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Phosphorus, Sulfur, and Silicon and the Related Elements Volume 194, 2019 - Issue 4-6: Proceedings of the 2018 International Conference on Phosphorus Chemistry, ICPC-22
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Short Communication

Rational synthesis of α-hydroxyphosphonic derivatives including dronic acids

Alajos GrünDepartment of Organic Chemistry and Technology, Budapest University of Technology and Economics, Budapest, Hungary; Correspondence[email protected]
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,
Zita RádaiDepartment of Organic Chemistry and Technology, Budapest University of Technology and Economics, Budapest, Hungary; View further author information
,
Dávid Illés Sőregi-NagyDepartment of Organic Chemistry and Technology, Budapest University of Technology and Economics, Budapest, Hungary; View further author information
,
István GreinerGedeon Richter Plc, Budapest, HungaryView further author information
&
György KeglevichDepartment of Organic Chemistry and Technology, Budapest University of Technology and Economics, Budapest, Hungary; View further author information
Pages 386-387 | Received 28 Sep 2018, Accepted 30 Nov 2018, Published online: 09 Jan 2019

References

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  • Keglevich, G.; Rádai, Z.; Kiss, N. Z. To Date the Greenest Method for the Preparation of α-Hydroxyphosphonates from Substituted Benzaldehydes and Dialkyl Phosphites. Green Process. Synth. 2017, 6, 197–201.
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  • Nagy, D. I.; Grün, A.; Pavela, O.; Garadnay, S.; Greiner, I.; Keglevich, G. Efficient Synthesis of Ibandronate in the Presence of an Ionic Liquid. Lett. Drug. Des. Disc. 2018, 15,713–720. DOI:10.2174/1570180814666171027160324.
  • Nagy, D. I.; Grün, A.; Lévay, K.; Garadnay, S.; Greiner, I.; Keglevich, G. Efficient Syntheses of Zoledronic Acid as an Active Ingredient of a Drug against Osteoporosis. Synt. Comm. 2018, 48, 663–671. DOI:10.1080/00397911.2017.1410894.
  • Nagy, D. I.; Grün, A.; Sinkovicz, J.; Garadnay, S.; Greiner, I.; Keglevich, G. A Study on the Synthesis of Risedronic Acid; The Role of an Ionic Liquid Additive. Lett. Drug. Des. Disc. 2019, 16, in press.

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