References
- Amidon, G. L., Lennernas, H., Shah, V. P., & Crison, J. R. (1995). A theoretical basis for a biopharmaceutical drug classification: the correlation of in vitro drug product, dissolution and in vivo bioavailability. Pharmaceutical Research, 12, 413–420., [PUBMED], [INFOTRIEVE], [CSA]
- Artursson, P., & Karlsson, J. (1991). Correlation between oral drug absorption in humans and apparent drug permeability coefficients in human intestinal epithelial Caco-2 cells. Biochemical and Biophysical Research Communications, 175, 880–885., [PUBMED], [INFOTRIEVE], [CSA], [CROSSREF]
- Bohets, H., Annaert, P., Mannens, G., Van Beijsterveldt, L., Anciaux, K., Verboven, P., Meudermans, W., & Lavrijsen, K. (2001). Strategies for absorption screening in drug discovery and development. Current Topics in Medicinal Chemistry, 5, 367–383., [CROSSREF]
- Camenish, G., Alsenz, J., Van DE Waterbeemd, H., & Folkers, G. (1998). Estimation of permeability by passive diffusion through Caco-2 Cell monolayers using the drug lipophilicity and molecular weight. European Journal of Pharmaceutical Sciences, 6, 313–319., [CROSSREF]
- Dressman, J. B., & Reppas, C. (2000). In vitro–in vivo correlations for lipophilic, poorly water soluble drugs. European Journal of Pharmaceutical Sciences, 11, S73–S80., [PUBMED], [INFOTRIEVE], [CROSSREF]
- Dressman, J. B., Amidon, G. L., Reppas, C., & Shah, V. P. (1998). Dissolution testing as a prognostic tool for oral drug absorption: immediate release dosage forms. Pharmaceutical Research, 15, 11–22., [PUBMED], [INFOTRIEVE], [CSA], [CROSSREF]
- Dunne, A., O'Hara, T., & Devane, J. (1999). A new approach to modelling the relationship between in vitro and in vivo drug dissolution/absorption. Statistics in Medicine, 18, 1865–1876., [PUBMED], [INFOTRIEVE], [CSA], [CROSSREF]
- Frick, A., Moller, H., & Wirbitzki, E. (1998). Biopharmaceutical characterization or oral immediate release drug products. In vitro/in vivo comparison of phenoxymethylpenicillin potassium, glimepride and levofloxacin. European Journal of Pharmaceutics and Biopharmaceutics, 46, 305–311., [PUBMED], [INFOTRIEVE], [CSA], [CROSSREF]
- Ginski, M. J., & Polli, J. E. (1999). Prediction of dissolution-absorption relationships from a dissolution/Caco-2 system. International Journal of Pharmaceutics, 177, 117–125., [PUBMED], [INFOTRIEVE], [CSA], [CROSSREF]
- Hilgers, A. R., Conradi, R. A., & Burton, P. S. (1990). Caco-2 cell monolayers as a model for drug transport across the intestinal mucosa. Pharmaceutical Research, 7, 902–910., [PUBMED], [INFOTRIEVE], [CROSSREF]
- Ingels, F., Destexhe, B., Oth, M., Van Den Mooter, G., & Augustuns, P. (2002). Simulated intestinal fluid as transport medium in the Caco-2 cell culture model. International Journal of Pharmaceutics, 232, 183–192., [PUBMED], [INFOTRIEVE], [CSA], [CROSSREF]
- Ogata, H., Shibazaki, T., Inoue, T., & Ejima, A. (2001). Comparative studies on eight dissolution methods using 21 commercial chloramphenicol tablet and a non disintegrating benzoic acid tablet. Journal of Pharmaceutical Sciences, 5, 367–383.
- Pather, S. I., Russel, I., Syce, J. A., & Neau, S. H. (1998). Sustained release theophylline tablets by direct compression. Part 1: Formulation and in vitro testing. International Journal of Pharmaceutics, 164, 1–10., [CROSSREF]
- Picker, K. M., & Bikane, F. (1998). Tablet formation and release from matrix tablets manufactured with cellulose acetate. International Journal of Pharmaceutics, 175, 147–164., [CROSSREF]
- Polli, J. E., Grison, J. R., & Amidon, G. L. (1996). Novel approach to the analysis of in vitro–in vivo relationships. Journal of Pharmaceutical Sciences, 85, 753–760., [PUBMED], [INFOTRIEVE], [CROSSREF]
- (2004). R: A Language and Environment for Statistical Computing. ISBN 3-900051-00-3. , http://www.R-project.org.
- Siewert, M. (1993). Perspectives of in vitro dissolution tests in establishing in vivo/in vitro correlations. European Journal of Drug Metabolism and Pharmacokinetics, 18, 7–18., [PUBMED], [INFOTRIEVE]
- Yamashita, S., Furubayashi, T., Kataoka, M., Sakane, T., Sezak, H., & Tokuda, H. (2000). Optimised conditions for prediction of intestinal drug permeability using Caco-2 cells. European Journal of Pharmaceutical Sciences, 10, 195–204., [PUBMED], [INFOTRIEVE], [CSA], [CROSSREF]
- Zerrouk, N., Chemtob, C., Arnaud, P., Toscani, S., & Dugue, J. (2001). In vitro and in vivo evaluation of carbamazepine-Peg 6000 solid dispersions. International Journal of Pharmaceutics, 28, 49–62., [CROSSREF]