77
Views
4
CrossRef citations to date
0
Altmetric
Research Article

Agglomeration of celecoxib by quasi-emulsion solvent diffusion method without stabilizer: effect of good solvent

&
Pages 1037-1046 | Received 13 Jul 2016, Accepted 04 Dec 2016, Published online: 12 Jan 2017

References

  • Al-Hamidi H, Edwards AA, Mohammad MA, Nokhodchi A. 2010. Glucosamine HCl as a new carrier for improved dissolution behaviour: effect of grinding. Colloids Surf B. 81:96–109.
  • Beck C, Dalvi SV, Dave RN. 2010. Controlled liquid antisolvent precipitation using a rapid mixing device. Chem Eng Sci. 65:5669–5675.
  • Berkovitch-Yellin Z. 1985. Towards an abinitio derivation of crystal morphology. J Amer Chem Soc. 107:8239–8253.
  • Bhadra S, Kumar M, Jain S, Agrawal S, Agrawal GP. 2004. Spherical crystallization of mefenamic acid. Pharm Tech. 28:66–76.
  • Blandin AF, Mangin D, Rivoire A, Kelin JP, Bossoutrot JM. 2003. Agglomeration in suspension of salicylic acid fine particles: influence of some process parameters on kinetics and agglomerates final size. Powder Technol. 130:316–323.
  • Capes C, Fouda A. 1984. Agglomeration in liquid systems. In: Fayed ME, Otten LP, editors. Handbook of powder science and technology. New York: VanNostrand Reinhold; p. 331–344.
  • Carr RL. 1965a. Classifying flow properties of solids. Chem Eng. 72:69–72.
  • Carr RL. 1965b. Evaluation flow properties of solids. Chem Eng. 72:163–168.
  • Chawla G, Gupta P, Thilagavathi R, Chakraborti AK, Bansal AK. 2003. Characterization of solid-state forms of celecoxib. Eur J Pharm Sci. 20:305–317.
  • Davey RJ. 1982. Solvent effects in crystallization processes. In: Kaldis E, editor. Current topics in materials science. Amsterdam: North-Holland; p. 429–479.
  • Di Martino P, Di Cristofaro R, Barthélémy C, Joiris E, Palmieri FG, Sante M. 2000. Improved compression properties of propyphenazone spherical crystals. Int J Pharm. 197:95–106.
  • Fiese EF, Hagen TA. 1986. Preformulation. In: Lachman L, Lieberman HA, Kanig JL, editors. Theory and practice of industrial pharmacy. 3rd ed. Philadelphia: Lea and Febiger; p. 171–196.
  • Fouad EA, El-Badry M, Mahrous GM, Alanazi FK, Neau SH, Alsarra IA. 2011. The use of spray-drying to enhance celecoxib solubility. Drug Dev Ind Pharm. 37:1463–1472.
  • George M, Ghosh I. 2013. Identifying the correlation between drug/stabilizer properties and critical quality attributes (CQAs) of nanosuspension formulation prepared by wet media milling technology. Euro J Pharm Sci. 48:142–152.
  • Gohle MC, Parikh RK, Shen H, Rubey RR. 2003. Improvement in flowability and compressibility of AmpicillineTrihydrate by spherical crystallization. Ind J Pharm Sci. 65:634–637.
  • Gupta VR, Mutalik S, Patel MM, Jani GK. 2007. Spherical crystals of celecoxib to improve solubility, dissolution rate and micromeritic properties. Acta Pharm. 57:173–184.
  • Homayouni A, Sadeghi F, Varshosaz J, AfrasiabiGarekani H, Nokhodchi A. 2014. Comparing various techniques to produce micro/nanoparticles for enhancing the dissolution of celecoxib containing PVP. Eur J Pharm Biopharm. 88:261–274.
  • Horn D, Rieger J. 2001. Organic nanoparticles in the aqueous phase-theory, experiment, and use. Angew Chem Int Ed Engl. 40:4330–4361.
  • Horter D, Dressman JB. 2001. Influence of physicochemical properties on dissolution of drugs in the gastrointestinal trac. Adv Drug Deliv Rev. 46:75–87.
  • Jbilou M, Ettabia A, Guyot-Hermann AM, Guyot JC. 1999. Ibuprofen agglomerates preparation by phase separation. Drug Dev Ind Pharm. 25:297–305.
  • Kachrimanis K, Ktistis G, Malamataris S. 1998. Crystallization conditions and physicochemical properties of ibuprofen-Eudragit S100 spherical crystal agglomerates prepared by the solvent-change technique. Int J Pharm. 173:61–74.
  • Kawashima Y. 1994. New process-application of spherical crystallization to particulate design of pharmaceuticals for direct tabletting and coating.and new drug delivery systems. In: Chulia D, Deleuil M, Pourcelot Y, editors. Powder technology and pharmaceutical processes. New York: Elsevier; p. 493–512.
  • Kawashima Y, Cui F, Takeuchi H, Niwa T, Hino T, Kiuchi K. 1994. Improvement in flowability and compressibility of pharmaceutical crystals for direct tableting by spherical crystallization with a two solvent system. Powder Technol. 78:151–157.
