Physicochemical Properties of Phytopharmaceutical Preparations as Affected by Drying Methods and Carriers

REFERENCES

• Oliveira , W.P. ; Bott , R.F. ; Souza , C.R.F. Manufacture of standardized dried extracts from medicinal Brazilian plants . Drying Technology 2006 , 24 ( 4 ), 523 – 533 .
   Web of Science ®Google Scholar
• Bott , R.F. ; Labuza , T.P. ; Oliveira , W.P. Stability testing of spray- and spouted bed–dried extracts of Passiflora alata . Drying Technology 2010 , 28 ( 11 ), 1255 – 1265 .
   Web of Science ®Google Scholar
• Oliveira , W.P. ; Freitas , L.A.P. ; Freire , J.T. Drying of pharmaceutical products . In: Transport Phenomena in Particulate Systems ; Freire , J.T. , Silveira , A.M. , Ferreira , M.C. , Eds.; Bethan Science : Oak Park, IL , 2012 ; 148–171 .
   Google Scholar
• Bringas-Lantigua , M. ; Expósito-Molina , I. ; Reineccius , G.A. ; López-Hernández , O. ; Pino , J.A. Influence of spray-dryer air temperatures on encapsulated mandarin oil . Drying Technology 2011 , 29 ( 5 ), 520 – 526 .
   Web of Science ®Google Scholar
• Huynh , T.V. ; Caffin , N. ; Dykes , G.A. ; Bhandari , B. Optimization of the microencapsulation of lemon myrtle oil using response surface methodology . Drying Technology 2008 , 26 ( 3 ), 357 – 368 .
   Web of Science ®Google Scholar
• Ré , M.I. Formulating drug delivery systems by spray drying . Drying Technology 2006 , 24 ( 4 ), 433 – 448 .
   Web of Science ®Google Scholar
• Oliveira , O.W. ; Petrovick , P.R. Spray drying of plant extracts: Basic remarks and application . Brazilian Journal of Pharmacognosy 2010 , 20 ( 4 ), 641 – 650 (in Portuguese) .
   Google Scholar
• Sahin-Nadeem , H. ; Torun , M. ; Ozdemir , F. Spray drying of the mountain tea (Sideritis stricta) water extract by using different hydrocolloid carriers . LWT – Food Science and Technology 2011 , 44 ( 7 ), 1626 – 1635 .
   Web of Science ®Google Scholar
• Sansone , F. ; Mencherini , T. ; Picerno , P. ; D'amore , M. ; Aquino , R.P. ; Lauro , M.R. Maltodextrin/pectin microparticles by spray drying as carrier for nutraceutical extracts . Journal of Food Engineering 2011 , 105 ( 3 ), 468 – 476 .
   Web of Science ®Google Scholar
• Rocha , G.A. ; Fávaro-Trindade , C.S. ; Grosso , C.R.F. Microencapsulation of lycopene by spray drying: Characterization, stability and application of microcapsules . Food and Bioproducts Processing 2012 , 90 ( 1 ), 37 – 42 .
   Web of Science ®Google Scholar
• Tonon , R.V. ; Grosso , C.R.F. ; Hubinger , M.D. Influence of emulsion composition and inlet air temperature on the microencapsulation of flaxseed oil by spray drying . Food Research International 2010 , 44 ( 1 ), 282 – 289 .
   Web of Science ®Google Scholar
• Quispe-Condori , S. ; Saldaña , M.D.A. ; Temelli , F. Microencapsulation of flax oil with zein using spray and freeze drying . LWT – Food Science and Technology 2011 , 44 ( 9 ), 1880 – 1887 .
   Web of Science ®Google Scholar
• Gallo , L. ; Llabot , J.M. ; Allemandi , D. ; Bucalá , V. ; Piña , J. Influence of spray-drying operating conditions on Rhamnus purshiana (cáscara sagrada) extract powder physical properties . Powder Technology 2011 , 208 ( 1 ), 205 – 214 .
   Web of Science ®Google Scholar
• Kalogeropoulos , N. ; Yannakopoulou , K. ; Gioxari , A. ; Chiou , A. ; Makris , D.P. Polyphenol characterization and encapsulation in β-cyclodextrin of a flavonoid-rich Hypericum perforatum (St. John's wort) extract . LWT - Food Science and Technology 2010 , 43 , 882 – 889 .
   Web of Science ®Google Scholar
• Souza , C.R.F. ; Oliveira , W.P. Powder properties and system behavior during spray drying of Bauhinia forficata Link extract . Drying Technology 2006 , 24 ( 6 ), 735 – 749 .
