THE STUDY OF THE LIPOPHILICITY OF NOVEL ANTIBACTERIAL ACTIVE PYRAZOLE DERIVATIVES CONTAINING A CARBOXAMIDE GROUP

REFERENCES

• Yukihito , H. ; Daisuke , J. ; Kazuaki , C. ; Masao , Y. 3-Methyl-1-phenyl-2-pyrazolin-5-one, A Novel Free Radical Scavenger, for Treatment of Cardiovascular Diseases . Recent Pat. Cardiovasc. Drug Discov. 2006 , 1 , 85 – 93 .
   PubMedGoogle Scholar
• Uramaru , N. ; Shigematsu , H. ; Toda , A. ; Eyanagi , R. ; Kitamura , S. ; Ohta , S. Design, Synthesis, and Pharmacological Activity of Nonallergenic Pyrazolone-type Antipyretic Analgesics . J. Med. Chem. 2010 , 53 ( 24 ), 8727 – 8733 .
   PubMed Web of Science ®Google Scholar
• Patel , R. G. ; Patel , C. K. ; Patel , V. I. ; Sen , D. J. ; Panigrahi , B. ; Patel , C. N. Synthesis and Biological Evaluation of Anti-tubercular Activity of Some Synthesized Pyrazole Derivatives . J. Chem. Pharm. Res. 2010 , 2 ( 2 ), 112 – 117 .
   Google Scholar
• Rahimizadeh , M. ; Pordel , M. ; Bakavoli , M. ; Rezaeian , S. ; Sadeghian , A. World J. Microbiol. Biotechnol. 2010, 26, 317–321.
   Web of Science ®Google Scholar
• Gumieniczek , A. ; Berecka , A. ; Matosiuk , D. ; Hopkała , H. Standarized Reversed-Phase Thin-Layer Chromatographic Study of the Lipophilicity of Five Anti-Diabetic Thiazolidinediones . J. Planar Chromatogr.- Mod. TLC 2007 , 20 ( 4 ), 261 – 265 .
   Web of Science ®Google Scholar
• Hansch , C. ; Leo , A. Substituent Constants for Correlation Analysis in Chemistry and Biology , Wiley-Interscience : New York , 1979 .
   Google Scholar
• Margabandu , R. ; Subramani , K. Experimental and Theoretical Study on Lipophilicity and Antibacterial Activity of Biphenylamine Derivatives . Int. J. ChemTech Res. 2010 , 2 ( 3 ), 1501 – 1506 .
   Google Scholar
• Valko , K. Application of High-performance Liquid Chromatography Based Measurements of Lipophilicity to Model Biological Distribution . J. Chromatogr. A 2004 , 1037 , 299 – 310 .
   PubMed Web of Science ®Google Scholar
• Virtual Computational Chemistry Laboratory (http://www.vcclab.org) .
   Google Scholar
• Liu , X. H. ; Cui , P. ; Song , B. A. ; Bhadury , P. S. ; Zhu , H. L. ; Wang , S. F. Synthesis, Structure and Antibacterial Activity of Novel 1-(5-Substituted-3-substituted-4,5-dihydropyrazol-1-yl)ethanone Oxime Ester Derivatives . Bioorg. Med. Chem. 2008 , 16 , 4075 – 4082 .
   PubMed Web of Science ®Google Scholar
• Genin , M. J. ; Biles , C. ; Keiser , B. J. ; Poppe , S. M. ; Swaney , Tarpley; W. G. ; Yagi , Y. ; Romero , D. L. Novel 1,5-Diphenylpyrazole Nonnucleoside HIV-1 Reverse Transcriptase Inhibitors with Enhanced Activity Versus the Delavirdine-resistant P236 L Mutant: Lead Identification and SAR of 3- and 4-Substituted Derivatives . J. Med. Chem. 2000 , 43 , 1034 – 1040 .
