Application of a three-fluid nozzle for the preparation of amorphous solid dispersions

References

• Percy, S. Improvement in Drying and Concentrating of Liquid Substances by Atomizing. 125.406. USA, 1872.
   Google Scholar
• Shirkole, S. S. A Bibliometric Analysis of Publications in Drying Technology in Selected Drying Areas. Drying Technol. 2020, 38, 2115–2117. DOI: 10.1080/07373937.2020.1834260.
   Web of Science ®Google Scholar
• Deshmukh, R.; Wagh, P.; Naik, J. Solvent Evaporation and Spray Drying Technique for Micro- and Nanospheres/Particles Preparation: A Review. Drying Technol. 2016, 34, 1758–1772. DOI: 10.1080/07373937.2016.1232271.
   Web of Science ®Google Scholar
• Sollohub, K.; Cal, K. Spray Drying Technique: II. Current Applications in Pharmaceutical Technology. J. Pharm. Sci. 2010, 99, 587–597. DOI: 10.1002/jps.21963.
   PubMed Web of Science ®Google Scholar
• Mendonsa, N.; Almutairy, B.; Kallakunta, V. R.; Sarabu, S.; Thipsay, P.; Bandari, S.; Repka, M. A. Manufacturing Strategies to Develop Amorphous Solid Dispersions: An Overview. J. Drug Deliv. Sci. Technol. 2020, 55, 101459. DOI: 10.1016/j.jddst.2019.101459
   Web of Science ®Google Scholar
• Martins, R. M.; Machado, M. O.; Pereira, S. V.; Nosari, A. B. F. L.; Tacon, L. A.; Freitas, L. A. P. Microparticulated Hydrochlorothiazide Solid Dispersion: Enhancing Dissolution Properties via Spray Drying. Drying Technol. 2012, 30, 959–967. DOI: 10.1080/07373937.2011.652268.
   Web of Science ®Google Scholar
• Davis, M.; Walker, G. Recent Strategies in Spray Drying for the Enhanced Bioavailability of Poorly Water-Soluble Drugs. J. Control. Release 2018, 269, 110–127. DOI: 10.1016/j.jconrel.2017.11.005.
   PubMed Web of Science ®Google Scholar
• Taylor, L. S.; Zhang, G. G. Physical Chemistry of Supersaturated Solutions and Implications for Oral Absorption. Array, Ed 2016, 101, 122–142. DOI: 10.1016/j.addr.2016.03.006.
   Google Scholar
• Williams, H. D.; Trevaskis, N. L.; Charman, S. A.; Shanker, R. M.; Charman, W. N.; Pouton, C. W.; Porter, C. J. Strategies to Address Low Drug Solubility in Discovery and Development. Pharmacol. Rev. 2013, 65, 315–499. DOI: 10.1124/pr.112.005660.
   PubMed Web of Science ®Google Scholar
• Frank, K. J.; Rosenblatt, K. M.; Westedt, U.; Holig, P.; Rosenberg, J.; Magerlein, M.; Fricker, G.; Brandl, M. Amorphous Solid Dispersion Enhances Permeation of Poorly Soluble ABT-102: true Supersaturation vs. apparent Solubility Enhancement. Int. J. Pharm. 2012, 437, 288–293. DOI: 10.1016/j.ijpharm.2012.08.014.
   PubMed Web of Science ®Google Scholar
• Mahmah, O.; Tabbakh, R.; Kelly, A.; Paradkar, A. A Comparative Study of the Effect of Spray Drying and Hot-Melt Extrusion on the Properties of Amorphous Solid Dispersions Containing Felodipine. J. Pharm. Pharmacol. 2014, 66, 275–284. DOI: 10.1111/jphp.12099.
   PubMed Web of Science ®Google Scholar
• Cal, K.; Sollohub, K. Spray Drying Technique. I: Hardware and Process Parameters. J. Pharm. Sci. 2010, 99, 575–586. DOI: 10.1002/jps.21886.
   PubMed Web of Science ®Google Scholar
• Caron, V.; Tajber, L.; Corrigan, O. I.; Healy, A. M. A Comparison of Spray Drying and Milling in the Production of Amorphous Dispersions of Sulfathiazole/Polyvinylpyrrolidone and Sulfadimidine/Polyvinylpyrrolidone. Mol. Pharm. 2011, 8, 532–542. DOI: 10.1021/mp1003674.
