Advanced search
Publication Cover
Drug Development and Industrial Pharmacy Volume 43, 2017 - Issue 8
Submit an article Journal homepage
246
Views
16
CrossRef citations to date
0
Altmetric
Research Article

Solubility and dissolution rate improvement of the inclusion complex of apigenin with 2-hydroxypropyl-β-cyclodextrin prepared using the liquid antisolvent precipitation and solvent removal combination methods

Weiwei WuKey Laboratory of Saline-alkali Vegetation Ecology Restoration in Oil Field (SAVER), Ministry of Education, Alkali Soil Natural Environmental Science Center (ASNESC), Northeast Forestry University, Harbin, China; View further author information
,
Yuangang ZuKey Laboratory of Forest Plant Ecology, Northeast Forestry University, Ministry of Education, Harbin, ChinaView further author information
,
Xiuhua ZhaoKey Laboratory of Forest Plant Ecology, Northeast Forestry University, Ministry of Education, Harbin, ChinaCorrespondence[email protected]
View further author information
,
Xinxin ZhangKey Laboratory of Saline-alkali Vegetation Ecology Restoration in Oil Field (SAVER), Ministry of Education, Alkali Soil Natural Environmental Science Center (ASNESC), Northeast Forestry University, Harbin, China; Correspondence[email protected]
View further author information
,
Lingling WangKey Laboratory of Forest Plant Ecology, Northeast Forestry University, Ministry of Education, Harbin, ChinaView further author information
,
Yuanyuan LiKey Laboratory of Forest Plant Ecology, Northeast Forestry University, Ministry of Education, Harbin, ChinaView further author information
,
Li WangKey Laboratory of Forest Plant Ecology, Northeast Forestry University, Ministry of Education, Harbin, ChinaView further author information
,
Yin ZhangKey Laboratory of Forest Plant Ecology, Northeast Forestry University, Ministry of Education, Harbin, ChinaView further author information
&
Bolin LianKey Laboratory of Forest Plant Ecology, Northeast Forestry University, Ministry of Education, Harbin, ChinaView further author information
 show all
Pages 1366-1377 | Received 17 Oct 2016, Accepted 03 Apr 2017, Published online: 24 Apr 2017

