Synthesis and Anti-Tubercular Screening of 8-Benzyloxy-5-[2-(Substituted-Phenyl)-Thiazol-4-yl]-1H-Quinolin-2-One Derivatives

References

• Ragnhild Münch, “Robert Koch,” Microbes and Infection 5, no. 1 (2003): 69–74.
   PubMed Web of Science ®Google Scholar
• Stefan H.E. Kaufmann, “A Short History of Robert Koch’s Fight against Tuberculosis: Those Who Do Not Remember the past Are Condemned to Repeat It,” Tuberculosis 83, no. 1–3 (2003): 86–90.
   PubMed Web of Science ®Google Scholar
• Marcus Vinícius Nora de Souza, and Thatyana Rocha Alves Vasconcelos, “Fármacos No Combate à Tuberculose: Passado, Presente e Futuro,” Química Nova 28, no. 4 (2005): 678–82.
   Google Scholar
• Marcus V.N. De Souza, Thatyana R.A. Vasconcelos, Mauro V.D. Almeida, and Silvia H. Cardoso, “Fluoroquinolones: An Important Class of Antibiotics against Tuberculosis,” Current Medicinal Chemistry 13, no. 4 (2006): 455–63.
   PubMed Web of Science ®Google Scholar
• Sevim Rollas and Ş. Güniz. Küçükgüzel, “Biological Activities of Hydrazone Derivatives,” Molecules (Basel, Switzerland) 12, no. 8 (2007): 1910–39.
   PubMed Web of Science ®Google Scholar
• Ameya A. Chavan and Nandini R. Pai, “Synthesis and Antimicrobial Screening of 5-Arylidene-2-Imino-4-Thiazolidinones,” Arkivoc 2007, no. 16 (2007): 148–55.
   Google Scholar
• Geoffrey Wells, Tracey D. Bradshaw, Patrizia Diana, Angela Seaton, Dong-Fang Shi, Andrew D. Westwell, and Malcolm F. G. Stevens, “Antitumour Benzothiazoles. Part 10: The Synthesis and Antitumour Activity of Benzothiazole Substituted Quinol Derivatives,” Bioorganic & Medicinal Chemistry Letters 10, no. 5 (2000): 513–5.
   PubMed Web of Science ®Google Scholar
• Atsushi Satoh, Yasushi Nagatomi, Yukari Hirata, Satoru Ito, Gentaroh Suzuki, Toshifumi Kimura, Shunsuke Maehara, Hirohiko Hikichi, Akio Satow, Mikiko Hata, et al, “Discovery and in Vitro and in Vivo Profiles of 4-fluoro-N-[4-[6-(Isopropylamino) Pyrimidin-4-yl]-1, 3-Thiazol-2-yl]-N-Methylbenzamide as Novel Class of an Orally Active Metabotropic Glutamate Receptor 1 (mGluR1) Antagonist,” Bioorganic & Medicinal Chemistry Letters 19, no. 18 (2009): 5464–8.
   PubMed Web of Science ®Google Scholar
• Nadeem Siddiqui and Waquar Ahsan, “Synthesis, Anticonvulsant and Toxicity Screening of Thiazolyl–Thiadiazole Derivatives,” Medicinal Chemistry Research 20, no. 2 (2011): 261–8.
   Web of Science ®Google Scholar
• Shashikant R. Pattan, Ch Suresh, V.D. Pujar, V.V.K. Reddy, V.P. Rasal, and Basavaraj C. Koti, “Synthesis and Antidiabetic Activity of 2-Amino [5'(4-Sulphonylbenzylidine)-2, 4-Thiazolidinedione]-7-Chloro-6-Fluorobenzothiazole,” Indian Journal of Chemistry Section B: Organic Chemistry Including Medicinal Chemistry 44 (2005): 2404–8.
   Google Scholar
• Mayura S. Pingle, Sambhaji P. Vartale, Vijay N. Bhosale, and Sharad V. Kuberkar, “A Convenient Synthesis of 3-Cyano-4-Imino-2-Methylthio-4H-Pyrimido [2, 1-b][1, 3] Benzothiazole and Its Reactions with Selected Nucleophiles,” Arkivoc 2006, no. 10 (2006): 190–8.
   Google Scholar
• Devendra S. Wagare, Prashant D. Netankar, Mujahed Shaikh, Mazahar Farooqui, and Ayesha. Durrani, “Highly Efficient Microwave-Assisted One-Pot Synthesis of 4-Aryl-2-Aminothiazoles in Aqueous Medium,” Environmental Chemistry Letters 15, no. 3 (2017): 475–9.
   Web of Science ®Google Scholar
• H.I. El-Subbagh, and A.M. Al-Obaid, “2, 4-Disubstituted Thiazoles II. A Novel Class of Antitumor Agents, Synthesis and Biological Evaluation,” European Journal of Medicinal Chemistry 31, no. 12 (1996): 1017–21.
   Web of Science ®Google Scholar
• Tukaram S. Choudhare, Devendra S. Wagare, Vijay T. Kadam, Ajit A. Kharpe, and Prashant D. Netankar, “Rapid One-Pot Multicomponent Dioxane-HCl Complex Catalyzed Solvent-Free Synthesis of 3,4-Dihydropyrimidine-2-One Derivatives,” Polycyclic Aromatic Compounds 42, no. 6 (2022): 3865–73.
