165
Views
3
CrossRef citations to date
0
Altmetric
Research Article

Development and Evaluation of a pH-Dependent Sustained Release Tablet for Irritable Bowel Syndrome

, , , , &
Pages 57-64 | Published online: 01 Jan 2009

REFERENCES

  • S. Appel, A. Kumle, M. Hubert, and T. Duvauchelle. (1997). First pharmacokinetic-pharmacodynamic study in humans with a selective 5-hydroxytryptamine4 receptor agonist. J. Clin. Pharmacol 37:229–237.
  • S. Appel-Dingemanse, Y. Hirschberg, S. Osborne, F. Pommier, and J. McLeod. (2001a). Multiple-dose pharmacokinetics confirm no accumulation and dose proportionality of the novel promotile drug tegaserod (HTF 919). Eur. J. Clin. Pharmacol 56:889–891.
  • S. Appel-Dingemanse, A. Horowitz, J. Campestrini, S. Osborne, and J. McLeod. (2001b). The pharmacokinetics of the novel promotile drug, tegaserod, are similar in healthy subjects-male and female, elderly and young. Aliment. Pharmacol. Ther 15:937–944.
  • S. Appel-Dingemanse, M. O. Lemarechal, A. Kumle, M. Hubert, and E. Legangneux. (1999). Integrated modelling of the clinical pharmacokinetics of SDZ HTF 919, a novel selective 5-HT4 receptor agonist, following oral and intravenous administration. Br. J. Clin. Pharmacol 47:483–491.
  • M. Ashford, and T. Fell. (1994). Targeting drugs to the colon: delivery systems for oral administration. J. Drug Target. 2:241–258.
  • M. E. Aulton, and A. M. Twitchell. (1995). Solution properties and atomization in film coating. InJ. E. Hogan, M. E. Aulton. (Eds.), Pharmaceutical coating technology ( pp. 64–117). London: Taylor & Francis.
  • P. Costa, and J. M. Sousa Lobo. (2001). Modeling and comparison of dissolution profiles. Eur. J. Pharm. Sci. 13:123–133.
  • J. T. Fell, and E. Efentakis. (1979). Contact angle determinations on pharmaceutical powders: A comparison of two methods. Int. J. Pharm. 4:153–157.
  • M. A. Frohoff-Hulsmann, A. Schmitz, and B. C. Lippold. (1999). Aqueous ethyl cellulose dispersions containing plasticizer of different water solubility and hydroxypropyl methyl cellulose as coating material for diffusion pellets: I. Drug release rates from coated pellets. Int. J. Pharm. 177:69–82.
  • M. Fox, D. Menne, B. Stutz, M. Fried, and W. Schwizer. (2006). The effects of tegaserod on oesophageal function and bolus transport in healthy volunteers: studies using concurrent high-resolution manometry and videofluoroscopy. Aliment. Pharmacol. Ther. 24:1017–1027.
  • J. Gutiérrez-Rocca, and J. W. McGinity. (1994). Influence of water soluble and insoluble plasticizer on the physical and mechanical properties of acrylic resin copolymers. Int. J. Pharm. 103:293–301.
  • S. K. Hadley, and S. M. Gaarder. (2005). Treatment of irritable bowel syndrome. Am. Fam. Phys. 72:2501–2506.
  • J. E. Hogan. (Ed.). (1995). Film-coating materials and their properties. Pharmaceutical coating technology ( pp. 6–52). London: Taylor & Francis.
  • A. P. Hungin, P. J. Whorwell, J. Tack, and F. Mearin. (2003). The prevalence, patterns and impact of irritable bowel syndrome: An international survey of 40,000 subjects. Aliment. Pharmacol. Ther. 17:643–650.
  • C. F. Lerk, A. J. Schoonen, and J. T. Fell. (1976). Contact angles and wetting of pharmaceutical powders. J. Pharm. Sci. 65:843–847.
  • I. N. Levine. (1995). Physical chemistry (4th ed.). New York: McGraw-Hill.
  • Organization for Economic Co-operation and Development. (2006). Guidelines for the testing of chemicals, partition coefficient (1-octanol/water): Slow-stirring method. http//www.sourceoecd.org/vl=12691240/cl=13/nw=1rpsv/cgibin/fulltextew.pl?prpsv=/ij/oecdjournals/1607310x/v1n1/s22/p1.idx.
  • A. Rivkin. (2003). Tegaserod maleate in the treatment of irritable bowel syndrome: A clinical review. Clin. Ther. 25:1952–1974.
  • V. P. Shah, Y. Tsong, P. Sathe, and J. P. Liu. (1998). In vitro dissolution profile comparison-statistics and analysis of the similarity factor, f2. Pharm. Res. 15:889–896.
  • S. K. Swan, H. Zhou, A. Horowitz, L. Alladina, M. Hubert, S. Appel-Dingemanse, S. Osborne, L. Lambrecht, and J. F. McLeod. (2003). Tegaserod pharmacokinetics are similar in patients with severe renal insufficiency and in healthy subjects. J. Clin. Pharmacol. 43:359–364.
  • N. J. Talley, M. Camilleri, D. Burton, G. Thomforde, K. Koch, M. J. Rucker, J. Peterson, A. R. Zinsmeister, and D. L. Earnest. (2006). Double-blind, randomized, placebo-controlled study to evaluate the effects of tegaserod on gastric motor, sensory and myoelectric function in healthy volunteers. Aliment. Pharmacol. Ther. 24:859–867.
  • U.S. Food and Drug Administration. (1997). Guidance for industry, extended release oral dosage forms: Development, evaluation, and application of in vitro/in vivo correlations. http://www.fda.gov/cder/guidance/1306fnl.pdf.
  • H. Zhou, S. Khalilieh, H. Lau, M. Guerret, S. Osborne, L. Alladina, A. L. Laurent, and J. F. McLeod. (1999). Effect of meal timing not critical for the pharmacokinetics of tegaserod (HTF 919). J. Clin. Pharmacol. 39:911–919.

Reprints and Corporate Permissions

Please note: Selecting permissions does not provide access to the full text of the article, please see our help page How do I view content?

To request a reprint or corporate permissions for this article, please click on the relevant link below:

Academic Permissions

Please note: Selecting permissions does not provide access to the full text of the article, please see our help page How do I view content?

Obtain permissions instantly via Rightslink by clicking on the button below:

If you are unable to obtain permissions via Rightslink, please complete and submit this Permissions form. For more information, please visit our Permissions help page.