HPTLC METHOD FOR DETERMINATION OF DARUNAVIR IN RAT PLASMA AND ITS APPLICATION IN PHARMACOKINETIC STUDIES

REFERENCES

• Koh , Y. ; Nakata , H. ; Maeda , K. ; Ogata , H. ; Bilcer , G. ; Devasamudram , T. ; Kincaid , J. F. ; Boross , P. ; Wang , Y. F. ; Tie , Y. ; Volarath , P. ; Gaddis , L. ; Harrison , R. W. ; Weber , I. T. ; Ghosh , A. K. ; Mitsuya , H. Novel Bis-tetrahydrofuranylurethane-containing Nonpeptidic Protease Inhibitor (PI) UIC-94017 (TMC114) with Potent Activity against Multi-PI-resistant Human Immunodeficiency Virus in vitro . Antimicrob. Agents Chemother. 2003 , 47 , 3123 – 3129 .
   PubMed Web of Science ®Google Scholar
• De Meyer , S. ; Azijn , H. ; Surleraux , D. ; Jochmans , D. ; Tahri , A. ; Pauwels , R. ; Wigerinck , P. ; de Bethune , M. P. TMC114, A Novel Human Immunodeficiency Virus Type 1 Protease Inhibitor Active Against Protease Inhibitor-Resistant Viruses, Including a Broad Range of Clinical Isolates. Antimicrob. Agents Chemother. 2005, 49, 2314–2321.
   PubMed Web of Science ®Google Scholar
• Tie , Y. ; Boross , P. I. ; Wang , Y. F. ; Gaddis , L. ; Hussain , A. K. ; Leshchenko , S. ; Ghosh , A. K. ; Louis , J. M. ; Harrison , R. W. ; Weber , I. T. High Resolution Crystal Structures of HIV-1 Protease with a Potent Non-peptide Inhibitor (UIC-94017) active Against Multi-Drug-Resistant Clinical Strains . J. Mol. Biol. 2004 , 338 , 341 – 352 .
   PubMed Web of Science ®Google Scholar
• King , N. M. ; Prabu-Jeyabalan , M. ; Nalivaika , E. A. ; Wigerinck , P.; de Bethune M. P. ; Schiffer , C. A. Structural and Thermodynamic Basis for the Binding of TMC114, a Next-Generation Human Immunodeficiency Virus Type 1 Protease Inhibitor . J. Virol. 2004 , 78 , 12012 – 12021 .
   PubMed Web of Science ®Google Scholar
• Poveda , E. ; Blanco , F. ; Garcia-Gasco , P. ; Alcolea , A. ; Briz , V. ; Soriano , V. Successful Rescue Therapy with Darunavir (TMC114) in HIV-infected Patients who have Failed Several Ritonavir-Boosted Protease Inhibitors . AIDS 2006 , 20 , 1558 – 1560 .
   PubMed Web of Science ®Google Scholar
• Kovalevsky , A. Y. ; Tie , Y. ; Liu , F. ; Boross , P. I. ; Wang , Y. F. ; Leshchenko , S. ; Ghosh , A. K. ; Harrison , R. W. ; Weber , I. T. Effectiveness of Nonpeptide Clinical Inhibitor TMC-114 on HIV-1 Protease with Highly Drug Resistant Mutations D30 N, I50 V, and L90 M . J. Med. Chem. 2006 , 49 , 1379 – 1387 .
   PubMed Web of Science ®Google Scholar
• Katlama , C. ; Esposito , R. ; Gatell , J. M. ; Goffard , J. C. ; Grinstein , B. ; Pozniak , A. ; Rockstroh , J. ; Stoehr , A. ; Vetter , N. ; Yeni , P. ; Parys , W. ; Vangeneugden , T. Efficacy and Safety of TMC114/ritonavir in Treatment-Experienced HIV Patients: 24-week Results of Power 1 . AIDS 2007 , 21 , 395 – 402 .
   PubMed Web of Science ®Google Scholar
• Clotet , B. ; Bellos , N. ; Molina , J. M. ; Cooper , D. ; Goffard , J. C. T. ; Hebraic , R. ; Cohen , C. ; Farthing , C. ; Jayaweera , D. ; Markowitz , M. ; Ruane , P. ; Spinosa-Guzman , S. Efebvre , E. Efficacy and Safety of Darunavir-Ritonavir at Week 48 in Treatment-Experienced Patients with HIV-1 infection in POWER 1 and 2: A Pooled Subgroup Analysis of Data from Two Randomised Trials . Lancet 2007 , 369 , 1169 – 1178 .
   PubMed Web of Science ®Google Scholar
• Bouche , M. P. ; Michielsen , L. ; Piot , M. ; Timmerman , P. Swift and Simultaneous Determination of Darunavir (TMC 114) and Ritonavir in Human Plasma using LC-MS/MS. Proc. of the 17th International Mass Spectrometry Conference, Prague, TUP-042, 2006.
   Google Scholar
• Takahashi , M. ; Yoshida , M. ; Oki , T. ; Okumura , N. ; Suzuki , T. ; Kaneda , T. Conventional HPLC Method Used for Simultaneous Determination of the Seven HIV Protease Inhibitors and Nonnucleoside Reverse Transcription Inhibitor Efavirenz in Human Plasma . Biol. Pharm. Bull. 2005 , 28 , 1286 – 1290 .
   PubMed Web of Science ®Google Scholar
• Takahashi , M. ; Yoshida , M. ; Oki , T. ; Okumura , N. ; Suzuki , T. ; Kaneda , T. The Validation of Plasma Darunavir Concentrations Determined by the HPLC Method for Protease Inhibitors . Biol. Pharm. Bull. 2007 , 30 , 1947 – 1949 .
   PubMed Web of Science ®Google Scholar
• Antonio , D. ; Siccardi , M. ; Sciandra , M. ; Lorena , B.; Bonora. S. ; Trentini , L.; Di Perri G. HPLC-MS Method for the Simultaneous Quantification of the New HIV Protease Inhibitor Darunavir, and 11 other Antiretroviral Agents in Plasma of HIV-infected Patients. J. Chromatogr. B. 2007 , 859 , 234 – 240 .
   PubMed Web of Science ®Google Scholar
• Pandya , K. K. ; Mody , V. D. ; Satia , M. C. ; Modi , I. A. ; Modi , R. I. ; Chakravarthy , B. K. ; Gandhi , T. P. High-Performance Thin-Layer Chromatographic Method for the Detection and Determination of Lansoprazole in Human Plasma and its Use in Pharmacokinetic Studies . J. Chromatogr. B. 1997 , 23 , 199 – 204 .
   Web of Science ®Google Scholar