References and Notes
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- The acetylation of an unsbstituted indole 2-carboxylated ester, under Friedel-Crafts condition, was found to be dependent on the acidity of the carboxylic acid used; stronger acid derivatives tend to give the C-5 acylated product with respect to the acylation of C-3 position. Murakami Y. Tani M. Tanaka K. Yokoyama Y. Chem. Pharm. Bull. 1988 36 2023
- Using carboxylic acid/ trifluoroacetic anhydride/ poliphosphoric acid method, stronger acid derivatives tend to give lower yield of the acetylated product. Murakami Y. Tani Suzuki M. Sudoh K. Uesato M. M. Tanaka K. Yokoyama Y. Chem. Pharm. Bull. 1985 33 4707
- Dalla Croce , P. , Ferraccioli , R. and Ritieni , A. 1990 . Synthesis , : 212
- After the conclusion of our work, an alternative procedure for the selective bromination of the α carbon of ethyl 3-acetyl-1H-indole-2-carboxylate has been published. Suzuki H. Shinpo K. Yamazaki T. Niwa S. Yokoyama Y. Murakami Y. Heterocycles 1996 42 83