Publication Cover
Synthetic Communications
An International Journal for Rapid Communication of Synthetic Organic Chemistry
Volume 26, 1996 - Issue 3
29
Views
15
CrossRef citations to date
0
Altmetric
Original Articles

A New Access to 2,3-Dihydro Imidazo [1,2-c] Pyrimidines

, , &
Pages 453-458 | Received 30 Jun 1995, Published online: 21 Aug 2006

References and Notes

  • Rahmouni , M. , Derdour , A. , Bazureau , J. P. and Hamelin , J. 1994 . Tetrahedron Lett. , 35 : 563 – 64 .
  • Rogers , R. and Neilson , D.G. 1961 . Chem. Rev. , 6 ( 1 ) : 179
  • Bader , H. 1965 . J. Org. Chem. , 30 : 707
  • Cado , F. , Di-Martino , J. L. , Jacquault , P. , Bazureau , J. P. and Hamelin , J. 1995 . Tetrahedron Lett. , submitted. 2-(cyanomethylene) imidazolidine 2a is synthetized in one step by condensation of ethylene diamine with the appropriate imino-ether12 in CH2Cl2 at 41°C during 48h, in 62% yield. For another application of this imino-ether, see also :
  • Jones , R. C.F. and Hirst , S. C. 1989 . Tetrahedron Lett. , 30 : 5361
  • Huang , Z. T. and Wang , M. X. 1994 . Heterocycles , 37 : 2
  • Rajappa , S. 1981 . Tetrahedron , 37 : 1453 – 80 .
  • Huang , Z. T. and Liu , Z. R. 1989 . Chem. Ber. , 122 : 95
  • Huang , Z. T. and Wang , M. X. 1993 . J. Chem. Soc., Perkin Trans. I , : 1085
  • Commarmot , R. , Didenot , R. and Gardais , J. F. 1986 . Chem. Abstr. , 105 : 17442e Fr. 2, 560, 529 (Cl. BO1J19/12), 06 Sep. 1985, Appl. 84/3, 496, 02 Mar 1984;
  • Dugosz , A. 1991 . Wiadomosci Chem. , 45 : 177 – 92 .
  • Lerestif , J. M. , Bazureau , J. P. and Hamelin , J. 1993 . Tetrahedron Lett. , 34 : 4639 – 42 .
  • Rechsteiner , B. , Texier-Boullet , F. and Hamelin , J. 1993 . Tetrahedron Lett. , 34 : 5071 – 74 .
  • Abdallah-El Ayoubi , S. , Texier-Boullet , F. and Hamelin , J. 1994 . Synthesis , : 258 – 60 .
  • Lerestif , JM. , Perrocheau , J. , Tonnard , F. , Bazureau , J. P. and Hamelin , J. 1995 . Tetrahedron , 5 ( 1 ) : 6757 – 74 .
  • Jolivet , S. , Di-Martino , J. L. , Jacquault , P. , Texier-Boullet and Hamelin , J. 1995 . Heteroatom. Chem. , in the press.
  • Dugosz , A. 1991 . Wiadomosci Chem. , 45 : 707 – 16 . and references cited therein.
  • Duschinsky , R. and Gabriel , T. F. Pat. USA . 3, 320, 256 . 1965 . Chem. Abstr. 1967 67 108666
  • Sté Prolabo, 54 rue Roger Salengro, 94126 - Fontenay sous Bois (France).
  • Initial attempts to separate the regioisomers 3b, 3b' by chromatography on silica or alumina gel were unsuccessful.
  • Mc Elvain , S. M. and Schroeder , T. F. 1949 . J. Amer. Chem. Soc. , 71 : 40 – 46 .

Reprints and Corporate Permissions

Please note: Selecting permissions does not provide access to the full text of the article, please see our help page How do I view content?

To request a reprint or corporate permissions for this article, please click on the relevant link below:

Academic Permissions

Please note: Selecting permissions does not provide access to the full text of the article, please see our help page How do I view content?

Obtain permissions instantly via Rightslink by clicking on the button below:

If you are unable to obtain permissions via Rightslink, please complete and submit this Permissions form. For more information, please visit our Permissions help page.