Preparation and characterization of spray-dried mucoadhesive microspheres of aceclofenac

References

• Zgoulli S, Grek V, Barre G, Goffinet G, Thonart P, Zinner S. (1999). Microencapsulation of erythromycin using a spray-drying technique. J Microencapsul, 16:565–71.
   PubMed Web of Science ®Google Scholar
• Desai K, Park H. (2005). Preparation and characterization of drug-loaded chitosan–tripolyphosphate microspheres by spray drying. Drug Dev Res, 64:114–28.
   Web of Science ®Google Scholar
• Parfitt K. (1996). Analgesics anti-inflammatory and antipyretics. In: Reynolds JEF, ed. Martindale: The complete drug reference. London: Royal pharmaceutical society, 2–12.
   Google Scholar
• Brogden R, Wiseman L. (1996). Aceclofenac: A review of its pharmacodynamic properties and therapeutic potential in the treatment of rheumatic disorders and in pain management. Drugs, 52(1):113–24.
   PubMed Web of Science ®Google Scholar
• Mutalik S, Naha A, Usha A, Ranjith A, Musmade P, Manoj K, al et. (2007). Preparation, in vitro, preclinical and clinical evaluations of once daily sustained release tablets of aceclofenac. Arch Pharm Res, 30(2):222–34.
   PubMed Web of Science ®Google Scholar
• Dashora K, Saraf S, Saraf S. (2006). Effect of processing variables on microparticulate system of aceclofenac. Pak J Pharm Sci, 19(1):1–6.
   PubMedGoogle Scholar
• Lee J, Lee Y, Kim J, Yoon M, Choi Y. (1995). Formulation of microemulsion systems for transdermal delivery of aceclofenac. Arch Pharm Res, 28(9):1097–102.
   Web of Science ®Google Scholar
• Burjak M, Bogataj M, Velnar M, Grabnar I, Mrhar A. (2001). The study of drug release from microspheres adhered on pig vesical mucosa. Int J Pharm, 224:123–30.
   PubMed Web of Science ®Google Scholar
• Harikarnpakdee S, Lipipun V, Sutanthavibul RG. (2006). Spray dried mucoadhesive microspheres: Preparation and transport through nasal cell monolayer. AAPS PharmSciTech, 7(1):E1–E10.
   PubMed Web of Science ®Google Scholar
• Mi F, Sung H, Shyu S. (2001). Release of indomethacin from a novel chitosan microsphere prepared by a naturally occurring crosslinker: Examination of crosslinking and polycation–anionic drug interaction. J Appl Polym Sci, 81:1700–11.
   Web of Science ®Google Scholar
• Arica B, Calis S, Atilla P, Durlu NT, Cakar N, Kash S, al et. (2005). In vitro and in vivo studies of ibuprofen-loaded biodegradable alginate beads. J Microencapsul, 22(2):153–65.
   PubMed Web of Science ®Google Scholar
• Acikgoz M, Kas HS, Hascelik Z, Milli U, Hincal AA. (1995). Chitosan microspheres of diclofenac sodium. II: In vitro and in vivo evaluation. Pharmazie, 50:275–7.
   PubMed Web of Science ®Google Scholar
• Calis S, Arica B, Atilla P, Durlu T, Cakar N, Hincal AA. (2003). Effect of ibuprofen and ibuprofen incorporated biodegradable alginate beads on gastric and duodenal mucosa (a comparative histological study). Controlled Release Society 30th Annual Meeting Proceedings, 19–23, 495.July
   Google Scholar
• Chowdhary KPR, Rao YM. (2003). Preparation and evaluation of mucoadhesive microcapsules of indomethacin. Saudi Pharm J, 11(3):97–103.
   Google Scholar
• Sakagami M, Kinoshita W, Sakon K, Sato J, Makino Y. (2002). Mucoadhesive beclomethasone microspheres for powder inhalation: Their pharmacokinetics and pharmacodynamics evaluation. J Control Release, 80:207–18.
   PubMed Web of Science ®Google Scholar
• Filipovic J, Becirevic M, Skalko N, Jalsenjak I. (1996). Chitosan microspheres of nifedipine and nifedipine–cyclodextrin inclusion complexes. Int J Pharm, 135:183–90.
   Web of Science ®Google Scholar
• Jain S, Chourasia M, Jain A, Jain R. (2004). Development and characterization of mucoadhesive microspheres bearing salbutamol for nasal delivery. Drug Deliv, 11:113–22.
   PubMed Web of Science ®Google Scholar
• Soni T, Nagda C, Gandhi T, Chotai N. (2008). Development of discriminating method for dissolution of aceclofenac marketed formulations. Dissol Tech, 15(2):31–5.
