Lecithin-Based Microemulsion of a Peptide for Oral Administration: Preparation, Characterization, and Physical Stability of the Formulation

REFERENCES

• Aboofazeli R., Lawrence M. J. Investigations into the formation and characterization of phospholipid microemulsions. I. Pseudo-ternary phase diagrams of systems containing water-lecithin-alcohol-isopropyl myristate. Int. J. Pharm 1993; 93: 161–175, [CSA]
   Web of Science ®Google Scholar
• Aboofazeli R., Lawrence M. J. Investigations into the formation and characterization of phospholipid microemulsions. II. Pseudo-ternary phase diagrams of systems containing water-lecithin-isopropyl myristate and alcohol: influence of purity of lecithin. Int. J. Pharm 1994a; 106: 51–61, [CROSSREF], [CSA]
   Web of Science ®Google Scholar
• Aboofazeli R., Lawrence C. B., Wicks S. R., Lawrence M. J. Investigations into the formation and characterization of phospholipid microemulsions. III. Pseudo-ternary phase diagrams of systems containing water-lecithin-isopropyl myristate and either an alkanoic acid, amine, alkanediol, polyethylene glycol alkyl ether or alcohol as cosurfactant. Int. J. Pharm 1994b; 111: 63–72, [CROSSREF], [CSA]
   Web of Science ®Google Scholar
• Aboofazeli R., Patel N., Thomas M., Lawrence M. J. Investigations into the formation and characterization of phospholipid microemulsions. IV. Pseudo-ternary phase diagrams of systems containing water-lecithin-alcohol and oil. Int. J. Pharm 1995; 125: 107–116, [CROSSREF], [CSA]
   Web of Science ®Google Scholar
• Attwood D., Mallon C., Taylor C. J. Phase studies on oil-in-water phospholipid microemulsions. Int. J. Pharm. 1992; 84: R5–R8, [CROSSREF], [CSA]
   Web of Science ®Google Scholar
• Bagve R. P., Kanicky J. R., Palla B. J., Patanjali P. K., Shah D. O. Improved drug delivery using microemulsions: rationale, recent progress, and new horizons. Crit. Rew. Ther. Drug Carr. Sys. 2001; 18: 77–140, [CSA]
   PubMed Web of Science ®Google Scholar
• Baker R. C., Florence A. T., Ottewill R. H., Tadros T. F. Investigations into the formation and characterization of microemulsions: 2. Light scattering conductivity and viscosity studies of microemulsions. J. Colloid Interface Sci 1984; 100: 332–349, [CSA]
   Web of Science ®Google Scholar
• Bhargava H. N., Narurkar A., Lieb L. M. Using microemulsions for drug delivery. Pharm. Technol. 1987; 11: 46–52, [CSA]
   Google Scholar
• Brime B., Moreno M. A., Frutos G., Ballesteros P., Frutos P. Amphotericin B in oil-water lecithin-based microemulsions: formulation and toxicity evaluation. J. Pharm. Sci. 2002; 91: 1178–1185, [PUBMED], [INFOTRIEVE], [CROSSREF], [CSA]
   PubMed Web of Science ®Google Scholar
• Constantinides P. P. Lipid microemulsions for improving drug dissolution and oral absorbsion: physical and biopharmaceutical aspects. Pharm. Res. 1995; 12: 1561–1572, [PUBMED], [INFOTRIEVE], [CROSSREF], [CSA]
   PubMed Web of Science ®Google Scholar
• Constantinides P. P., Scalart J. P. Formulation and physical characterization of water-in-oil microemulsions containing long-versus medium-chain glycerides. Int. J. Pharm. 1997; 158: 57–68, [CROSSREF], [CSA]
   Web of Science ®Google Scholar