   Web of Science ®Google Scholar
• Runha , F.P. ; Cordeiro , D.S. ; Pereira , C.A.M. ; Vilegas , J. ; Oliveira , W.P. Production of dry extracts of medicinal Brazilian plants by spouted bed process: Development of the process and evaluation of thermal degradation during the drying operation. Transactions of the Institution of Chemical Engineers 2001, 79, 160–168.
   Google Scholar
• Souza , C.R.F. ; Oliveira , W.P. Spouted bed drying of Bauhinia forficata Link extract: The effects of feed atomizer position and operating conditions on equipment performance and product properties . Brazilian Journal of Chemical Engineering 2005 , 22 ( 2 ), 239 – 247 .
   Web of Science ®Google Scholar
• Chu , K.K.W. ; Chow , A.H.L. Impact of carbohydrate constituents on moisture sorption of herbal extracts . Pharmaceutical Research 2000 , 17 ( 9 ), 1133 – 1137 .
   PubMed Web of Science ®Google Scholar
• Gharsallaoui , A. ; Roudaut , G. ; Chambin , O. ; Voilley , A. ; Saurel , R. Applications of spray-drying in microencapsulation of food ingredients: An overview . Food Research International 2007 , 40 ( 9 ), 1107 – 1121 .
   Web of Science ®Google Scholar
• Fernandes , L.P. ; Oliveira , W.P. ; Sztatisz , J. ; Szilágyi , I.M. ; Novák , CS. Solid state studies on molecular inclusions of Lippia sidoides essential oil obtained by spray drying . Journal of Thermal Analysis and Calorimetry 2009 , 95 ( 3 ), 855 – 863 .
   Web of Science ®Google Scholar
• Brandão , M.G.L. ; Krettli , A.U. ; Soares , L.S.R. ; Nery , C.G.C. ; Marinuzzi , H.C. Antimalarial activity of extracts and fractions from Bidens pilosa and other Bidens species (Asteraceae) correlated with the presence of acetylene and flavonoid compounds . Journal of Ethnopharmacology 1997 , 57 ( 2 ), 131 – 138 .
   Web of Science ®Google Scholar
• Ubillas , R.P. ; Mendez , C.D. ; Jolad , S.D. ; Luo , J. ; King , S.R. ; Carlson , T.J. ; Fort , M.D. Antihyperglycemic acetylenic glucosides from Bidens pilosa . Planta Medica 2000 , 66 ( 1 ), 82 – 83 .
   Web of Science ®Google Scholar
• Wang , R. ; Wu , Q. ; Shi , Y. Polyacetylenes and flavonoids from de aerial parts of Bidens pilosa . Planta Medica 2010 , 76 ( 9 ), 893 – 896 .
   PubMed Web of Science ®Google Scholar
• Wu , L. ; Ching , Y. ; Chuang , H. ; Lo , C. ; Yang , K. ; Wang , S. ; Shyur , L. A novel polyacetylene significantly inhibits angiogenesis and promotes apaptosis in human endothelial cells through activation of the CDK inhibitors and caspase-7 . Planta Medica 2007 , 73 ( 7 ), 655 – 661 .
   Web of Science ®Google Scholar
• Silva , D.B. Anti-allergic activity and chemistry studies of Bidens gardeni Bak. and Bidens sulpurea (Cav.) Sch. Bip. (Asteraceae). Doctoral thesis, Faculdade de Ciências Farmacêuticas de Ribeirão Preto, Brazil, 2009 (in Portuguese).
   Google Scholar
• Chien , S. ; Young , P. ; Hsu , Y. ; Chen , C. ; Tien , Y. ; Shiu , S. ; Li , T. ; Yang , C. ; Marimuthu , P. ; Tsai , L.F. ; Yang , W. Anti-diabetic properties of three common Bidens pilosa variants in Taiwan . Phytochemistry 2009 , 70 ( 10 ), 1246 – 1254 .
   PubMed Web of Science ®Google Scholar
• Kviecinski , M.R. ; Benelli , P. ; Felipe , K.B. ; Correia , J.F.G. ; Pich , C.T. ; Ferreira , S.R.S. ; Pedrosa , R.C. SFE from Bidens pilosa Linné to obtain extracts rich in cytotoxic polyacetylenes with antitumor activity . Journal of Supercritical Fluids 2011 , 56 ( 3 ), 243 – 248 .
   Web of Science ®Google Scholar
• Rojas , J.J. ; Ochoa , V.J. ; Ocampo , S.A. ; Muñoz , J.F. Screening for antimicrobial activity of ten medicinal plants used in Colombian folkloric medicine: A possible alternative in the treatment of non-nosocomial infections . BMC Complementary and Alternative Medicine 2006 , 6 ( 2 ), 1 – 6 .