   PubMed Web of Science ®Google Scholar
• Wei , F. ; Zhao , B. X. ; Huang , B. ; Zhang , L. ; Sun , C. H. ; Dong , W. L. ; Shin , D. S. Miao , J. Y. Design, Synthesis, and Preliminary Biological Evaluation of Novel Ethyl 1-(2′-hydroxy-3′-aroxypropyl)-3-aryl-1H-pyrazole-5-carboxylate . Bioorg. Med. Chem. Lett. 2006 , 16 , 6342 – 6347 .
   PubMed Web of Science ®Google Scholar
• Pitucha , M. ; Kosikowska , U. ; Mazur , L. ; Malm , A. Synthesis, Structure and Antibacterial Evaluation of Some N-substituted 3-amino-5-hydroxy-4-phenyl-1H-pyrazole-1-carboxamides . Med. Chem. 2011 , 7 , 697 – 703 .
   PubMed Web of Science ®Google Scholar
• Bate-Smith , E. C. ; Westall , R. G. Chromatographic Behavior and Chemical Structure. I. Some Naturally Occurring Phenolic substances . Biochim. Biophys. Acta 1950 , 4 , 427 – 440 .
   Web of Science ®Google Scholar
• Soczewiński , E. ; Wachtmeister , C. A. The Relation Between the Composition of Certain Ternary Two-Phase Solvent Systems and RM Values . J. Chromatogr. 1962 , 7 , 311 – 320 .
   Web of Science ®Google Scholar
• Molinspiration Cheminformatics (http://www.molinspiration.com) .
   Google Scholar
• Pedretti , A. ; Villa , L. ; Vistoli , G. Vega - An Open Platform to Develop Chemo-Bio-Informatics Applications, Using Plug-In Architecture and Script Programming , Journal of Computer-Aided Molecular Design , 2004 , 18 , 167 – 173 .
   PubMed Web of Science ®Google Scholar
• CompuDrug International Inc. 2004. South San Francisco, USA .
   Google Scholar
• Statistica 7.1 2005. StatSoft Inc., Tulsa, OK, USA .
   Google Scholar
• Biagi , G. L. ; Barbaro , A. M. ; Sapone , A. ; Recanatini , M. Determination of Lipophilicity by Means of Reversed-phase Thin-layer Chromatography II. Influence of the Organic Modifier on the Slope of the Thin-layer Chromatographic Equation . J. Chromatogr. A 1994 , 669 , 246 – 253 .
   Web of Science ®Google Scholar
• Taillardat-Bertschinger , A. ; Galland , A. ; Carrupt , P. A. ; Testa , B. Immobilized Artificial Membrane Liquid Chromatography: Proposed Guidelines for Technical Optimization of Retention Measurements . J. Chromatogr. A 2002 , 953 , 39 – 53 .
   PubMed Web of Science ®Google Scholar
• Verma , R. P. ; Hansch , C. An approach Toward the Problem of Outliers in QSAR . Bioorg. Med. Chem. 2005 , 13 ( 15 ), 4597 – 4621 .
   PubMed Web of Science ®Google Scholar
• Hansch , C. ; Garg , R. ; Kurup , B. ; Mekapati , S. B. Allosteric Interactions and QSAR: On the Role of ligand Hydrophobicity . Bioorg. Med. Chem. 2003 , 11 ( 9 ), 2075 – 2084 .
   PubMed Web of Science ®Google Scholar
• Matysiak , J. ; Niewiadomy , A. ; Senczyna , B. ; Żabińska , A. ; Różyło , J. K. Relationships between LC Retention, Octanol-Water Partition Coefficient, and Fungistatic Properties of 2-(2,4-Dihydroxyphenyl)benzothiazoles . J. AOAC Int. 2004 , 87 ( 3 ), 579 – 586 .
   PubMed Web of Science ®Google Scholar
• Rożyło , J. K. ; Matysiak , J. ; Niewiadomy , A. ; Żabinska , A. Reversed-phase HPLC and HPTLC Characterization of Potential Fungicides . J. Planar Chromatogr.-Mod. TLC 2000 , 13 ( 3 ), 176 – 181 .
   Web of Science ®Google Scholar