• Çilek A., Çelebi N., Ocak F., Tay A. Oral absorption of recombinant insulin from microemulsion in rats. EUFEPS World Conference on Drug Absorption and Drug Delivery Benefiting from the New Biology and Informatics, CopenhagenDenmark, June, 18–20, 2001, Proceedings, Abstracts, 81, 82
   Google Scholar
• Fletcher P. D. I., Morris J. S. Turbidity of oil-in-water microemulsion droplets stabilized by nonionic surfactants. Colloids Surfaces A: Physicochemi Engi Aspects 1995; 98: 147–154, [CROSSREF], [CSA]
   Web of Science ®Google Scholar
• Ho H. O., Hsiao C. C., Sheu M. T. Preparation of microemulsions using polyglycerol fatty acid esters as surfactant for the delivery of protein drugs. J. Pharm. Sci. 1996; 85: 138–143, [PUBMED], [INFOTRIEVE], [CROSSREF], [CSA]
   PubMed Web of Science ®Google Scholar
• Ktistis G. Viscosity study on oil-in water microemulsions. Int. J. Pharm. 1990; 61: 213–218, [CROSSREF], [CSA]
   Web of Science ®Google Scholar
• Lawrence M. J., Rees G. D. Microemulsion-based media as novel drug delivery systems. Adv. Drug Del. Rev. 2000; 45: 89–121, [CROSSREF], [CSA]
   PubMed Web of Science ®Google Scholar
• Paolino D., Ventura C. A., Nistico S., Puglisi G., Fresta M. Lecithin microemulsions for the topical administration of ketoprofen: percutaneous adsorption through human skin and in vivo human skin tolerability. Int. J. Pharm. 2002; 244: 21–31, [PUBMED], [INFOTRIEVE], [CROSSREF], [CSA]
   PubMed Web of Science ®Google Scholar
• Park K. M., Lee M. K., Hwang K. J., Kim C. K. Phospholipid-based microemulsions of flurbiprofen by the spontaneous emulsification process. Int. J. Pharm. 1999; 183: 145–154, [PUBMED], [INFOTRIEVE], [CROSSREF], [CSA]
   PubMed Web of Science ®Google Scholar
• Radomska A., Dobrucki R. The use of some ingredients for microemulsion preparation containing retinol and its esters. Int. J. Pharm. 2000; 196: 131–134, [PUBMED], [INFOTRIEVE], [CROSSREF], [CSA]
   PubMed Web of Science ®Google Scholar
• Ritschel W. A. Microemulsions for improved peptide absorption from the gastrointestinal tract. Meth. Find. Exp. Clin. Pharmacol. 1991; 13: 205–220, [CSA]
   PubMed Web of Science ®Google Scholar
• Ruth H. S., Attwood D., Ktistis G., Taylor C. J. Phase studies and particle size analysis of oil-in-water phospholipid microemulsions. Int. J. Pharm. 1995; 116: 253–261, [CROSSREF], [CSA]
   Web of Science ®Google Scholar
• Sarciaux J. M., Acar L., Sado P. A. Using microemulsion formulations for oral drug delivery of therapeutic peptides. Int. J. Pharm. 1995; 120: 127–136, [CROSSREF], [CSA]
   Web of Science ®Google Scholar
• Shinoda K., Araki M., Sadaghiani A., Khan A., Lindman B. Lecithin-based microemulsions: phase behaviour and microstructure. J. Phys. Chem. 1991; 95: 989–993, [CROSSREF], [CSA]
   Web of Science ®Google Scholar
• Tenjarla S. Microemulsions: an overview and pharmaceutical applications. Crit. Rev. Ther. Drug Carr. Sys. 1999; 16: 461–521, [CSA]
   PubMed Web of Science ®Google Scholar
• Trotta M., Pattarino F., Grosa G. Formulation of lecithin-based microemulsions containing n-alkanol phosphocholines. Int. J. Pharm. 1998; 174: 253–259, [CROSSREF], [CSA]
   Web of Science ®Google Scholar
• Türkyílmaz A., Çelebi N., Gönül B., Alkan-Önyüksel H. Physical characterization and stability of a microemulsion for potential oral administration of a peptide. Biomedical Science and Technology, A. Híncal, S. Kaş. Plenum Press, New York 1998; 65–72
   Google Scholar