   Google Scholar
• Kviecinski , M.R. ; Felipe , K.B. ; Correia , J.F.G. ; Ferreira , E.A. ; Rossi , M.A. ; Gatti , F.M. ; Wilhelm , D. ; Pedrosa , R.C. Brazilian Bidens pilosa Linné yields fraction containing quercetin-derived flavonoid with free radical scavenger activity and hepatoprotective effects . Libyan Journal of Medicine 2011 , 6 , 5651 .
   PubMed Web of Science ®Google Scholar
• Yuan , L. ; Chen , F. ; Ling , L. ; Dou , P. ; Bo , H. ; Zhong , M. ; Xia , L. Protective effects of total flavonoids of Bidens pilosa L. (TFB) on animal liver injury and liver fibrosis . Journal of Ethnopharmacology 2008 , 116 ( 3 ), 539 – 546 .
   PubMed Web of Science ®Google Scholar
• Chiang , Y. ; Chuang , D. ; Wang , S. ; Kuo , Y. ; Tsai , P. ; Shyur , L. Metabolite profiling and chemopreventive bioactivity of plant extracts from Bidens pilosa . Journal of Ethnopharmacology 2004 , 95 ( 2–3 ), 409 – 419 .
   Web of Science ®Google Scholar
• Brazilian Sanitary Surveillance Agency. Resolution RDC No. 10; Ministry of Health: Brasilia D. F., 2010.
   Google Scholar
• Cortés-Rojas , D.F. ; Souza , C.R.F. ; Oliveira , W.P. Optimisation of the extraction of phenolic compounds and antioxidant activity from aerial parts of Bidens pilosa L. using response surface methodology . International Journal of Food Science and Technology 2011 , 46 ( 11 ), 2420 – 2427 .
   Web of Science ®Google Scholar
• Cano-Chauca , M. ; Stringheta , P.C. ; Ramos , A.M. ; Cal-Vidal , J. Effect of the carriers on the microstructure of mango powder obtained by spray drying and its functional characterization . Innovative Food Science and Emerging Technologies 2005 , 6 ( 4 ), 420 – 428 .
   Web of Science ®Google Scholar
• Souza , C.R.F. ; Oliveira , W.P. Microencapsulation of ketoprofen in blends of acrylic resins by spray drying . Drying Technology 2012 , 30 ( 3 ), 263 – 275 .
   Web of Science ®Google Scholar
• Aulton , M.E. Pharmaceutics: The Science of Dosage Form Design, , 2nd ed. ; Churchill Livingstone : New York , 2002 .
   Google Scholar
• U.S. Food and Drug Administration. Q4B evaluation and recommendation of pharmacopoeial texts for use in the ICH regions, Annex 13: Bulk density and tapped density of powders; US FDA: Silver Spring, MD, 2010.
   Google Scholar
• Goula , A.M. ; Adamopoulos , K.G. Spray drying of tomato pulp: Effect of feed concentration . Drying Technology 2004 , 22 ( 10 ), 2309 – 2330 .
   Web of Science ®Google Scholar
• Martin del Valle , E.M. Cyclodextrins and their uses: A review . Process Biochemistry 2004 , 39 ( 9 ), 1033 – 1046 .
   Web of Science ®Google Scholar
• Georgetti , S.R. ; Casagrande , R. ; Vicentini , F.T.M.D. ; Verri , W.A. ; Fonseca , M.J.V. Evaluation of the antioxidant activity of soybean extract by different in vitro methods and investigation of this activity after its incorporation in topical formulations . European Journal of Pharmaceutics and Biopharmaceutics 2006 , 64 ( 1 ), 99 – 106 .
   PubMed Web of Science ®Google Scholar
• Souza , J.P.B. ; Tacon , L.A. ; Correia , C.C. ; Bastos , J.K. ; Freitas , L.A.P. Spray-dried propolis extract, II: Prenylated components of green propolis . Pharmazie 2007 , 62 ( 7 ), 488 – 492 .
   PubMed Web of Science ®Google Scholar
• Pérez-Serradilla , J.A. ; Luque de Castro , M.D. Microwave-assisted extraction of phenolic compounds from wine lees and spray-drying of the extract . Food Chemistry 2011 , 124 ( 4 ), 1652 – 1659 .
   Web of Science ®Google Scholar
• Bakowska-Barczak , A.M. ; Kolodziejczyk , P.P. Black currant polyphenols: Their storage stability and microencapsulation . Industrial Crops and Products 2010 , 34 ( 2 ), 1301 – 1309 .