   Web of Science ®Google Scholar
• Y. Sindhu, C.J. Athira, M.S. Sujamol, and K. Mohanan, “Synthesis, Characterization, and Antibacterial Studies of Oxovanadium (IV) Complexes with Thiazole-Derived Schiff Bases,” Phosphorus, Sulfur, and Silicon 185, no. 9 (2010): 1955–63.
   Web of Science ®Google Scholar
• Daniele Castagnolo, Mafalda Pagano, Martina Bernardini, and Maurizio Botta, “Domino Alkylation-Cyclization Reaction of Propargyl Bromides with Thioureas/Thiopyrimidinones: A New Facile Synthesis of 2-Aminothiazoles and 5H-Thiazolo[3,2-a]Pyrimidin-5-Ones,” Synlett 2009, no. 13 (2009): 2093–6.
   Google Scholar
• Tukaram S. Choudhare, Devendra S. Wagare, Sagar E. Shirsath, and Prashant D. Netankar, “H3PO4 Catalyzed One-Pot Synthesis of 1,3-Diphenyl-1H-Pyrazole-4-Carbaldehyde to Novel 1,3-Diphenyl-1H-Pyrazole-4-Carbonitrile,” Journal of Chemical Sciences 133, no. 3 (2021): 69.
   Web of Science ®Google Scholar
• Bhaskar S. Dawane, Shankaraiah G. Konda, Vinod T. Kamble, Sanjay A. Chavan, Raghunath B. Bhosale, and Shaikh Baseer M, “Multicomponent One-Pot Synthesis of Substituted Hantzsch Thiazole Derivatives under Solvent Free Conditions,” E-Journal of Chemistry 6, no. S1 (2009): S358–S362.
   Google Scholar
• Majid M. Heravi, Nargess Poormohammad, Yahia S. Beheshtiha, and Bita Baghernejad, “Efficient Synthesis of 2, 4-Disubstituted Thiazoles under Grinding,” Synthetic Communications 41, no. 4 (2011): 579–82.
   Web of Science ®Google Scholar
• Tukaram S. Choudhare, Devendra S. Wagare, Vasant B. Jagrut, and Prashant D. Netankar, “Three Component One-Pot Synthesis of Novel 8-Benzyloxy-5-{2-[N′-(1,3-Diphenyl-1H-Pyrazol-4-Ylmethylene)-Hydrazino]-Thiazol-4-yl}-3,4-Dihydro-1H-Quinolin-2-Ones,” Polycyclic Aromatic Compound 43, 2672–9.
   Web of Science ®Google Scholar
• Santosh Raut, Bharat Dhotre, Atul Tidke, and Mohammad A. Pathan, “An Operationally Simple and Efficient Synthesis of 7-Benzylidene-Substitutedphenyl-3, 3a, 4, 5, 6, 7-Hexahydro-2H-Indazole by Grinding Method,” Current Organic Synthesis 17, no. 4 (2020): 313–21.
   PubMed Web of Science ®Google Scholar
• Javad Safari, Zahra Abedi-Jazini, Zohre Zarnegar, and Masoud Sadeghi, “Nanochitosan: A Biopolymer Catalytic System for the Synthesis of 2-Aminothiazoles,” Catalysis Communications 77 (2016): 108–12.
   Web of Science ®Google Scholar
• Tukaram S. Choudhare, Devendra S. Wagare, Vijay T. Kadam, and Prashant D. Netankar, “Synthesis and Microbial Screening of 8-(Benzyloxy)-5-(2-[1,3-Diphenyl-1H-Pyrazol-4-yl]Thiazol-4-yl)Quinolin-2(1H)-One Derivatives,” Journal of Heterocyclic Chemistry 58, no. 8 (2021): 1637–44.
   Web of Science ®Google Scholar
• Gareth J. Rowlands, Rebecca J. Severinsen, Jenna K. Buchanan, Karl J. Shaffer, Heather T. Jameson, Nishani Thennakoon, Ivo Leito, Märt Lõkov, Agnes Kütt, Robert Vianello, et al, “Synthesis and Basicity Studies of Quinolino [7, 8-h] Quinoline Derivatives,” The Journal of Organic Chemistry 85, no. 17 (2020): 11297–308.
   PubMed Web of Science ®Google Scholar
• Ida Boček, Marijana. Hranjec, and Robert. Vianello, “Imidazo [4, 5-b] Pyridine Derived Iminocoumarins as Potential pH Probes: Synthesis, Spectroscopic and Computational Studies of Their Protonation Equilibria,” Journal of Molecular Liquids 355 (2022): 118982.
   Web of Science ®Google Scholar
• Tukaram S. Choudhare, Devendra S. Wagare, Vasant B. Jagrut, and Prashant D. Netankar, “Three Component One-Pot Synthesis of Novel 8-Benzyloxy-5-{2-[N′-(1, 3-Diphenyl-1 H-Pyrazol-4-Ylmethylene)-Hydrazino]-Thiazol-4-yl}-3, 4-Dihydro-1 H-Quinolin-2-Ones,” Polycyclic Aromatic Compounds 43, no. 3 (2022): 1–8.
   Google Scholar
• J.S.V. Soundarya, Uma Devi. Ranganathan, and Srikanth P. Tripathy, “Current Trends in Tuberculosis Vaccine,” Medical Journal, Armed Forces India 75, no. 1 (2019): 18–24.
   PubMedGoogle Scholar
• A.K. Njoku, “Tuberculosis: Current Trends in Diagnosis and Treatment,” Nigerian Journal of Clinical Practice 8, no. 2 (2005): 118–24.
   PubMedGoogle Scholar