Microencapsulation of chlorthalidone by spray-drying of double emulsion and melt granulation coating

References

• USP-NF. Test solutions. Unites States Pharmacopoeia 35/National Formulary 30. 2012. http://www.usp.org
   Google Scholar
• Bonfilio, R.; Leal, J.S.; Santos, O.M.M.; Pereira, G.R., Doriguetto, A.C.; de Araújo, M.B. Analysis of chlorthalidone polymorphs in raw materials and tablets and the effect of forms I and II on the dissolution properties of drug products. Journal of Pharmaceutical and Biomedical Analysis 2014, 88, 562–570.
   PubMed Web of Science ®Google Scholar
• Sica, D.A. Chlorthalidone: Has it always been the best thiazide-type diuretic? Hypertension 2006, 47, 321–322.
   PubMed Web of Science ®Google Scholar
• Vázquez, N.; Monroy, A.; Dorantes, E.; Munoz-Clares, R.A.; Gamba, G. Functional differences between flounder and rat thiazide-sensitive Na–Cl cotransporter. American Journal of Physiology Renal Physiology 2002, 282, F599–F607.
   Google Scholar
• Sumiye, L.; Vivian, A.S.; Frisof, K.B.; Podany, E.C. Potassium loss associated with hydrochlorothiazide versus chlorthalidone. Clinical Theraupeutics 1981, 4, 308–320.
   PubMed Web of Science ®Google Scholar
• Carrillo-Navas, H.; Cruz-Olivares, J.; Barrera-Pichardo, J.F.; Pérez-Alonso, C. Rheological properties of a double emulsion nutraceutical system incorporating chia essential oil and ascorbic acid stabilized by carbohydrate polymer–protein blends. Carbohydrate Polymers 2012, 87, 1231–1235.
   Web of Science ®Google Scholar
• Pimentel-González, D.J.; Campos-Montiel, R.G.; Lobato-Calleros, C.; Pedroza-Islas, R.; Vernon-Carter, E.J. Encapsulation of Lactobacillus rhamnosus in double emulsions formulated with sweet whey as emulsifier and survival in simulated gastrointestinal conditions. Food Research International 2009, 42, 292–297.
   Web of Science ®Google Scholar
• Rodríguez-Huezo, M.E.; Pedroza-Islas, R.; Prado-Barragán, L.A.; Beristain, C.I.; Vernon-Carter, E.J. Microencapsulación by spray drying of multiple emulsions containing carotenoids. Journal of Food Science 2004, 69, E351–E359.
   Web of Science ®Google Scholar
• Souza, C.R.F.; Oliveira, W.P. Microencapsulation of Ketoprofen in blends of acrylic resins by spray drying. Drying Technology 2012, 30(3), 263–275.
   Web of Science ®Google Scholar
• Varma, M.V.; Rotter, C.J.; Chupka, J.; Whalen, K.M.; Duignan, D.B.; Feng, B.; Litchfield, J.; Goosen, T.C.; El-Kattan, A.F. pH-sensitive interaction of HMG-CoA reductase inhibitors (Statins) with organic anion transporting polypeptide 2B1. Molecular Pharmaceutics 2011, 8, 1303–1313.
   PubMed Web of Science ®Google Scholar
• Leal-Calderon, F.; Schmitt, V.; Bibette, J. Emulsion Science: Basic Principles, 2nd Edn. Springer: New York, 2007.
   Google Scholar
• Qi, X.; Wang, L.; Zhu, J. Water-in-oil-in-water double emulsions: An excellent delivery system for improving oral bioavailability of pidotimod in rats. Journal of Pharmaceutical Sciences 2011, 100, 2203–2211.
   PubMed Web of Science ®Google Scholar
• Pulido, A.; Beristain, C.I. Spray-dried encapsualtion of ascorbic acid using chitosan as wall material. Revista Mexicana de Ingeniería Química 2010, 9, 189–195.
   Web of Science ®Google Scholar
• Vlaia, L.; Vlaia, V.; Miclea, L.M.; Olariu, I.; Coneac, G. Topical W/O/W double emulsions of Piroxicam: In vitro drug release study. Farmacia 2009, 57, 639–647.
   Web of Science ®Google Scholar
• Oster, C.G.; Kissel, T. Comparative study of DNA encapsulation into PLGA microparticles using modified double emulsion methods and spray drying techniques. Journal of Microencapsulation 2005, 22, 235–244.
