204
Views
43
CrossRef citations to date
0
Altmetric
Original Article

Selected polysaccharides at comparison for their mucoadhesiveness and effect on precorneal residence of different drugs in the rabbit model

, , &
Pages 941-949 | Received 26 Aug 2008, Accepted 26 Dec 2008, Published online: 19 May 2009

References

  • Chrai SS, Robinson JR. (1974). Ocular evaluation of methylcellulose vehicle in albino rabbits. J Pharm Sci, 63:1218–23.
  • Lee VHL, Robinson JR. (1986). Review: Topical ocular drug delivery: Recent developments and future challenges. J Ocul Pharmacol, 2:67–108.
  • Patton TF, Robinson JR. (1975). Ocular evaluation of polyvinylalcohol vehicle in rabbits. J Pharm Sci, 64:1312–6.
  • Saettone MF, Giannaccini B, Ravecca S, La Marca F, Tota G. (1984). Polymer effects on ocular bioavailability—the influence of different liquid vehicles on the mydriatic response of tropicamide in humans and rabbits. Int J Pharm, 20:187–202.
  • Saettone MF, Giannaccini B, Teneggi A, Savigni P, Tellini N. (1982). Vehicle effects on ophthalmic bioavailability: The influence of different polymers on the activity of pilocarpine in rabbit and man. J Pharm Pharmacol, 34:464–6.
  • Trueblood JH, Rossomondo RM, Wilson LA, Carlton WH. (1975). Corneal contact times of ophthalmic vehicles. Evaluation by microscintigraphy. Arch Ophthalmol, 93:127–30.
  • Hui H-W, Robinson JR. (1985). Ocular drug delivery of progesterone using a bioadhesive polymer. Int J Pharm, 26:203–13.
  • Winfield AJ, Jessiman D, Williams A, Esakowitz L. (1990). A study of the causes of non-compliance by patients prescribed eyedrops. Br J Ophthalmol, 74:477–80.
  • Burgalassi S, Nicosia N, Monti D, Falcone G, Boldrini E, Chetoni P. (2007). Larch arabinogalactan for dry eye protection and treatment of corneal lesions: Investigation in rabbits. J Ocul Pharmacol Ther, 23:541–9.
  • Saettone MF, Burgalassi S, Boldrini P, Bianchini G. (1997). Ophthalmic solutions viscosified with tamarind seed polysaccharide. International patent application PCT/IT97/00026, International Publication number WO 97/28787.
  • Gregory S, Kelly ND. (1999). Larch arabinogalactan: Clinical relevance of a novel immune-enhancing polysaccharide. Altern Med Rev, 4:96–103.
  • Lee JW, Park JH, Robinson JR. (2000). Bioadhesive-based dosage forms: The next generation. J Pharm Sci, 89:850–66.
  • Mikos AG, Peppas NA. (1986). Systems for controlled release of drugs: V. Bioadhesive systems. S. T. P. Pharma Sci, 2:705–16.
  • Hassan EE, Gallo JM. (1990). A simple rheological method for the in vitro assessment of mucin-polymer bioadhesive bond strength. Pharm Res, 7:491–5.
  • Hägerström H, Edsman K. (2003). Limitations of the rheological mucoadhesion method: The effect of the choice of conditions and the rheological synergism parameter. Eur J Pharm Sci, 18:349–57.
  • Bottari F, Di Colo G, Nannipieri E, Saettone MF, Serafini MF. (1975). Evaluation of a dynamic permeation technique for studying drug–macromolecule interaction. J Pharm Sci, 64:946–9.
  • Greaves JL, Wilson CG. (1993). Treatment of diseases of the eye with mucoadhesive delivery systems. Adv Drug Deliv Rev, 11:349–83.
  • Saettone MF, Giannaccini B, Barattini F, Tellini N. (1982). The validity of rabbits for investigations on ophthalmic vehicles: A comparison of four different vehicles containing tropicamide in humans and rabbits. Pharm Acta Helv, 57:47–55.
  • Zaki I, Fitzgerald P, Hardy JG, Wilson CG. (1986). A comparison of the effects of viscosity on the precorneal residence of solutions in rabbit and man. J Pharm Pharmacol, 38:463–6.
  • Clausen AE, Bernkop-Schnürch A. (2000). In vitro evaluation of the permeation-enhancing effect of thiolated polycarbophil. J Pharm Sci, 89:1253–61.
  • Clausen AE, Bernkop-Schnürch A. (2001). Thiolated carboxymethylcellulose: In vitro evaluation of its permeation-enhancing effect on peptide drugs. Eur J Pharm Biopharm, 51:25–32.
  • Weast RC, ed. (1975). Handbook of chemistry and physics. 56th ed. Cleveland, (OH): CRC Press, F-49.
  • Uccello-Barretta G, Nazzi S, Balzano F, Di Colo G, Zambito Y, Zaino C, (2008). Enhanced affinity of ketotifen toward tamarind seed polysaccharide in comparison with hydroxyethylcellulose and hyaluronic acid: A nuclear magnetic resonance investigation. Bioorg Med Chem, 16:7371–6.

Reprints and Corporate Permissions

Please note: Selecting permissions does not provide access to the full text of the article, please see our help page How do I view content?

To request a reprint or corporate permissions for this article, please click on the relevant link below:

Academic Permissions

Please note: Selecting permissions does not provide access to the full text of the article, please see our help page How do I view content?

Obtain permissions instantly via Rightslink by clicking on the button below:

If you are unable to obtain permissions via Rightslink, please complete and submit this Permissions form. For more information, please visit our Permissions help page.