246
Views
5
CrossRef citations to date
0
Altmetric
Research Articles

Solvents effects on crystallinity and dissolution of β-artemether*

, , , , , , , , & show all
Pages 372-378 | Received 28 Jun 2016, Accepted 20 Oct 2016, Published online: 14 Nov 2016

References

  • Mishra SK, Wiese L. Advances in the management of cerebral malaria in adults. Curr Opin Neurol 2009;22:302–7.
  • Terkuile F, White NJ, Holloway P, et al. Plasmodium falciparum: in vitro studies of the pharmacodynamic properties of drugs used for the treatment of severe malaria. Exp Parasitol 1993;76:85–95.
  • Hien T, Davis T, Chuong L, et al. Comparative pharmacokinetics of intramuscular artesunate and artemether in patients with severe falciparum malaria. Antimicrob Agents Chemother 2004;48:4234–9.
  • Suputtamongkol Y, Newton PN, Angus B, et al. A comparison of oral artesunate and artemether antimalarial bioactivities in acute falciparum malaria. Br J Clin Pharmacol 2001;52:655–61.
  • Li QG, Peggins JO, Fleckenstein LL, et al. The pharmacokinetics and bioavailability of dihydroartemisinin, arteether, artemether, artesunic acid and artelinic acid in rats. J Pharm Pharmacol 1998;50:173–82.
  • Joshi M, Pathak S, Sharma S, Patravale V. Design and in vivo pharmacodynamic evaluation of nanostructured lipid carriers for parenteral delivery of artemether: Nanoject. Int J Pharm 2008;364:119–26.
  • Zhang Y, Liu QZ, Zhang DK, Jiang YB. Polymorphism, crystal structure and crystal habit of β-artemether. J Chem Indus Eng (China) 2011;62:2958–63.
  • Gao H, Chen L, Chen W, Bao S. Thermal stability evaluation of β-artemether by DSC and ARC. Thermochimica Acta 2013;569:134–8.
  • Zhang Y, Jiang Y, Zhang D, et al. Metastable zone width, crystal nucleation and growth kinetics measurement in anti-solvent crystallization of β-artemether in the mixture of ethanol and water. Adv Space Res 2015;95:454–62.
  • Vippagunta SR, Brittain HG, Grant DJ. Crystalline solids. Adv Drug Deliv Rev 2001;48:3–26.
  • Kapoor A, Majumdar DK, Yadav MR. Crystal forms of nimesulide: a sulfonanilide(non-steroidal anti-inflammatory drug). Indian J Chem 1998;6:572–5.
  • Aguiar AJ, Krc J, Kinkel AW, Samyn JC. Effect of polymorphism on the absorption of chloramphenicol from chloramphenicol palmitate. J Pharm Sci 1967;56:847–53.
  • Kato Y, Okamoto Y, Nagasawa K, Ishihara I. New polymorphic forms of phenobarbital. Chem Pharm Bull 1984;32:4170
  • Salole E, Al-Sarraj F. Spironolactone crystal forms. Drug Develop Indus Phar 1985;11:855–64.
  • Kobayashi Y, Ito S, Itai S, Yamamoto K. Physicochemical properties and bioavailability of carbamazepine polymorphs and dihydrate. Int J Pharm 2000;193:137–46.
  • Tiwary A. Modification of crystal habit and its role in dosage form performance. Drug Develop Indust Pharm 2001;27:699–709.
  • Burt HM, Mitchell A. Dissolution anisotropy in nickel sulfate α hexahydrate crystals. Int J Pharm 1979;3:261–74.
  • Hammouda Y, El-Khordagui L, Darwish I, El-Kamel A. Manipulation of powder characteristics by interactions at the solid–liquid interface: 1-sulphadiazine. Eur J Pharm Sci 1999;8:283–90.
  • Burt HM, Mitchell A. Effect of habit modification on dissolution rate. Int J Pharm 1980;5:239–51.
  • Chow A-L, Chow P, Zhongshan W, Grant D. Modification of acetaminophen crystals: influence of growth in aqueous solutions containing p-acetoxyacetanilide on crystal properties. Int J Pharm 1985;24:239–58.
  • Femi-Oyewo MN, Spring M. Studies on paracetamol crystals produced by growth in aqueous solutions. Int J Pharm 1994;112:17–28.
  • Garekani HA, Ford JL, Rubinstein MH, Rajabi-Siahboomi AR. Highly compressible paracetamol—II. Compression properties. Int J Pharm 2000;208:101–10.
  • Lahav M, Leiserowitz L. The effect of solvent on crystal growth and morphology. Chem Eng Sci 2001;56:2245–53.
  • Fule RA, Meer TS, Sav AR, Ameen PD. Artemether-soluplus hot-melt extrudate solid dispersion systems for solubility and dissolution rate enhancement with amorphous state characteristics. J Pharm 2013;2013:151432.
  • Keraliya RA, Soni TG, Thakkar VT, Gandhi TR. Effect of solvent on crystal habit and dissolution behavior of tolbutamide by initial solvent screening. Dissol Technol 2010;1:16–21.
  • Assaf SM, Mai SK, Obeidat R, Arida AI. Effect of different organic solvents on crystal habit of mefenamic acid. Jordan J Pharmaceut Sci 2009;2:150–57.
  • Wang Z, Chen J, Li L, et al. Detailed structural study of β-artemether: density functional theory (DFT) calculations of infrared, Raman spectroscopy, and vibrational circular dichroism. J Mol Struct 2015;1097:61–8.
  • Ramteke KH, Dighe PA, Kharat AR, Patil SV. Mathematical models of drug dissolution: a review. Sch Acad J Pharmacy 2014;3:388–96.

Reprints and Corporate Permissions

Please note: Selecting permissions does not provide access to the full text of the article, please see our help page How do I view content?

To request a reprint or corporate permissions for this article, please click on the relevant link below:

Academic Permissions

Please note: Selecting permissions does not provide access to the full text of the article, please see our help page How do I view content?

Obtain permissions instantly via Rightslink by clicking on the button below:

If you are unable to obtain permissions via Rightslink, please complete and submit this Permissions form. For more information, please visit our Permissions help page.