432
Views
18
CrossRef citations to date
0
Altmetric
Research Article

Raft-Forming Agents: Antireflux Formulations

&
Pages 1350-1361 | Published online: 25 Sep 2008

REFERENCES

  • Beekman S. M. Preparation and properties of new gastric antacids. J. Am. Pharm. Assoc. Sci. Ed. 1960; 49: 191–200
  • Brooks W. J. Rafting antacid formulation. US Patent 5,360,793, 1994, November 1, 1994
  • Chavkin L. Dry, water-foamable pharmaceutical compositions. US Patent 4,613,497, 1986, September 23, 1986
  • Davies N. M., Farr S. J., Kellaway I. W., Taylor G., Thomas M. A comparison of the gastric retention of alginate containing tablet formulations with and without the inclusion of excipient calcium ions. Int. J. Pharm. 1994; 105: 97–101
  • Dettmar P. W., Dickson A. P., Hampson C. F., Jolliffe G. I. Compositions for treatment of disorders of the oesophagus. US Patent 6,610,667, 2003, August 26, 2003
  • Dettmar P. W., Little S. L., Baxter T. The Effect of omeprazole pre-treatment on rafts formed by reflux suppressant tablets containing alginate. J. Int. Med. Res. 2005; 33: 301–308
  • Eccleston G., Paterson R. Gastric raft composition. US Patent Application 20050063980, 2005, March 24 2005
  • Field F. P. Composition and method for treatment of gastrointestinal distress. US Patent 5,681,827, 1997, October 28, 1997
  • Foldager J., Toftkjor H., Kjornos K. Antacid composition. US Patent 5,068,109, 1991, November 26, 1991
  • Fuchs C. Antacids, their function, formulation, and evaluation. Drug Cosmetic Ind. 1949; 64: 692–773
  • Gayst S., Maguire M. J. Pharmaceutical formulation of guar gum. US Patent 4,315,918, 1982, February 16, 1982
  • Geoffrey C. W., Henry I. J. Gastroesophageal reflux disease. Am. J. Pharm. Edu. 2003; 66: 148–152
  • Goodall J. S., Orwin J. M., Imrie M. J. A combined pH and X-ray study of liquid alginate/antacid formulation using a novel X-ray contrast medium. Acta Therapeutica 1977; 3: 141–153
  • Grant G. T, Morris E. R, Rees D. A, Smith P. J. C., Thom D. Biological interactions between polysaccharides and divalent cations: the egg box model. FEBS Lett. 1973; 32: 195–198
  • Gregory S., Kelly N. D. Hydrochloric Acid: Physiological Functions and Clinical Implications. Alt. Med. Rev. 1997; 2(2)116–127
  • Hampson F. C., Farndale A., Strugala V., Sykes J., Dettmar P. W. Alginate rafts and their characterization. Int. J. Pharm. 2005; 294: 137–147
  • Havelund T., Aalykke C. The efficacy of a pectin-based raft-forming anti-reflux agent in endoscopy-negative reflux disease. Scand. J. Gastroenterol. 1997a; 32: 773–777
  • Havelund T., Aalykke C., Rasmussen L. Efficacy of a pectin-based anti-reflux agent on acid reflux and recurrence of symptoms and oesophagitis in gastro-oesophageal reflux disease. Eur. J. Gastroenterol. Hepatol. 1997b; 9(5)509–514
  • Hill E. A., Wade G. Investigation into the use of viscometry for in vitro characterization of the raft forming properties of tablets containing alginic acid and antacid components. Drug Dev. Ind. Pharm. 1993; 19(5)1931–1937
  • Holbert J. M., Noble N., Grote I. W. Study of antacid buffers, time factor in neutralization of gastric acidity. J. Am. Pharm. Assoc. Sci. Ed. 1947; 36: 149–151
  • Hoogerwerf W. A., Pasricha P. J. Goodman and Gilman's, The Pharmacological Basis of Therapeutics10th edition, International. 1005–1017
  • Irvine E. J. Quality of life assessment in gastro-oesophageal reflux disease. Gut 2004; 53(4)35–39
  • Jenkins J. R. F., Hardy J. G., Wilson C. G. Monitoring antacid preparations in the stomach using gamma scintigraphy. Int. J. Pharm. 1983; 14: 143–148
  • Johnson F. A., Craig D. Q. M., Mercer A. D., Chauhan S. The effects of alginate molecular structure and formulation variables on the physical characteristics of alginate raft systems. Int. J. Pharm. 1997; 159: 35–42
  • Johnson L. F., DeMeester T. R. Evaluation of elevation of the head of the bed, bethanechol, and antacid form tablets on gastroesophageal reflux. Dig. Dis. Sci. 1981; 26(8)673–680
  • Jolliffe I. G., Hampson F. C., Campbell R., Dettmar P. W. In vitro reflux resistance in alginate rafts. Gut 2001; 48: A26
  • Jung A. D. Gastroesophageal reflux in infants and children. Am. Fam. Physician. 2001; 64(11)1853–1860
  • Kulig M, Leodolter A, Vieth M, et al. Quality of life in relation to symptoms in patients with gastro-oesophageal reflux disease – an analysis based on the ProGERD initiative. Aliment. Pharmacol. Ther. 2003; 18: 767–776
