261
Views
11
CrossRef citations to date
0
Altmetric
Research Articles

Preparation and evaluation of metoprolol tartrate sustained-release pellets using hot melt extrusion combined with hot melt coating

, , &
Pages 939-946 | Received 23 Jun 2016, Accepted 23 Jan 2017, Published online: 09 Feb 2017

References

  • Kipping T, Rein H. A new method for the continuous production of single dosed controlled release matrix systems based on hot-melt extruded starch: analysis of relevant process parameters and implementation of an in-process control. Eur J Pharm Biopharm 2013;84:156–71.
  • Bialleck S, Rein H. Preparation of starch-based pellets by hot-melt extrusion. Eur J Pharm Biopharm 2011;79:440–8.
  • Pimparade MB, Morott JT, Park JB, et al. Development of taste masked caffeine citrate formulations utilizing hot melt extrusion technology and in vitro–in vivo evaluations. Int J Pharm 2015;487:167–76.
  • Repka MA, Gutta K, Prodduturi S, et al. Characterization of cellulosic hot-melt extruded films containing lidocaine. Eur J Pharm Biopharm 2005;59:189–96.
  • Verhoeven E, Vervaet C, Remon JP. Xanthan gum to tailor drug release of sustained-release ethylcellulose mini-matrices prepared via hot-melt extrusion: in vitro and in vivo evaluation. Eur J Pharm Biopharm 2006;63:320–30.
  • Özgüney I, Shuwisitkul D, Bodmeier R. Development and characterization of extended release Kollidon SR mini-matrices prepared by hot-melt extrusion. Eur J Pharm Biopharm 2009;73:140–5.
  • Young CR, Crowley M, Dietzsch C, et al. Physicochemical properties of film-coated melt-extruded pellets. J Microencapsul 2007;24:57–71.
  • Chansanroj K, Betz G, Leuenberger H, et al. Development of a multi-unit floating drug delivery system by hot melt coating technique with drug-lipid dispersion. J Drug Del Sci Tech 2007;17:333–8.
  • Jannin V, Cuppok Y. Hot-melt coating with lipid excipients. Int J Pharm 2013;457:480–7.
  • Kulah G, Kaya O. Investigation and scale-up of hot-melt coating of pharmaceuticals in fluidized beds. Powder Technol 2011;208:175–84.
  • Barthelemya P, Laforeta JP, Faraha N, et al. Compritol 888 ATO: an innovative hot-melt coating agent for prolonged-release drug formulations. Eur J Pharm Biopharm 1999;47:87–90.
  • DiNunzioa JC, Brough C, Millera DA, et al. Applications of KinetiSol dispersing for the production of plasticizer free amorphous solid dispersions. Eur J Pharm Sci 2010;40:179–87.
  • Young CR, Koleng JJ, McGinity JW, et al. Production of spherical pellets by a hot-melt extrusion and spheronization process. Int J Pharm 2002;242:87–92.
  • Quinten T, De Beer T, Vervaet C, et al. Evaluation of injection moulding as a pharmaceutical technology to produce matrix tablets. Eur J Pharm Biopharm 2009;71:145–54.
  • Goyanes A, Robles Martinez P, Buanz A, et al. Effect of geometry on drug release from 3D printed tablets. Int J Pharm 2015;494:657–63.
  • Verhoeven E, De Beer TR, Schacht E, et al. Influence of polyethylene glycol/polyethylene oxide on the release characteristics of sustained-release ethylcellulose mini-matrices produced by hot-melt extrusion: in vitro and in vivo evaluations. Eur J Pharm Biopharm 2009;72:463–70.
  • Chen H, Shi S, Liu A, et al. Combined application of extrusion-spheronization and hot-melt coating technologies for improving moisture-proofing of herbal extracts. J Pharm Sci 2010;99:2444–54.
  • Zhang Y, Luo R, Chen Y, et al. Application of carrier and plasticizer to improve the dissolution and bioavailability of poorly water-soluble baicalein by hot melt extrusion. AAPS PharmSciTech 2014;15:560–8.
  • Schilling SU, Shah NH, Waseem Malick A, et al. Properties of melt extruded enteric matrix pellets. Eur J Pharm Biopharm 2010;74:352–61.
  • Tiwari R, Agarwal SK, Murthy RSR, et al. Formulation and evaluation of sustained release extrudes prepared via novel hot melt extrusion technique. J Pharm Innov 2014;9:246–58.
  • Melocchi A, Loreti G, Del Curto MD, et al. Evaluation of hot-melt extrusion and injection molding for continuous manufacturing of immediate-release tablets. J Pharm Sci 2015;104:1971–80.
  • Repka MA, Langley N, DiNunzio J, 2013. Melt extrusion: materials, technology and drug product design. New York, NY: Springer.
  • Martin C. Continuous mixing of solid dosage forms via hot-melt extrusion. Pharm Technol 2008;32:76–86.
  • Gupta SS, Parikh T, Meena AK, et al. Effect of carbamazepine on viscoelastic properties and hot melt extrudability of Soluplus®. Int J Pharm 2015;478:232–9.

Reprints and Corporate Permissions

Please note: Selecting permissions does not provide access to the full text of the article, please see our help page How do I view content?

To request a reprint or corporate permissions for this article, please click on the relevant link below:

Academic Permissions

Please note: Selecting permissions does not provide access to the full text of the article, please see our help page How do I view content?

Obtain permissions instantly via Rightslink by clicking on the button below:

If you are unable to obtain permissions via Rightslink, please complete and submit this Permissions form. For more information, please visit our Permissions help page.