hafez , E. A. A. , Abed , N. M. , Elmoghayer , M. R. H. and El-Agamey , A. G. 1984 . Heterocyles , 22 : 1821
   Google Scholar
• Elnagdi , M. H. , Elgemeie , G. E. H. and Abd-Elaal , F. A. 1985 . Heterocyles , 23 : 3121
   Web of Science ®Google Scholar
• Patel , H. V. , Vyas , K. A. and Fernandes , P. S. 1990 . Indian J. Chem. , 29B : 966
   Google Scholar
• Patel , H. V. , Vyas , K. A. and Pernandes , P. S. 1990 . Indian J. Chem. , 29B : 836
   Google Scholar
• Patel , H. V. and Fernandes , P. S. 1989 . Indian J. Chem. , 28B : 470
   Google Scholar
• Patel , H. V. and Fernandes , P. S. 1989 . Indian J. Chem. , 28B : 56
   Google Scholar
• Moriarty , R. M. and Prakash , O. 1986 . Acc. Chem. Res. , 19 : 244
   Web of Science ®Google Scholar
• Moriarty , R. M. , Vaid , R. K. and Koser , G. F. 1990 . Synlett , : 365
   Web of Science ®Google Scholar
• Moriarty , R. M. and Vaid , R. K. 1990 . Synthesis , : 431
   Web of Science ®Google Scholar
• Merkushev , E. B. 1987 . Russ. Chem. Rev. (Eng. Transl.) , 56 : 826
   Google Scholar
• Varvoglis , A. 1984 . Synthesis , : 709
   Google Scholar
• Varvoglis , A. 1981 . Chem. Soc. Rev. , 10 : 377
   Web of Science ®Google Scholar
• Koser , G. F. 1983 . The Chemistry of Functional Groups, Supplement D , Edited by: Patai , S. and Rappoport , Z. 721 Chichester : Wiley . Chap. 18 Chap. 25, p1265
   Google Scholar
• Banks , D. F. 1966 . Chem. Rev. , 66 : 243
   Web of Science ®Google Scholar
• Koser , G. F. , Relenyi , A. G. , Kalos , A. N. , Rebrovic , L. and Wettach , R. H. 1982 . J. Org. Chem. , 47 : 2487
   Web of Science ®Google Scholar
• Moriarty , R. M. , Penmasta , R. , Awasthi , A. K. , Epa , W. R. and Prakash , I. 1989 . J. Org. Chem. , 54 : 1101
   Web of Science ®Google Scholar
• Parmerter , S. M. 1959 . Organic Reactions , 10 : 1 For preparation of compounds 1 see
   Google Scholar
• HTIB was obtained from Aldrich.
   Google Scholar
• Wolff , L. and Fertig , E. 1990 . Ann , 313 : 1
   Google Scholar
• Chattaway , F. D. and Ashworth , D. R. 1933 . J. Chem. Soc. , : 475
   Google Scholar
• Chattaway , F. D. and Parkes , G. D. 1935 . J. Org. Chem. , : 1005
   Google Scholar
• Chattaway , F. D. and Lye , R. J. 1932 . Proc. Roy. Soc. (London) , A135 : 282
   Google Scholar