   PubMed Web of Science ®Google Scholar
• Ré, M.I. Formulating drug delivery system by spray drying. Drying Technology 2006, 24, 433–446.
   Web of Science ®Google Scholar
• Passerini, N.; Calogerà, G.; Albertini, B.; Rodriguez, L. Melt granulation of pharmaceutical powders: A comparison of high-shear mixer and fluidised bed processes. International Journal of Pharmaceutics 2010, 391, 177–186.
   PubMed Web of Science ®Google Scholar
• Schilling, S.U.; McGinity, J.W. Novel application of hot-melt extrusion for the preparation of monolithic matrices containing enteric-coated particles. International Journal of Pharmaceutics 2010, 400, 24–31.
   PubMed Web of Science ®Google Scholar
• Wagdare, N.A.; Marcelis, A.T.M.; Boom, R.M.; van Rijn, C.J.M. Porous microcapsule formation with microsieve emulsification. Journal of Colloid and Interface Science 2011, 355, 453–457.
   PubMed Web of Science ®Google Scholar
• Dzul-Cauich, J.G.; Lobato-Calleros, C.; Pérez-Orozco, J.P.; Alvarez-Ramirez, J.; Vernon-Carter, E.J. Stability of water-in-oil-in-water multiple emulsions: Influence of the interfacial properties of milk fat globule membrane. Revista Mexicana de Ingeniería Química 2013, 12, 425–436.
   Web of Science ®Google Scholar
• Carrillo-Navas, H.; González-Rodea, D.A.; Cruz-Olivares, J.; Barrera-Pichardo, J.F.; Román-Guerrero, A.; Pérez-Alonso, C. Storage stability and physicochemical properties of passion fruit juice microcapsules by spray-drying. Revista Mexicana de Ingeniería Química 2011, 10, 421–430.
   Web of Science ®Google Scholar
• Sánchez-Sáenz, E.O.; Pérez-Alonso, C.; Cruz-Olivares, J.; Román-Guerrero, A.; Baéz-González, J.G.; Rodríguez-Huezo, M.E. Establishing the most suitable storage conditions for microencapsulated Allspice essential oil entrapped in blended biopolymers matrices. Drying Technology 2011, 29(8), 863–872.
   Web of Science ®Google Scholar
• Adamiec, J.; Borompichaichartkul, C.; Srzednicki, G.; Panket, W.; Piriyapunsakul, S.; Zhao, J. Microencapsulation of Kaffir lime oil and its functional properties. Drying Technology 2012, 30(9), 914–920.
   Web of Science ®Google Scholar
• Kowalski, J.; Kalb, O.; Joshi, Y.M.; Serajuddin, A.T.M. Application of melt granulation technology to enhance stability of a moisture sensitive immediate-release drug product. International Journal of Pharmaceutics 2009, 381, 56–61.
   PubMed Web of Science ®Google Scholar
• Cortés-Rojas, D.F.; Oliveira, W.P. Physicochemical properties of phytopharmaceutical preparations as affected by drying methods and carriers. Drying Technology 2012, 30(9), 921–934.
   Web of Science ®Google Scholar
• Lobato-Calleros, C.; Sosa-Pérez, A.; Rodríguez-Tafoya, J.; Sandoval-Castilla, O.; Pérez-Alonso, C.; Vernon-Carter, E.J. Structural and textural characteristics of reduced-fat cheese-like products made from W1/O/W2 emulsions and skim milk. LWT Food Science and Technology 2008, 41, 1847–1856.
   Web of Science ®Google Scholar
• Lobato-Calleros, C.; Rodriguez, E.; Sandoval-Castilla, O.; Vernon-Carter, E.J.; Alvarez-Ramirez, J. Reduced-fat white fresh cheese-like products obtained from W1/O/W2 multiple emulsions: Viscoelastic and high-resolution image analyses. Food Research International 2006, 39, 678–685.
   Web of Science ®Google Scholar
• Quintanilla-Carvajal, M.X.; Meraz-Torres, L.S.; Alamilla-Beltrán, L.; Chanona-Pérez, J.J.; Terres-Rojas, E.; Hernández-Sánchez, H.; Jiménez-Aparicio; A.R.; Gutiérrez-López, G.F. Morphometric characterization of spray-dried microcapsules before and after α -tocopherol extraction. Revista Mexicana de Ingeniería Química 2011, 10, 301–312.
