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Research Article

Diclofenac sodium loaded-cellulose acetate butyrate: Effect of processing variables on microparticles properties, drug release kinetics and ulcerogenic activity

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Pages 31-45 | Received 06 Mar 2007, Accepted 16 Oct 2007, Published online: 08 Oct 2008

References

  • Beyger JW, Nairn JG. Some factors affecting the miroencapsultion of pharmaceuticals with cellulose acetate phthalate. J Pharm Sci 1986; 75: 573–578
  • Biju SS, Saisivam S, Maria Gerald Rajan NS, Mishra PR. Dual coated erodible microparticles for modified release of diclofenac sodium. Eur J Pharm Biopharm 2004; 58: 61–67
  • Choi HS, Seo SA, Khang G, Rhee JM, Lee HB. Preparation and characterization of fentanyl-loaded PLGA microspheres: In vitro release profiles. Int J Pharm 2002; 234: 195–203
  • Çomoğlu T, Gönül N, Baykara T. Preparation and in vitro evaluation of modified release ketoprofen microsponges. Il Farmaco 2003; 58: 101–106
  • Cooke PM. Side-effects of non-steroidal anti-inflammatory drugs. Med J Aust 1988; 148: 248–251
  • Costa P, Lobo JMS. Modeling and comparison of dissolution profiles. Eur J Pharm Sci 2001; 13: 123–133
  • Daumesnil R. Multiparticulate oral drug delivery. Marcel Dekker, New York 1994; 457–474
  • Deasy PB. Microencapsulation and related drug processes. Marcel Dekker, New York 1988
  • Del Favero A. Side effects of drugs: Anti-inflammatory and antipyretic analgesics and drugs used in gout, Ann. 12, MNG Dukes, L Beeley. Elsevier, Amsterdam 1988; 80
  • Delgado M, Spanka C, Kerwin LD, Wentworth P, Jr, Janda KD. A tunable hydrogel for encapsulation and controlled release of bioactive proteins. Biomacromolecules 2002; 3: 262–271
  • Ebba F, Piccerelle P, Prinderre P, Opota D, Joachim J. Stress relaxation of granules as a function of different lubricants. Eur J Pharm Biopharm 2001; 52: 211–220
  • FDA Guidance for Industry. Dissolution testing of immediate release solid and dosage forms. Food and Drug Administration, Center for Drug Evaluation and Research, Rockville, MD 1997
  • Follonier N, Doelker E. Biopharmaceutical comparison of oral multiple-unit and single-unit sustained release dosage forms. STP Pharma Sci 1992; 2: 141–158
  • Gamberini MT, Skorupa LA, Souccar C, Lapa AJ. Inhibition of gastric-secretion by a water extract from Baccharis-Triptera. Mem Inst Oswaldo Cruz 1991; 86: 137–139
  • Gilman AG, Ralf TW, Nile AS. The pharmacological basis of therapeutics: Volume IB, 8th ed. Maxwell Publishing Corporation. 1991; 669
  • Gohel MC, Amin AF. Formulation design and optimization of modified-release microspheres of diclofenac sodium. Drug Dev Ind Pharm 1999; 25: 247–251
  • Hermann J, Bodmeier R. Biodegradable, somatostatin acetate containing microspheres prepared by various aqueous and non-aqueous solvent evaporation methods. Eur J Pharm Biopharm 1998; 45(1)75–82
  • Hickey A, Concessio N, Ort M, Platz R. Factors influencing the dispersion of drug powder as aerosols. Pharm Tech 1994, (August):58
  • Hörter D, Dressman JB. Influence of physicochemical properties of dissolution of drugs in the gastrointestinal tract. Adv Drug Del Rev 2001; 46: 75–87
  • Khang G, Lee JH, Lee JW, Cho JC, Lee HB. Preparation and characterization of PLGA microparticles for the sustained release of AZT. Korea Polym J 2000; 8: 80–88
  • Khopade AJ, Jain NK. Long-circulating multiple-emulsion system for improved delivery of an anticancer agent. Drug Del 1999; 6: 107–110
  • Kim CK, Kim SC, Shin HJ, Kim KM, Oh KH, Lee YB, Oh JJ. Preparation and characterization of cytarabine-loaded w/o/w multiple emulsions. Int J Pharm 1995; 124: 61–67
