124
Views
7
CrossRef citations to date
0
Altmetric
Research Article

Supercritical Antisolvent Versus Coevaporation— Preparation and Characterization of Solid Dispersions

, , , , , & show all
Pages 975-983 | Published online: 26 Sep 2008

REFERENCES

  • Amidon G. L., Lunnernas H., Shah V. P., Crison J. R. A theoretical basis for a biopharmaceutic drug classification: the correlation of in vitro drug product dissolution and in vivo bioavailability. Pharm. Res. 1995; 12: 413–420
  • Badens E., Fargeot C., Bosc N., Veesler S., Teillaud E., Charbit G. Polymorph control of drug in supercritical CO2. Proceedings of the European Conference on Drug Delivery and Pharmaceutical Technology, Sevilla, May, 10–12, 2004; 46
  • Badens E., Teillaud E., Charbit G., Horváth G., Szokonya L., Bosc N., Majerik V. Solubility enhancement of a pharmaceutical ingredient using supercritical antisolvent and spray-freezing techniques. Proceedings of The 7th International Symposium on Supercritical Fluids, Orlando, May, 1–4, 2005
  • Beach S., Lathan D., Sidgwick C., Hanna M., York P. Control of the physical form of Salmeterol Xinafoate. Org. Proc. Res. Dev. 1999; 3: 370–376
  • Bitz C., Doelker E. Influence of the preparation method on residual solvents in biodegradable microspheres. Int. J. Pharm. 1996; 131: 171–181
  • Bristow S., Shekunov T., Shekunov B. Yu., York P. Analysis of the supersaturation and precipitation process with supercritical CO2. J. Supercrit. Fluids 2001; 21: 257–271
  • Cassidy O. E., Haskayne L., Rowley G. Electrostatic charge and dissolution of surface modified phenylbutazone. Eur. J. Pharm. Sci. 1998; 6: S23
  • Charbit G., Badens E., Boutin O. Methods of particle production. Supercritical Fluid Technology for Drug Product Development, Drugs and Pharmaceutical Sciences Vol. 138, P. York, U. B. Kompella, B. Y. Shekunov. Marcel Dekker, Inc, New York 2004; 159–212
  • Coates J. Interpretation of Infrared Spectra, A Practical Approach. Encyclopedia of Analytical Chemistry, R. A. Meyers. John Wiley & Sons Ltd, Chichester 2000; 10815–10837
  • Delneuville I., Dechesne J. P., Delattre L. Preparation and study of the characteristics of dithranol:polyvinylpyrrolidone coevaporates. Int. J. Pharm. 1998; 168: 109–118
  • Fargeot C., Badens E., Charbit G., Bosc N., Teillaud E., Veesler S. Cristallisation d'un prinicipe actif: comparaison des méthodes par voie liquide et supercritique. Proceedings of The Cristal2, Toulouse, Novembre, 12–13, 2003; 55–60
  • FDA. International Conference on Harmonisation, ICH Guidance on Impurities: Residual Solvents, Federal Register. 1997; 62: 67377–67388
  • FDA. (2002). Draft—Guidance for Industry: Bioavailability and Bioequivalence Studies for Orally Administered Drug Products. US Department of Health and Human Services, Food and Drug Administration, Center for Drug Evaluation and Research (CDER).
  • Forster A., Hempenstall J., Rades T. Investigation of drug / polymer interaction in glass solutions prepared by melt extrusion. Int. J. Vib. Spec. 2001; 5: 6, www.ijvs.com
  • Jannin V., Pochard E., Chambin O. Influence of poloxamers on the dissolution performance and stability of controlled-release formulations containing Precirol® ATO 5. Int. J. Pharm. 2006; 309: 6–15
  • Kaczmarek H., Szalla A., Kaminska A. Study of poly(acrylic acid)-poly(vinylpyrrolidone) complexes and their photostability. Polymer 2001; 42: 6057–6069
  • Kim E. -J., Chun M. -K., Jang J. -S., Lee I. -H., Lee K. -R., Choi H.-K. Preparation of a solid dispersion of felodipine using a solvent wetting method. Eur. J. Pharm. Biopharm. 2006; 64: 200–205
  • Korsmeyer R. W., Gurny R., Doelker E. M., Buri P., Peppas N. A. Mechanism of solute release from porous hydrophilic polymers. Int. J. Pharm. 1983; 15: 25–35
  • Leuner C., Dressman J. Improving drug solubility for oral delivery using solid dispersions. Eur. J. Pharm. 2000; 50: 47–60