   Web of Science ®Google Scholar
• Soltoft , M. ; Eriksen , M.R. ; Trager , A.W.B. ; Nielsen , J. ; Laursen , K.H. ; Husted , S. ; Halekoh , U. ; Knuthsen , P. Comparison of polyacetylene content in organically and conventionally grown carrots using a fast ultrasonic liquid extraction method . Journal of Agriculture and Food Chemistry 2010 , 58 ( 13 ), 7673 – 7679 .
   Web of Science ®Google Scholar
• Murray , D.G. ; Luft , L.R. Low-DE corn starches hydrolysates. Multi-functional carbohydrates aid in food formulation . Food Technology 1973 , 27 ( 3 ), 32 – 40 .
   Web of Science ®Google Scholar
• Keey , R.B. Drying of Loose and Particulate Solids Materials ; Hemisphere Publishing Co. : New York , 1992 .
   Google Scholar
• Onwulata , C.I. ; Konstance , R.P. ; Holsinger , V.H. Flow properties of encapsulated milk fat powders as affected by flow agent . Journal of Food Science 1996 , 61 ( 6 ), 1211 – 1215 .
   Web of Science ®Google Scholar
• Chiou , D. ; Langrish , T.A.G. ; Braham , R. Partial crystallization behavior during spray drying: Simulations and experiments . Drying Technology 2008 , 26 ( 1 ), 27 – 38 .
   Web of Science ®Google Scholar
• Bhandari , B.R. ; Howes , T. Implication of glass transition for the drying and stability of dried foods . Journal of Food Engineering 1999 , 40 ( 1–2 ), 71 – 79 .
   Web of Science ®Google Scholar
• Rowe , R.C. ; Sheskey , P.J. ; Quinn , M.E. Handbook of Pharmaceutical Excipients, , 6th Ed ; Pharmaceutical Press : London , 2009 .
   Google Scholar
• Roos , Y. ; Karel , M. Water and molecular weight effects on glass transitions in amorphous carbohydrates and carbohydrate solutions . Journal of Food Science 1991 , 56 , 1676 – 1681 .
   Web of Science ®Google Scholar
• Zhu , P. ; Méjean , S. ; Blanchard , E. ; Jeantet , R. ; Schuck , P. Prediction of dry mass glass transition temperature and the spray drying behaviour of a concentrate using a desorption method. Journal of Food Engineering 2011, 105(3), 460–467.
   Web of Science ®Google Scholar
• Yu , L. Amorphous pharmaceutical solids: Preparation, characterization and stabilization . Advanced Drug Delivery Reviews 2001 , 48 ( 1 ), 27 – 42 .
   PubMed Web of Science ®Google Scholar
• Toneli , J. ; Park , K. ; Negreiros , A. ; Murr , F. Spray-drying process optimization of chicory root inulin . Drying Technology 2010 , 28 ( 3 ), 369 – 379 .
   Web of Science ®Google Scholar
• Islam , M.I.U. ; Langrish , T.A.G. ; Chiou , D. Particle crystallization during spray drying in humid air . Journal of Food Engineering 2010 , 99 ( 1 ), 55 – 62 .
   Web of Science ®Google Scholar
• Langrish , T.A.G. ; Wang , S. Crystallization rates for amorphous sucrose and lactose powders from spray drying: A comparison . Drying Technology 2009 , 27 ( 4 ), 606 – 614 .
   Web of Science ®Google Scholar
• Tabary , N. ; Mahieu , A. ; Willart , J.F. ; Dudognon , E. ; Danède , F. ; Descamps , M. ; Bacquet , M. ; Martel , B. Characterization of the hidden glass transition of amorphous cyclomaltoheptaose . Carbohydrate Research 2011 , 346 ( 14 ), 2193 – 2199 .
   PubMed Web of Science ®Google Scholar
• Picker , K.M. ; Hoag , S.W. Characterization of the thermal properties of microcrystalline cellulose by modulated temperature differential scanning calorimetry . Journal of Pharmaceutical Sciences 2002 , 91 ( 2 ), 342 – 349 .
   PubMed Web of Science ®Google Scholar
• Terinte , N. ; Ibbett , R. ; Schuster , K.C. Overview on native cellulose and microcrystalline cellulose I structure studied by X-ray diffraction (WAXD): Comparison between measurement techniques . Lenzinger Berichte 2011 , 89 , 118 – 131 .
   Google Scholar
• Loftsson , T. ; Brewster , M.E. Pharmaceutical applications of cyclodextrins. 1. Drug solubilization and stabilization . Journal of Pharmaceutical Sciences 1996 , 85 ( 10 ), 1017 – 1025 .
   PubMed Web of Science ®Google Scholar