   Web of Science ®Google Scholar
• Costa P, Lobo J. (2001). Modeling and comparison of dissolution profiles. Eur J Pharm Sci, 13:123–33.
   PubMed Web of Science ®Google Scholar
• Grabovac V, Guggi D, Bernkop-Schnurch A. (2005). Comparison of the mucoadhesive properties of various polymers. Adv Drug Deliv Rev, 57:1713–23.
   PubMed Web of Science ®Google Scholar
• Martinac A, Filipovic-Grcic J, Voinovich D, Perissutti B, Franceschinis E. (2005). Development and bioadhesive properties of chitosan-ethylcellulose microspheres for nasal delivery. Int J Pharm, 291:69–77.
   PubMed Web of Science ®Google Scholar
• Stahl K, Claesson M, Lillihorn P, Linden H, Backstrom K. (2002). The effect of process variables on the degradation and physical properties of spray dried insulin intended for inhalation. Int J Pharm, 233(1–2):227–37.
   PubMed Web of Science ®Google Scholar
• Hafner A, Filipove-Gri J, Voinovich D, Jalsenjak I. (2007). Development and in vitro characterization of chitosan-based microspheres for nasal delivery of promethazine. Drug Dev Ind Pharm, 33:427–36.
   PubMed Web of Science ®Google Scholar
• Gavini E, Rassu G, Muzzarelli C, Cossu M, Giunchedi P. (2008). Spray-dried microspheres based on methylpyrrolidinone chitosan as new carrier for nasal administration of metoclopramide. Eur J Pharm Biopharm, 68:245–52.
   PubMed Web of Science ®Google Scholar
• Agarwal V, Mishra B. (1999). Design, development, and biopharmaceutical properties of buccoadhesive compacts of pentazocine. Drug Dev Ind Pharm, 25:701–9.
   PubMed Web of Science ®Google Scholar
• Davis S. (2005). Formulation strategies for absorption windows. Drug Discov Today, 10(4):249–57.
   PubMed Web of Science ®Google Scholar
• Carelli V, Di Colo G, Gesi M, Marteni F, Nannipieri E. (1997). Mechanism of drug release from silicone microspheres containing polycarbophil. Int J Pharm, 153:105–14.
   Web of Science ®Google Scholar
• Akiyama Y, Nagahara N, Kashihara T, Hirai S, Toguchi H. (1995). In vitro and in vivo evaluation of mucoadhesive microspheres prepared for the gastrointestinal tract using polyglycerol ester of fatty acids and a poly (acrylic acid) derivatives. Pharm Res, 12(3):397–405.
   PubMed Web of Science ®Google Scholar
• Kockish S, Rees GD, Young SA, Tsibouklis J, Smart JD. (2004). In situ evaluation of drug-loaded microspheres on a mucosal surface under dynamic test conditions. Int J Pharm, 276:51–8.
   PubMed Web of Science ®Google Scholar
• He P, Davis SS, Illum L. (1998). In vitro evaluation of the mucoadhesive properties of chitosan microspheres. Int J Pharm, 166:75–88.
   Web of Science ®Google Scholar
• Pritchard K, Lansley AB, Martin GP, Helliwell M, Marriott C, Benedetti LM. (1996). Evaluation of bioadhesive properties of hyaluronan derivatives: Detachment weight and mucocilliary transport rate. Int J Pharm, 129:137–45.
   Web of Science ®Google Scholar
• Kockish S, Rees GD, Young SA, Tsibouklis J, Smart JD. (2003). Polymeric microspheres for drug delivery to the oral cavity: An in vitro evaluation of mucoadhesive potential. J Pharm Sci, 92(8):1614–23.
   PubMed Web of Science ®Google Scholar
• Martinac A, Filipovic-Grcic J, Perissutti B, Voinovich D, Pavelic Z. (2005). Spray-dried chitosan/ethylcellulose microspheres for nasal drug delivery: Swelling study and evaluation of in vitro drug release properties. J Microencapsul, 22(5):549–61.
   PubMed Web of Science ®Google Scholar
• Rama Rao K, Senapati P, Das MK. (2005). Formulation and in vitro evaluation of ethyl cellulose microspheres containing zidovudine. J Microencapsul, 22(8):863–76.
   PubMed Web of Science ®Google Scholar
• Das MK, Maurya PK. (2008). Evaluation of diltiazem hydrochloride-loaded mucoadhesive microspheres prepared by emulsification-internal gelation technique. Acta Pol Pharm, 65(2):249–59.
   PubMed Web of Science ®Google Scholar