   PubMed Web of Science ®Google Scholar
• Lavra, Z. M. M.; Pereira de Santana, D.; Ré, M. I. Solubility and Dissolution Performances of Spray-Dried Solid Dispersion of Efavirenz in Soluplus. Drug Dev. Ind. Pharm. 2017, 43, 42–54. DOI: 10.1080/03639045.2016.1205598.
   PubMed Web of Science ®Google Scholar
• Jiang, H.; Zhang, M.; McKnight, S.; Adhikari, B. Microencapsulation of α-Amylase by Carrying out Complex Coacervation and Drying in a Single Step Using a Novel Three-Fluid Nozzle Spray Drying. Drying Technol. 2013, 31, 1901–1910. DOI: 10.1080/07373937.2013.771365.
   Web of Science ®Google Scholar
• Kauppinen, A.; Broekhuis, J.; Grasmeijer, N.; Tonnis, W.; Ketolainen, J.; Frijlink, H. W.; Hinrichs, W. L. J. Efficient Production of Solid Dispersions by Spray Drying Solutions of High Solid Content Using a 3-Fluid Nozzle. Eur. J. Pharm. Biopharm. 2018, 123, 50–58. DOI: 10.1016/j.ejpb.2017.11.009.
   PubMed Web of Science ®Google Scholar
• Chen, R.; Okamoto, H.; Danjo, K. Particle Design of Indomethacin Using a Four-Fluid-Nozzle Spray-Drying Technique. J. Drug Delivery Sci. Technol. 2007, 17, 129–135. DOI: 10.1016/S1773-2247(07)50020-1.
   Web of Science ®Google Scholar
• Ozeki, T.; Beppu, S.; Mizoe, T.; Takashima, Y.; Yuasa, H.; Okada, H. Preparation of Two-Drug Composite Microparticles to Improve the Dissolution of Insoluble Drug in Water for Use with a 4-Fluid Nozzle Spray Drier. J. Control. Release 2005, 107, 387–394. DOI: 10.1016/j.jconrel.2005.06.012.
   PubMed Web of Science ®Google Scholar
• Schram, C. J.; Taylor, L. S.; Beaudoin, S. P. Influence of Polymers on the Crystal Growth Rate of Felodipine: Correlating Adsorbed Polymer Surface Coverage to Solution Crystal Growth Inhibition. Langmuir 2015, 31, 11279–11287. DOI: 10.1021/acs.langmuir.5b02486.
   PubMed Web of Science ®Google Scholar
• Higashi, K.; Yamamoto, K.; Pandey, M. K.; Mroue, K. H.; Moribe, K.; Yamamoto, K.; Ramamoorthy, A. Insights into Atomic-Level Interaction between Mefenamic Acid and Eudragit EPO in a Supersaturated Solution by High-Resolution Magic-Angle Spinning NMR Spectroscopy. Mol. Pharm. 2014, 11, 351–357. DOI: 10.1021/mp4005723.
   PubMed Web of Science ®Google Scholar
• Hancock, B. C.; Shamblin, S. L.; Zografi, G. Molecular Mobility of Amorphous Pharmaceutical Solids below Their Glass Transition Temperatures. Pharm. Res. 1995, 12, 799–806. DOI: 10.1023/a:1016292416526.
   PubMed Web of Science ®Google Scholar
• Patterson, J. E.; James, M. B.; Forster, A. H.; Rades, T. Melt Extrusion and Spray Drying of Carbamazepine and Dipyridamole with Polyvinylpyrrolidone/Vinyl Acetate Copolymers. Drug Dev. Ind. Pharm. 2008, 34, 95–106. DOI: 10.1080/03639040701484627.
   PubMed Web of Science ®Google Scholar
• Hamzehloo, M.; Karimi, J.; Eghbali, N.; Mirzakhani, M.; Aghapoor, K.; Darabi, H. R. A New Blend of Polymeric Encapsulation of Azithromycin by Spray-Drying with a pH Responsive in Drug Release. Drying Technol. 2017, 35, 1688–1695. DOI: 10.1080/07373937.2016.1269807.
