24
Views
19
CrossRef citations to date
0
Altmetric
Original Articles

A new Synthesis of 1-(2,3-Dideoxy-β-D-Glycero-Pent-2-Enofuranosyl)- Thymine. A Highly Potent and Selective Anti-Hiv Agent

, &
Pages 245-258 | Received 19 Jun 1989, Published online: 04 Oct 2006

References

  • Barré-Sinoussi , F. , Chermann , J. C. , Rey , F. , Bygetre , M. T. , Chamaret , S. , Gruest , J. , Dauguet , C. , Axler-Blin , C. , Vézinet-Brun , F. , Rouzioux , C. , Rozenbaum , W. and Montagnier , L. 1983 . Science Vol. 220 , 868 Washington, D. C.
  • Gallo , R. C. , Sarin , P. S. , Gelmann , E. P. , Robert-Guroff , M. , Richardson , E. , Kalyanaraman , V. S. , Mann , D. , Sidhu , G. D. , Stahl , R. E. , Zolla-Pazner , S. , Leibowitch , J. and Popovic , M. 1983 . Science Vol. 220 , 865 Washington, D. C.
  • de Clercq , E. 1986 . J. Med. Chem. , 29 : 1561
  • Balzarini , J. , Baba , M. , Pauwels , R. , Herdewijn , P. , Wood , S. E. , Robins , M. J. and De Clercq , E. 1988 . Mol. Pharmacol. , 33 : 243
  • Mitsuya , H. and Broder , S. 1986 . Proc. Natl. Acad. Sci. U. S. A. , 83 : 1911
  • Balzarini , J. , Pauwels , R. , Baba , M. , Robins , M. , Zou , R. , Herdewijn , P. and De Clercq , E. 1987 . Biochem. Biophys. Res. Commun. , 145 : 269
  • Kim , C.-H. , Marquez , V. E. , Broder , S. , Mitsuya , H. and Driscoll , J. 1987 . J. Med. Chem. , 30 : 862
  • Baba , M. , Pauwels , R. , Herdewijn , P. , De Clercq , E. , Desmyter , J. and Vandeputte , M. 1987 . Biochem. Biophys. Res. Comrnun. , 142 : 128
  • Bazin , H. , Datema , R. , Remaud , G. , Ericson , A-C. , Gilljam , G. , Johansson , N. G. , Hansen , J. , Koshida , R. , Moelling , K. , Öberg , B. , Stening , G. , Vrang , L. , Wahren , B. , Wu , J-C. and Chattopadhyaya , J. 1989 . Biochemical Pharmacology , 38 ( 1 ) : 109 – 119 .
  • Lin , T. S. , Chen , M. S. , McLaren , C. , Gao , Y.-S. , Ghazzouli , L. and Prusoff , W. H. 1987 . J. Med. Chem. , 30 : 440
  • Lin , T. S. , Schinazi , R. F. and Prusoff , W. H. 1987 . Biochem. Pharmacol. , 17 : 2713
  • Baba , M. , Pauwels , R. , Herdewijn , P. , De Clercq , E. , Desmyter , J. and Vandeputte , M. 1987 . Biochem. Biophys. Res. Commun. , 142 : 128
  • Balzarini , J. , Kang , G.-J. , Dalal , M. , Herdewijn , P. , De Clercq , E. , Broder , S. and Johns , D. G. 1987 . Mol. Pharmacol. , 32 : 162
  • Hamamoto , Y. , Nakashima , H. , Matsui , T. , Matsuda , A. , Ueda , T. and Yamamoto , N. 1987 . Antimicrob. Agents Chemother. , 31 : 907
  • Mansuri , M. M. , Starrett , J. E. Jr. , Ghazzouli , I. , Hitchcock , M. J. M. , Sterzycki , R. Z. , Brankovan , V. , Lin , T.-S. , August , E. M. , Prusoff , W. H. , Sommadossi , J.-P. and Martin , J. C. 1989 . J. Med. Chem. , 32 : 461
  • Horwitz , J. and Chua , J. 1968 . Synthetic Procedures in Nucleic Acid Chemistry , Edited by: Zorbach , W. W. and Tipson , R. S. Vol. 1 , 344 New York : Interscience .
  • Horwitz , J. , Chua , J. , Da Rooge , M. A. , Noel , M. and Klundt , I. L. 1966 . J. Org. Chem. , 31 : 205
  • Verheyden , J. P. H. and Moffatt , J. G. 1974 . J. Org. Chem. , 39 : 3573
  • Fox , J. J. 1969 . Pure and Applied Chemistry , 18 : 223 – 254 .
  • Paulmiere , C . 1986 . “Selenium Reagents and Intermediates in Organic Synthesis” , Oxford, , England : Pergamon Press .
  • Walker , R. T. , De Clercq , E. and Eckstein , F. , eds. 1979 . “Nucleoside Analogues” , NATO Advanced Study Institutes Seris New York : Plenum Press .
  • Nyilas , A. and Chattopadhyaya , J. 1986 . Acta Chem. Scand. , B40 : 826
  • Vial , J.-M. , Balgobin , N. , Remaud , G. , Nyilas , A. and Chattopadhyaya , J. 1987 . Nucleosides & Nucleotides , 6 : 209
  • Chu , C. K. , Bhadti , V. S. , Doboszewski , B. , Gu , Z. P. , Kosugi , Y. , Pullaiah , K. C. and Van Roey , P. 1989 . J. Org. Chem. , 54 : 2217

Reprints and Corporate Permissions

Please note: Selecting permissions does not provide access to the full text of the article, please see our help page How do I view content?

To request a reprint or corporate permissions for this article, please click on the relevant link below:

Academic Permissions

Please note: Selecting permissions does not provide access to the full text of the article, please see our help page How do I view content?

Obtain permissions instantly via Rightslink by clicking on the button below:

If you are unable to obtain permissions via Rightslink, please complete and submit this Permissions form. For more information, please visit our Permissions help page.