   Web of Science ®Google Scholar
• Naeem-Aamir, M.; Ahmad, M.; Akhtar, N.; Murtaza, G.; Khan, S.A.; Shahiq-uz-Zaman; Nokhodchi, A. Development and in vitro–in vivo relationship of controlled-release microparticles loaded with tramadol hydrochloride. International Journal of Pharmaceutics 2011, 407, 38–43.
   PubMed Web of Science ®Google Scholar
• ICH. Stability testing of new drug substances and products Q1A(R2). Q1A(R2), quality guidelines. In International Conference on Harmonization, Geneva, Switzerland, 2006, 1–18.
   Google Scholar
• Pérez-Alonso, C.; Cruz-Olivares, J.; Barrera-Pichardo, J.F.; Rodríguez-Huezo, M.E.; Báez-González, J.G.; Vernon-Carter, E.J. DSC thermo-oxidative stability of red chili oleoresin microencapsulated in blended biopolymers matrices. Journal of Food Engineering 2008, 85, 613–624.
   Web of Science ®Google Scholar
• Pu, J.; Bankston, J.D.; Sathivel, S. Production of microencapsulated crawfish (Procambarus clarkii) astaxanthin in oil by spray drying technology. Drying Technology 2011, 29(10), 1150–1160.
   Web of Science ®Google Scholar
• Alhnan, M.A.; Kidia, E.; Basit, A.W. Spray-drying enteric polymers from aqueous solutions: A novel, economic, and environmentally friendly approach to produce pH-responsive microparticles. European Journal of Pharmaceutics and Biopharmaceutics 2011, 79, 432–439.
   PubMed Web of Science ®Google Scholar
• Albertini, B.; Passerini, N.; Gonzalez-Rodriguez, M.L.; Cavallari, C.; Cini, M.; Rodriguez, L. Wet granulation as innovative and fast method to prepare controlled release granules based on an ion-exchange resin. Journal of Pharmaceutical Sciences 2008, 97, 1313–1324.
   PubMed Web of Science ®Google Scholar
• Borini, G.B.; Andrade, T.C.; Freitas, L.A.P. Hot melt granulation of coarse pharmaceutical powders in a spouted bed. Powder Technology 2009, 189, 520–527.
   Web of Science ®Google Scholar
• Hu, R.; Zhu, J.; Chen, G.; Sun, Y.; Li, M.; Li, S. Preparation of sustained-release simvastatin microspheres by the spherical crystallization technique. Asian Journal of Pharmaceutical Sciences 2006, 1, 47–52.
   Google Scholar
• Albertini, B.; Cavallari, C.; Passerini, N.; Voinovich, D.; Gonzalez-Rodriguez, M.L.; Magarotto, L.; Rodriguez, L. Characterization and taste-masking evaluation of acetaminophen granules: Comparison between different preparation methods in a high-shear mixer. European Journal of Pharmaceutical Sciences 2004, 21, 295–303.
   PubMed Web of Science ®Google Scholar
• Martins, R.M.; Machado, M.O.; Pereira, S.V.; Nosari, A.B.F.L.; Tacon, L.A.; Freitas, L.A.P. Microparticulated hydrochlorothiazide solid dispersion: Enhancing dissolution properties via spray drying. Drying Technology 2012, 30(9), 956–967.
   Google Scholar
• Nerkar, P.; Gattani, S. Spray-dried buccal mucoadhesive microparticles of venlafaxine based on cress seed mucilage: In vitro, in vivo evaluation in rabbits. Drying Technology 2012, 30(9), 968–978.
   Web of Science ®Google Scholar
• Schoubben, A.; Blasi, P.; Giovagnoli, S.; Perioli, L.; Rossi, C.; Ricci, M. Novel composite microparticles for protein stabilization and delivery. European Journal of Pharmaceutical Sciences 2009, 36, 226–234.
   PubMed Web of Science ®Google Scholar
• Hamedelniel, E.I.; Bajdik, J.; Sovány, T.; Pintye-Hódi, K. Delayed release matrix pellet preparation containing an alkalizing pore-former agent. Chemical Engineering Research and Design 2011, 89, 1006–1010.
   Web of Science ®Google Scholar
• Jeong, S.H.; Park, K. Development of sustained release fast-disintegrating tablets using various polymer-coated ion-exchange resin complexes. International Journal of Pharmaceutics 2008, 353, 195–204.
   PubMed Web of Science ®Google Scholar