References

  • Zhang J, Huang Y, Liu D, et al. Preparation of apigenin nanocrystals using supercritical antisolvent process for dissolution and bioavailability enhancement. Eur J Pharm Sci. 2013;48:740–747.
  • Ding SM, Zhang ZH, Song J, et al. Enhanced bioavailability of apigenin via preparation of a carbon nanopowder solid dispersion. Int J Nanomedicine. 2014;9:2327–2333.
  • Zhai Y, Guo S, Liu C, et al. Preparation and in vitro evaluation of apigenin-loaded polymeric micelles. Colloids Surf A: Physicochem Eng Aspects. 2013;429:24–30.
  • Shen L-N, Zhang Y-T, Wang Q, et al. Enhanced in vitro and in vivo skin deposition of apigenin delivered using ethosomes. Int J Pharm. 2014;460:280–288.
  • Duchěne D, Wouessidjewe D. Pharmaceutical uses of cyclodextrins and derivatives. Drug Dev Ind Pharm. 2008;16:2487–2499.
  • Zhao X, Wang Z, Li X. Preparation, in-vitro release and antioxidant potential of formulation of apigenin with hydroxypropyl-β-cyclodextrin modified microemulsion. J Incl Phenom Macrocycl Chem. 2016;86:1–10.
  • Sanghavi NM, Mayekar R, Fruitwala M. Inclusion complexes of terfenadine-cyclodextrins. Drug Dev Ind Pharm. 2008;21:375–381.
  • Zu Y, Wu W, Zhao X, et al. The high water solubility of inclusion complex of taxifolin-γ-CD prepared and characterized by the emulsion solvent evaporation and the freeze drying combination method. Int J Pharm. 2014;477:148–158.
  • Kim H, Kim HW, Jung S. Aqueous solubility enhancement of some flavones by complexation with cyclodextrins. Bull Korean Chem Soc. 2008;29:590–594.
  • Li J. Study and characterization of the antioxidant activity of the inclusion complex of apigenin with beta-cyclodextrin and HP-beta-cyclodextrin in solution. J Invest Biochem. 2014;3:107.
  • Pápay ZE, Sebestyén Z, Ludányi K, et al. Comparative evaluation of the effect of cyclodextrins and pH on aqueous solubility of apigenin. J Pharm Biomed Anal. 2016;117:210–216.
  • Huang Y, Zu Y, Zhao X, et al. Preparation of inclusion complex of apigenin-hydroxypropyl-β-cyclodextrin by using supercritical antisolvent process for dissolution and bioavailability enhancement. Int J Pharm. 2016;511:921–930.
  • Wang Z, Chen JF, Le Y, et al. Preparation of ultrafine beclomethasone dipropionate drug powder by antisolvent precipitation. Ind Eng Chem Res. 2007;46:4839–4845.
  • Luo X, Xu YH, Chen B, et al. Solubilization on cryptotanshinone by hydroxypropyl-beta-cyclodextrin and preparation of their inclusion compound. Zhongguo Zhong Yao Za Zhi. 2005;30:1328–1331.
  • Chen XY, Liu WY, Zhang J. Study on the characterization of beta-cyclodextrin-diferrocenylenone inclusion complex and micro-environmental effects. Guang Pu Xue Yu Guang Pu Fen Xi. 2006;26:1285–1289.
  • Ji MH, Shu HM, Guo FY, et al. Study on the preparation process of inclusion complex of volatile oil of Dalbergia odorifera-beta-cyclodextrin. Zhong Yao Cai. 2009;32:114–117.
  • Ahn BK, Lee SG, Kim SR, et al. Inclusion compound formulation of hirsutenone with beta-cyclodextrin. J Pharm Invest. 2013;43:453–459.
  • Li B, Robinson DH, Birt DF. Evaluation of properties of apigenin and [G-3H]apigenin and analytic method development. J Pharm Sci. 1997;86:721–725.
  • Romero S, Escalera B, Bustamante P. Solubility behavior of polymorphs I and II of mefenamic acid in solvent mixtures. Int J Pharm. 1999;178:193–202.
  • Park Y, Lee J, Sun HL, et al. Crystal structures of tetramorphic forms of donepezil and energy/temperature phase diagram via direct heat capacity measurements. Cryst Growth Des. 2013;13:5450–5458.
  • Zhu WZ, Wang JX, Shao L, et al. Liquid antisolvent preparation of amorphous cefuroxime axetil nanoparticles in a tube-in-tube microchannel reactor. Int J Pharm. 2010;395:260–265.
  • Zhang HX, Wang JX, Zhang ZB, et al. Micronization of atorvastatin calcium by antisolvent precipitation process. Int J Pharm. 2009;374:106–113.
  • Zhang J, Liu D, Huang Y, et al. Biopharmaceutics classification and intestinal absorption study of apigenin. Int J Pharm. 2012;436:311–317.

Reprints and Corporate Permissions

Please note: Selecting permissions does not provide access to the full text of the article, please see our help page How do I view content?

To request a reprint or corporate permissions for this article, please click on the relevant link below:

Order Reprints Request Corporate Permissions

Academic Permissions

Please note: Selecting permissions does not provide access to the full text of the article, please see our help page How do I view content?

Obtain permissions instantly via Rightslink by clicking on the button below:

Request Academic Permissions

If you are unable to obtain permissions via Rightslink, please complete and submit this Permissions form. For more information, please visit our Permissions help page.

Related research

People also read lists articles that other readers of this article have read.

Recommended articles lists articles that we recommend and is powered by our AI driven recommendation engine.

Cited by lists all citing articles based on Crossref citations.
Articles with the Crossref icon will open in a new tab.