DETERMINATION OF STEREO-SELECTIVE BINDINGS OF RACEMIC PROPRANOLOL WITH β₂-AD-GPCR IN HUMAN PLASMA

REFERENCES

• Basson , M. Cardiovascular Disease . Nat. Med. 2008 , 451 , 903 .
   Web of Science ®Google Scholar
• Meyers , E. H. ; Jawetz , E. ; Goldheim , A. A. Review of Medical Pharmacology Lange Medical Publication : Los Altos , CA , 1980 .
   Google Scholar
• Walle , T. ; Walle , U. K. ; Wilson , M. J. ; Fagan , T. C. ; Gaffney , T. E. Stereoselective Ring Oxidation of Propranolol in Man . Br. J. Clin. Pharmacol. 1984 , 18 , 741 – 748 .
   PubMed Web of Science ®Google Scholar
• Schmid , M. G. ; Gecse , O. ; Szaho , Z. ; Kilar , F. ; Gubitz , G. ; Ali , I. ; Aboul-Enein , H. Y. Comparative Study of the Chiral Resolution of β-blockers on Cellulose tris (3,5-dimethyl-phenylcarbamate) Phases in Normal and Reversed Phase Modes . J. Liq. Chromatogr. Related Technol. 2001 , 24 , 2493 – 2504 .
   Web of Science ®Google Scholar
• Lee , E. J. ; William , K. M. Chirality: Clinical Pharmacokinetic and Pharmacodynamic Considerations . Clin. Pharmacokinet. 1990 , 18 , 339 – 345 .
   PubMed Web of Science ®Google Scholar
• Nelson , W. L. ; Burke , T. R. Jr. Pathways of Propranolol Metabolism. Use of the Stable Isotope Twin-Ion GC-MS Technique to Examine the Conversion of Propranolol to Propranolol-diol by 9000 g Rat Liver Supernatant . Res. Commun. Chem. Pathol. Pharmacol. 1978 , 21 , 77 – 85 .
   PubMedGoogle Scholar
• Barrett , A. M. ; Cullum , V. A. Lack of Inter-action between Propranolol and Mebanazine. J. Pharmacol. 1968, 20, 911–915.
   Google Scholar
• Stevenson , D. ; Wilson , I. D. Chiral Separations , Plenum Press : New York , 1988 .
   Google Scholar
• Balmer , K. ; Lagerstrom , P. O. ; Persson , B. A. ; Schill , G. Reversed Retention Order and other Stereoselective Effects in the Separation of Amino Alcohols on Chiralcel OD . J. Chromatogr. A. 1992 , 592 , 331 – 337 .
   Web of Science ®Google Scholar
• Ram , C. V. Risk of New-Onset Diabetes Mellitus in Patients with Hypertension Treated with Beta Blockers . Amer. J. Cardiol. 2008 , 102 , 242 – 244 .
   PubMed Web of Science ®Google Scholar
• Belknap , S. Beta-blockers for Hypertension Increase Risk of New Onset Diabetes . Evid. Based Med. 2008 , 13 , 50 .
   PubMedGoogle Scholar
• FDA's Policy Statement for the Development of New Stereoisomeric Drugs . Chirality 1992 , 4 , 338 .
   PubMed Web of Science ®Google Scholar
• Aboul-Enein , H. Y. ; Ali , I. Chiral Separation by Liquid Chromatography and Related Technologies , Marcel Dekker Inc. : New York , 2003 .
   Google Scholar
• Cherezov1 , V. ; Rosenbaum , D. M. ; Hanson , M. A. ; Rasmussen , S. G. F. ; Thian , F. S. ; Kobilka , T. S. ; Choi , H. J. ; Kuhn , P. ; Weis , W. I. ; Kobilka , B. K. ; Stevens , R. C. High Resolution Crystal Structure of an Engineered Human β2-adrenergic G protein-Coupled Receptor . Science 2007 , 318 , 1258 – 1265 .
   PubMed Web of Science ®Google Scholar
• Albani , F. ; Riva , R. ; Contin , M. ; Baruzzi , A. Stereoselective Binding of Propranolol Enantiomers to Human α 1-acid Glycoprotein and Human Plasma . Br. J. Clin Pharmacol. 1984 , 18 , 244 – 246 .
   PubMed Web of Science ®Google Scholar
• Lowe , M. D. ; Lynham , J. A. ; Grace , A. A. ; Kauman , A. J. Comparison of the Affinity of Beta Blockers for Two States of the Beta 1-adrenoceptor in Ferret Ventricular Myocardium . Br. J. Pharmacol. 2002 , 135 , 451 – 461 .
   PubMed Web of Science ®Google Scholar
• Rasmussen , S. G. F. ; Choi , H. J. ; Rosenbaum , D. M. ; Kobilka , T. S. ; Thian , F. S. ; Edwards , P. C. ; Burghammer , M. ; Ratnala , V. R. P. ; Sanishvili , R. ; Fischetti , R. F. ; Schertler , G. F. X. ; Weis , W. I. ; Kobilka , B. K. Crystal Structure of the Human β2 Adrenergic G-Protein-Coupled Receptor . Nature 2007 , 450 , 383 – 389 .
   PubMed Web of Science ®Google Scholar
• Nelson , W. L. ; Burke , T. R. Jr. Absolute Configuration of Glycerol Derivatives. 5-oxprenolol enantiomers . J. Org. Chem. 1978 , 43 , 3641 – 3645 .
   Web of Science ®Google Scholar
• Barrett , A. M. ; Cullum , V. A. The Biological Properties of the Optical Isomers of Propranolol and Their Effects on Cardiac Arrhythmias . J. Pharmacol. 1968 , 34 , 43 – 55 .
   Google Scholar
• Danilewicz , J. C. ; Kemp , J. E. G. Absolute Configuration by Asymmetric Synthesis of (+)-1-(4-acetamidophenoxy)-3-(isopropylamino) propan-2-ol) (practolol) . J. Med. Chem. 1973 , 16 , 168 – 169 .
   PubMed Web of Science ®Google Scholar