  • Lu C. L., Lang H. C., Chang F. Y., Chan T. J., Chan C. Y., Luo J. C., Lee S. D. Social and medical impact, sleep quality and the pharmaceutical costs of heartburn in Taiwan. Aliment. Pharmacol. Ther. 2005; 22: 739–747
  • Malmud L. S., Charles N. D., Littlefield J. The mode of action of alginic acid compound in the reduction of gastroesophageal reflux. J. Nuc. Med. 1979; 20(10)1023–1028
  • Mandel K. G., Daggy B. P., Jacoby H. I. Review article: alginate-raft formulations in the treatment of heartburn and acid reflux. Aliment. Pharmacol. Ther. 2000; 1: 669–690
  • Mandlekar S. V., Marathe S. S., Devarajan P. V. A novel raft-forming antacid suspension using a natural dietary fibre. Int. J. Pharm. 1997; 148: 117–121
  • May H. A., Wilson C. G., Hardy J. G. Monitoring radiolabeled antacid preparations in the stomach. Int. J. Pharm. 1984; 19: 169–176
  • Moss H. A., Washington N., Greaves J. L., Wilson C. L. Anti-reflux agents, stratification or floatation?. Eur. J. Gastroenterol. Hepatol. 1990; 2: 45–51
  • Nebel O. T., Fornes M. F., Castell D. O. Symptomatic gastroesophageal reflux: Incidence and precipitating factors. Am. J. Dig. Dis. 1976; 21: 953–956
  • Richter J. E. Severe reflux esophagitis. Gastrointest. Endosc. Clin. North Am. 1994; 4: 677–698
  • Rossett N. E., Rice M. L. An in vitro evaluation of the efficacy of more frequently used antacids with particular attention to tablets. Gastroenterology 1954; 26(3)490–495
  • Sandler R. S., Everhart J. E., Donowitz M., et al. The burden of selected digestive diseases in the United States. Gastroenterology 2002; 122: 1500–1511
  • Scott M., Gelhot A. R. Gastroesophageal Reflux Disease: Diagnosis and Management. Am. Fam. Physician. 1999; 59(5)1161
  • Smyth R. D., Herczeg T., Wheatley T. A., House W., Reavey-Cantwell N. H. Correlation of in vitro and in vivo methodology for evaluation of antacids. J. Pharm. Sci. 1976; 65: 1045–1047
  • US Patent 2,774,710 issued to Thomson, K, December 1956 (crossreference obtained from US Patent 5,360,793).
  • US Patent 5,112,813 issued to Rhone, R., P, May 12, 1992 (crossreference obtained from US Patent 5,360,793).
  • Vatier J., Celice-Pinguad C., Farinotti. A computerized artificial stomach model to assess sodium alginate-induced pH gradient. Int. J. Pharm. 1998; 163: 225–229
  • Washington N., Washington C., Wilson C. G., Davis S. S. Effect of aluminium hydroxide on ‘raft forming’ antacids. J. Pharm. Pharmacol. 1985a; 37: 13P
  • Washington N., Washington C., Wilson C. G., Davis S. S. The effect of inclusion of aluminum hydroxide in alginate-containing raft-forming antacids. Int. J. Pharm. 1986; 28: 139–143
  • Washington N., Wilson C. G., Davis S. S. Evaluation of ‘raft-forming’ antacid neutralizing capacity : in vitro and in vivo correlations. Int. J. Pharm. 1985b; 27: 279–286
  • Washington N., Wilson C. G., Greaves L., Danneskiold-Samosøe P. An investigation into the floating behaviour of a pectin-Containing anti-reflux Formulation (FF5005) by means of gamma scintigraphy. Scand. J. Gastroenterol. 1988; 23: 920–924
  • Washington N., Wilson C. G., Williams D. L., Robertson C. An investigation into the effect of cimetidine pre-treatment on raft formation of an anti-reflux agent. Aliment. Pharmacol. Ther. 1993; 7: 553–559
  • Waterhouse E. T., Washington C., Washington N. An investigation into the efficacy of the pectin based anti-reflux formulation-Aflurax. Int. J. Pharm. 2000; 209: 79–85
  • http://class.fst.ohio-state.edu/FST605/lectures/lect20.html Web ref
  • http://www.cybercolloids.net/library/carob/structure.php Web ref
  • http://www.cybercolloids.net/library/carrageenan/structure.php Web ref
  • http://www.cybercolloids.net/library/pectin/structure.php Web ref
  • http://www.cybercolloids.net/library/xanthan/structure.php Web ref
  • http://www.foodproductdesign.com/archive/1999/1299ap.html Web ref
  • http://www.lsbu.ac.uk/water/hyalg.html Web ref

Reprints and Corporate Permissions

Please note: Selecting permissions does not provide access to the full text of the article, please see our help page How do I view content?

To request a reprint or corporate permissions for this article, please click on the relevant link below:

Academic Permissions

Please note: Selecting permissions does not provide access to the full text of the article, please see our help page How do I view content?

Obtain permissions instantly via Rightslink by clicking on the button below:

If you are unable to obtain permissions via Rightslink, please complete and submit this Permissions form. For more information, please visit our Permissions help page.