  • Lochard H., Sauceau M., Freiss B. Method for the preparation of molecular complexes. World Patent WO 04096284 A1, 2004
  • Majerik V., Charbit G., Badens E., Horváth G., Szokonya L., Bosc N., Teillaud E. Bioavailability enhancement of an active substance by supercritical antisolvent precipitation. J. Supercrit. Fluids 2007; 40: 101–110
  • Majerik V., Horváth G., Charbit G., Badens E., Szokonya L., Bosc N., Teillaud E. Novel particle engineering techniques in drug delivery: review of formulations using supercritical fluids and liquefied gases. Hung. J. Ind. Chem. 2004; 32: 41–56
  • Miranda S., Yaeger S. Homing in on the best size reduction method. Chem. Eng. 1998; 105: 102–110
  • Pasquali I., Bettini R., Giordano F. Solid-state chemistry and particle engineering with supercritical fluids in pharmaceutics. Eur. J. Pharm. Sci. 2006; 27: 299–310
  • Perrut M., Jung J., Leboeuf F., Fabing I. Method for making very fine particles consisting of a principle inserted in a host molecule. World Patent WO 0232462, 2002
  • Reverchon E. Supercritical antisolvent precipitation of micro- and nano-particles. J. Supercrit. Fluids 1999; 15: 1–21
  • Reverchon E., Della Porta G., De Rosa I., Subra P., Letourneur D. Supercritical antisolvent micronization of some biopolymers. J. Supercrit. Fluids 2000; 18: 239–245
  • Rogers T. L., Johnston K. P., Williams R. O., III. Solution-based particle formation of pharmaceutical powders by supercritical or compressed fluid CO2 and cryogenic spray-freezing technologies. Drug Dev. Ind. Pharm. 2001; 27: 1003–1015
  • Ruchatz F., Kleinebudde P., Müller B. W. Residual solvents in biodegradable microparticles. Influence of process parameters on the residual solvent in microparticles produced by the Aerosol Solvent Extraction System (ASES) process. Int. J. Pharm. Sci. 1997; 86: 101–105
  • Sethia S., Squillante E. Solid dispersions: revival with greater possibilities and applications in oral drug delivery. Crit. Rev. Ther. Drug Carrier Syst. 2003; 20: 215–247
  • Sethia S., Squillante E. Solid dispersions of carbamazepine in PVP K30 by conventional solvent evaporation and supercritical methods. Int. J. Pharm. 2004; 272: 1–10
  • Szente L., Szejtli J. Highly soluble cyclodextrin derivatives: chemistry, properties, and trends in development. Adv. Drug Delivery Rev. 1999; 36: 17–28
  • Van den Mooter G., Augustijns P., Blaton N., Kinget R. Physico-chemical characterization of solid dispersions of temazepam with polyethylene glycol 6000 and PVP K30. Int. J. Pharm. 1998; 164: 67–80
  • Van Nijlen T., Brennan K., Van den Mooter G., Blaton N., Kinget R., Augustijns P. Improvement of the dissolution rate of artemisinin by means of supercritical fluid technology and solid dispersions. Int. J. Pharm. 2003; 254: 173–181
  • Yong C. S., Lee M.-K., Park Y.-J., Kong K.-H., Xuan J. J., Kim J.-H., Kim J.-A., Lyoo W. S., Han S. S., Rhee J.-D., Kim J. O., Yang C. H., Kim C.-K., Choi H.-G. Enhanced oral bioavailability of ibuprofen in rats by poloxamer gel using poloxamer 188 and menthol. Drug. Dev. Ind. Pharm. 2005; 31: 615–622

Reprints and Corporate Permissions

Please note: Selecting permissions does not provide access to the full text of the article, please see our help page How do I view content?

To request a reprint or corporate permissions for this article, please click on the relevant link below:

Academic Permissions

Please note: Selecting permissions does not provide access to the full text of the article, please see our help page How do I view content?

Obtain permissions instantly via Rightslink by clicking on the button below:

If you are unable to obtain permissions via Rightslink, please complete and submit this Permissions form. For more information, please visit our Permissions help page.