  • Korsmeyer RW, Gurny R, Doelker EM, Buri P, Peppas NA. Mechanism of solute release from porous hydrophilic polymers. Int J Pharm 1983; 15: 25–35
  • Laugel C, Baillet A, Youenang Piemi MP, Marty JP, Ferrier D. Oil-water-oil multiple emulsion for prolonged delivery of hydrocortisone after topical application: Comparison with simple emulsions. Int J Pharm 1998; 160: 109–117
  • Lee G. Spray-drying of proteins. Pharm Biotechnol 2002; 13: 135–158
  • Lee HB, Khang G, Cho JC, Rhee JM, Lee JS. Fentanyl-loaded PLGA microsphere for local anesthesia. Polymer Preprints 1999; 40: 288–289
  • Mandal TK. Evaluation of a novel phase separation technique for the encapsulation of water-soluble drug in biodegradable polymer. Drug Dev Ind Pharm 1998; 24: 623–639
  • Mateovi·-Rojnik T, Frlan R, Bogataj M, Bukovec P, Mrhar A. Effect of preparation temperature in solvent evaporation process on Eudragit RS microspheres properties. Chem Pharm Bull 2005; 53: 143–146
  • Moore JW, Flanner HH. Mathematical comparison of dissolution profiles. Pharm Tech 1996; 20: 64–74
  • Murakami H, Kobayashi M, Takeuchi H, Kawashima Y. Preparation of poly (Dl-lactibe-co-glycolide) nanoparticles by modified spontaneous emulsification solvent diffusion method. Int J Pharm 1999; 187: 143–152
  • Murakami H, Kobayashi M, Takeuchi H, Kawashima Y. Further application of a modified spontaneous emulsification solvent diffusion method to various types of PLGA and PLA polymer for preparation of nanoparticles. Powder Tech 2000; 107: 137–143
  • Obeidat WM, Price JC. Preparation and in vitro evaluation of propylthiouracil microspheres made of Eudragit RL100 and cellulose acetate butyrate polymers using the emulsion-solvent evaporation method. J Microencapsulation 2005; 22: 281–289
  • Perumal D. Microencapsulation of ibuprofen and Eudragit RS® 100 by the emulsion solvent diffusion technique. Int J Pharm 2001; 218: 1–11
  • Robert A. Cytoprotection by prostaglandins. Gastroenterology 1979; 77: 761–767
  • Röhm Pharma. Information sheet ‘Eudragit Polymethacrylate for Pharmaceutical Applications’. Röhm Pharma 1995
  • Sanghvi SP, Nairn JG. Phase diagram studies for microencapsulation of pharmaceutics using cellulose acetate trimellitate. J Pharm Sci 1991; 80: 394–398
  • Sansdrap P, Moës AJ. Influence of additives on the release profile of nifedipine from poly (DL-lactide-co-glycolide) microspheres. J Microencapsulation 1998; 15: 545–553
  • Sheu MT, Chou HL, Kao CC, Liu CH, Sokoloski TD. Dissolution of diclofenac sodium from matrix tablets. Int J Pharm 1992; 85: 57–63
  • Song M, Li N, Sun S, Tiedt LR, Liebenberg W, deVillirs MM. Effects of viscosity and concentration of wall former, emulsifier and pore-inducer on the properties of amoxicillin microcapsule prepared by emulsion solvent evaporation. IL Farmaco 2005; 60: 261–267
  • The United State Pharmacopoeia 23. United State Pharmacopeial Convention, Inc.,. USP, Rockville, MD 1995
  • Todd PA, Sorkin EM. Diclofenac sodium, a reappraisal of its pharmacodynamic and pharmacokinetic properties, and therapeutic efficacy. Drugs 1988; 35: 244–285
  • Urata T, Arimori K, Nakano H. Modification of release rate of cyclosporine a from poly (L-lactic acid) microspheres by fatty acid esters and in vivo evaluation of the microspheres. J Control Rel 1999; 58: 133–141
  • Wadke DA, Serajuddin ATM, Jacobson H. Preformulation testing. Pharmaceutical dosage forms-tablets, HA Lieberman, L Lachman, JB Schwartz. Marcel Dekker, New York 1989; 55
  • Zuleger S, Lippold BC. Polymer particle erosion controlling drug release: I. Factors influencing drug release and characterization of the release mechanism. Int J Pharm 2001; 217: 139–152

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