   Web of Science ®Google Scholar
• Martins, R. M.; Machado, M. O.; Pereira, S. V.; Nosari, A. B. F. L.; Tacon, L. A.; Freitas, L. A. P. Engineering Active Pharmaceutical Ingredients by Spray Drying: Effects on Physical Properties and in Vitro Dissolution. Drying Technol. 2012, 30, 905–913. DOI: 10.1080/07373937.2012.679348.
   Web of Science ®Google Scholar
• Grzesiak, A. L.; Lang, M.; Kim, K.; Matzger, A. J. Comparison of the Four Anhydrous Polymorphs of Carbamazepine and the Crystal Structure of Form I. J. Pharm. Sci. 2003, 92, 2260–2271. DOI: 10.1002/jps.10455.
   PubMed Web of Science ®Google Scholar
• Halliwell, R. A.; Bhardwaj, R. M.; Brown, C. J.; Briggs, N. E. B.; Dunn, J.; Robertson, J.; Nordon, A.; Florence, A. J. Spray Drying as a Reliable Route to Produce Metastable Carbamazepine Form IV. J. Pharm. Sci. 2017, 106, 1874–1880. DOI: 10.1016/j.xphs.2017.03.045.
   PubMed Web of Science ®Google Scholar
• Lang, M.; Kampf, J. W.; Matzger, A. J. Form IV of Carbamazepine. J. Pharm. Sci. 2002, 91, 1186–1190. DOI: 10.1002/jps.10093.
   PubMed Web of Science ®Google Scholar
• Lang, M.; Grzesiak, A. L.; Matzger, A. J. The Use of Polymer Heteronuclei for Crystalline Polymorph Selection. J. Am. Chem. Soc. 2002, 124, 14834–14835. DOI: 10.1021/ja0286526.
   PubMed Web of Science ®Google Scholar
• Gover Antoniraj, M.; Maria Leena, M.; Moses, J. A.; Anandharamakrishnan, C. Cross-Linked Chitosan Microparticles Preparation by Modified Three Fluid Nozzle Spray Drying Approach. Int. J. Biol. Macromol. 2020, 147, 1268–1277. DOI: 10.1016/j.ijbiomac.2019.09.254.
   PubMed Web of Science ®Google Scholar
• Shayanfar, A.; Velaga, S.; Jouyban, A. Solubility of Carbamazepine, Nicotinamide and Carbamazepine–Nicotinamide Cocrystal in Ethanol–Water Mixtures. Fluid Phase Equilib. 2014, 363, 97–105. DOI: 10.1016/j.fluid.2013.11.024.
   Web of Science ®Google Scholar
• Healthcare, E. d f t q o m a. Pharmacopoeia European monography carbamazepinum; ISBN 978-3-7692-7515-5; 2020; pp 3122–3124.
   Google Scholar
• Li, N.; Gilpin, C. J.; Taylor, L. S. Understanding the Impact of Water on the Miscibility and Microstructure of Amorphous Solid Dispersions: An AFM-LCR and TEM-EDX Study. Mol. Pharm. 2017, 14, 1691–1705. DOI: 10.1021/acs.molpharmaceut.6b01151.
   PubMed Web of Science ®Google Scholar
• Paudel, A.; Worku, Z. A.; Meeus, J.; Guns, S.; Van den Mooter, G. Manufacturing of Solid Dispersions of Poorly Water Soluble Drugs by Spray Drying: Formulation and Process Considerations. Int. J. Pharm. 2013, 453, 253–284. DOI: 10.1016/j.ijpharm.2012.07.015.
   PubMed Web of Science ®Google Scholar
• Malzert-Freon, A.; Benoit, J. P.; Boury, F. Interactions between Poly(Ethylene Glycol) and Protein in Dichloromethane/Water Emulsions: A Study of Interfacial Properties. Eur. J. Pharm. Biopharm. 2008, 69, 835–843. DOI: 10.1016/j.ejpb.2008.01.021.
   PubMed Web of Science ®Google Scholar
• Kolter, K.; K, M.; Gryczke, A. Hot-Melt Extrusion with BASF Pharma Polymers Extrusion Compedium, 2012.
   Google Scholar
• Malwade, C. R.; Qu, H.; Rong, B.-G.; Christensen, L. P. Evaporative Crystallization of Carbamazepine from Different Organic Solvents. In 20th International Workshop on Industrial Crystallization, Syddansk Universitetsforlag, Odense Danmark, 2013; pp 364–371.
   Google Scholar