3,980
Views
85
CrossRef citations to date
0
Altmetric
Research Article

The Effect of Selected Water-Soluble Excipients on the Dissolution of Paracetamol and Ibuprofen

, , &
Pages 515-525 | Published online: 26 Sep 2008

References

  • Altomare, E., Vendemiale, G., Benvenuti, C. & Andreatta, P. (1997). Bioavailability of a new effervescent tablet of ibuprofen in healthy volunteers.European Journal of Clinical Pharmacology, 52, 505–506., [PUBMED], [INFOTRIEVE], [CSA]
  • Ameer, B., Divoll, M., Abernethy, D. R., Greenblatt, D. J., & Shargel, L. (1983). Absolute and relative bioavailability of oral acetaminophen preparations.Journal of Pharmaceutical Sciences, 72, 955–958., [PUBMED], [INFOTRIEVE]
  • El-Sayed, Y.-M., Gouda, M. W., Al-Khamis, K. I., Al-Meshal, M. A., Al-Dhawailie, A. A., Al-Rayes, S., Bin-Salih, S. A., & Al-Rashood, K. A. (1995). Comparative bioavailability of two tablet formulations of ibuprofen.International Journal of Clinical Pharmacology and Therapeutics, 33, 294–298., [PUBMED], [INFOTRIEVE], [CSA]
  • Fairbrother, J. E. (1974). Acetaminophen. In: Florey, K. (Ed.). Analytical Profiles of Drug Substances, Vol. 3. New York: Academic Press, 1–109.
  • Gazzaniga, A., Gianesello, W., Stroppolo, F., & Vigano, L. (1988). Water Soluble Analgesic Ibuprofen Formulation—Contains L-Arginine and Sodium Bicarbonate to Reduce Gastric Irritation. G.B. Patent 2193039.
  • Geisslinger, G., Dietzel, K., Bezler, H., Nuernberg, B., & Brune, K. (1989). Therapeutically relevant differences in the pharmacokinetic and pharmaceutical behavior of ibuprofen lysinate as compared to ibuprofen acid.International Journal of Clinical Pharmacology and Therapeutics, 27, 324–328.
  • Heading, R. C., Nimmo, L. F., Prescott, L. F., & Tothill, P. (1973). The dependence of paracetamol absorption on the rate of gastric emptying.British Journal of Pharmacology, 47, 415–421., [PUBMED], [INFOTRIEVE]
  • Herzfeldt, C. D., & Kummel, R. (1983). Dissociation constants, solubilities and dissolution rates of some selected non-steroidal anti-inflammatories.Drug Development and Industrial Pharmacy, 9, 767–793.
  • Jamali, F., Singh, N., Pasutto, F. M., Russel, A. S., & Coutts, R. T. (1988). Pharmacokinetics of ibuprofen enantiomers in humans following oral administration of tablets with different absorption rate.Pharmaceutical Research, 5, 40–43., [PUBMED], [INFOTRIEVE], [CROSSREF]
  • Kelly, K., O-Mahony, B., Lindsay, B., Jones, T., Grattan, T. J., Rostami-Hodjegan, A., Stevens, H.N.E., & Wilson, C. G. (2003). Comparison of the rates of disintegration. gastric emptying, and drug absorption following administration of a new and a conventional paracetamol formulation, using gamma scintigraphy.Pharmaceutical Research, 20, 1668–1673., [PUBMED], [INFOTRIEVE], [CSA], [CROSSREF]
  • Levis, K. A., Lane, M. E., & Corrigan, O. E. (2003). Effect of buffer composition on the solubility and effective permeability coefficient of ibuprofen.International Journal of Pharmaceutics, 253, 49–59., [PUBMED], [INFOTRIEVE], [CSA], [CROSSREF]
  • Lund, W. (Ed.). (1994). The Pharmaceutical Codex. London: The Pharmaceutical Press, 908.
  • Macheras, P., Reppas, C., & Dressman, J. B. (1995). Biopharamaceutics of Orally Administered Drugs. London: Ellis Horwood, , pp. 35–87, 127.
  • Mahmud, A., & Li Wan Po, A. (1991). Investigation of the effect of additives on the dissolution rates of aspirin and paracetamol using a factorial design.Drug Development and Industrial Pharmacy, 17, 709–724.
  • Marriott, C. (2002). Rheology and the flow of liquids. In: Aulton, M. E. (Ed.). Pharmaceutics—the Science of Dosage Form Design (2nd ed.). London: Churchill Livingstone, pp. 17–19.
  • Moffat, A. C. (Ed.). (1986). Clarkes Isolation and Identification of Drugs. London: The Pharmaceutical Press, , pp. 677, 849.
  • Petring, O. U., Adelhoj, B., Ibsenm, M., & Poulsen, H. E. (1986). The relationship between gastric emptying of semisolids and paracetamol absorption.British Journal of Clinical Pharmacology, 22, 659–662., [PUBMED], [INFOTRIEVE]
  • Sack-Walter, I., Lucklow, V., Guserle, R., Weber, E. (1989). The relative bioavailability of paracetamol following administration of solid and liquid oral preparations and rectal dosage forms.Arzneimittel-Forschung, 39, 719–724.
  • Shaw, L. R., Irwin, W. J., Grattan, T. J., & Conway, B. R. (2002). The development of a modified dissolution method suitable for investigating powder mixtures.Drug Development and Industrial Pharmacy, 28, 1147–1153., [PUBMED], [INFOTRIEVE], [CSA], [CROSSREF]
  • Stead, J. A., Freeman, M., John, E. G., Ward, G. T., & Whiting, B. (1983). Ibuprofen tablets: dissolution and bioavailability studies.International Journal of Pharmaceutics, 14, 59–72., [CROSSREF]
  • Yu, L. X., Carlin, A. S., Amidon, G. L., Hussain, A. S. (2004). Feasibility studies of utilizing disk instrinsic dissolution rate to classify drugs.International Journal of Pharmaceutics, 270, 221–227., [PUBMED], [INFOTRIEVE], [CSA], [CROSSREF]

Reprints and Corporate Permissions

Please note: Selecting permissions does not provide access to the full text of the article, please see our help page How do I view content?

To request a reprint or corporate permissions for this article, please click on the relevant link below:

Academic Permissions

Please note: Selecting permissions does not provide access to the full text of the article, please see our help page How do I view content?

Obtain permissions instantly via Rightslink by clicking on the button below:

If you are unable to obtain permissions via Rightslink, please complete and submit this Permissions form. For more information, please visit our Permissions help page.