  • Kawashima Y, Imai M, Takeuchi H, Yamamoto H, Kamiya K, Hino T. 2003. Improved flowability and compactibility of spherically agglomerated crystals of ascorbic acid for direct tableting designed by spherical crystallization process. Powder Technol. 130:283–289.
  • Kawashima Y, Okumura M, Takenaka H. 1982. Spherical crystallization: direct spherical agglomeration of salicylic acid crystals during crystallization. Science. 216:1127–1128.
  • Kawashima Y, Okumura M, Takenaka H. 1984. The effects of temperature on the spherical crystallization of salicylic acid. Powder Technol. 39:41–47.
  • Labouret A, Thioune O, Fessi H, Devissaguet JP. 1995. PuisieuxF. Application of an original process for obtaining colloidal dispersions of some coating polymers. Preparation, characterization, industrial scaling up. Drug Dev Ind Pharm. 21:229–241.
  • Maghsoodi M, Barghi L. 2011. Design of agglomerated crystals of ibuprofen during crystallization: influence of surfactant. IJBMS. 14:161–169.
  • Maghsoodi M, Hassan-Zadeh D, Barzegar-Jalali M, Nokhodchi A, Martin G. 2007. Improved compaction and packing properties of naproxen agglomerated crystals obtained by spherical crystallization technique. Drug Dev Ind Pharm. 33:1216–1224.
  • Maghsoodi M, TajalliBakhsh A. 2011. Evaluation of physicomechanical properties of drug-excipients agglomerates obtained by crystallization. Pharm DevTechnol. 16:243–249.
  • Merck & Co., Inc. 2000. The Merck Index. Rahway, NJ: Merck & Co., Inc.
  • Mersmann A. 1999. Crystallization and precipitation. 1. ChemEng Process. 38:345–353.
  • Paradkar AR, Pawar AP, Chordiya JK. 2002. Spherical crystallization of celecoxib. Drug Dev Ind Pharm. 28:1213–1220.
  • Puechagut HG, Bianchotti J, Chaile CA. 1998. Preparation of norfloxacin spherical agglomerates using the ammonia diffusion system. J Pharm Sci. 87:519–523.
  • Quintanar-Guerrero D, Tamayo-Esquivel D, Ganem-Quintanar A, Allémann E, Doelker E. 2005. Adaptation and optimization of the emulsification-diffusion technique to prepare lipidicnanospheres. Euro J Pharm Sci. 26:211–218.
  • Shekunov BY, York P. 2000. Crystallization processes in pharmaceutical technology and drug delivery design. J Crystal Growth. 211:122–136.
  • Shen SC, Ng WK, Chia L, Hu J, Tan RB. 2011. Physical state and dissolution of ibuprofen formulated by co-spray drying with mesoporous silica: effect of pore and particle size. Int J Pharm. 410:188–195.
  • Slavtchev S, Kalitzova-Kurteva P, Mendes MA. 2006. Marangoni instability of liquid–liquid systems with a surface-active solute. Colloid Surf. 282:37–49.
  • Staniforth J. 2002. Powder flow. In: Aulton ME, editor. Pharmaceutics. 2nd ed. London: Churchill Livingstone; p. 207–428.
  • Subero-Couroyer C, Mangin D, Rivoire A, Blandin AF, Kelin JP. 2005. Agglomeration in suspension of salicylic acid fine particles: analysis of the wetting period and effect of the binder injection mode on the final agglomerate size. Powder Technol. 161:98–109.
  • Teychené S, Sicre N, Biscans B. 2010. Is spherical crystallization without additive possible. Chem Eng Res Des. 88:1631–1638.
  • USP/NF. 2007. Powder flow <1174>, United State Pharmacopeial Convention. Rockville (MD): The United State Pharmacopeia30/National Formulary25.
  • Wehrle P, Magenheim B, Benita S. 1995. The influence of processparameters on PLA nanoparticles size distribution, evaluated by factorial design. Eur J Pharm Biopharm. 41:19–26.

Reprints and Corporate Permissions

Please note: Selecting permissions does not provide access to the full text of the article, please see our help page How do I view content?

To request a reprint or corporate permissions for this article, please click on the relevant link below:

Academic Permissions

Please note: Selecting permissions does not provide access to the full text of the article, please see our help page How do I view content?

Obtain permissions instantly via Rightslink by clicking on the button below:

If you are unable to obtain permissions via Rightslink, please complete and submit this Permissions form. For more information, please visit our Permissions help page.