65
Views
1
CrossRef citations to date
0
Altmetric
Research Article

Mechanical activation of Efavirenz: the effects on the dissolution and inhibitory behavior

ORCID Icon, , , &
Pages 1128-1135 | Received 01 Aug 2017, Accepted 22 Mar 2018, Published online: 08 May 2018

References

  • Bitterlich A, Laabs C, Krautstrunk I, Dengler M, Juhnke M, Grandeury A, Bunjes H, Kwade A. 2015. Process parameter dependent growth phenomena of naproxen nanosuspension manufactured by wet media milling. Eur J Pharm Biopharm. 92:171–179.
  • Broseghini M, D’Incau M, Gelisio L, Pugno NM, Scardi P. 2017. Homogeneity of ball milled ceramic powders: effect of jar shape and milling conditions. Data in Brief. 10:186–191.
  • Broseghini M, Gelisio L, D’Incau M, Azanza Ricardo CL, Pugno NM, Scardi P. 2016. Modeling of the planetary ball-milling process: the case study of ceramic powders. J Eur Ceram Soc. 36: 2205–2212.
  • Cappelletto E, Rebuffi L, Flor A, Scardi P. 2017. Microstructural effects of high-energy grinding on poorly soluble drugs: the case study of Efavirenz. Powder Diffr. 32(S1):S135–S140.
  • Chadha R, Arora P, Saini A, Jain DS. 2012. An insight into thermodynamic relationship between polymorphic forms of Efavirenz. J Pharm Pharm Sci. 15:234–251.
  • Chiappetta DA, Alvarez-Lorenzo C, Rey-Rico A, Taboada P, Concheiro A, Sosnik A. 2010. N-alkylation of poloxamines modulates micellar assembly and encapsulation and release of the antiretroviral efavirenz. Eur J Pharm Biopharm. 76:24–37.
  • Costa Pinto E, Cabral L, Pereira de Sousa V. 2014. Development of a discriminative intrinsic dissolution method for Efavirenz. Dissolution Technol. 21:31–40.
  • Fandaruff C, Segatto Silva MA, Galindo Bedor DC, Pereira de Santana D, Vinícius Antunes Rocha H, Rebuffi L, Azanza Ricardo CL, Scardi P, Cuffini SL. 2015. Correlation between microstructure and bioequivalence in anti-HIV drug Efavirenz. Eur J Pharm Biopharm. 91:52–58.
  • Fitriani L, Haqi A, Zaini E. 2016. Preparation and characterization of solid dispersion freeze-dried efavirenz - polyvinylpyrrolidone K-30. J Adv Pharm Technol Res. 7:105–109.
  • Kakran M, Li L, Muller RH. 2012. Overcoming the challenge of poor drug solubility. Pharma Eng. 32:1–7.
  • Kalepu S, Nekkanti V. 2015. Insoluble drug delivery strategies: review of recent advances and business prospects. Acta Pharm Sin B. 5:442–453.
  • Khadka P, Ro J, Kim H, Kim I, Tae Kim J, Kim H, Cho JM, Yun G, Lee J. 2014. Pharmaceutical particle technologies: an approach to improve drug solubility, dissolution and bioavailability. Asian J Pharm Sci. 9:304–316.
  • Klug HP, Alexander L. 1974. X-ray diffraction procedures: for polycrystalline and amorphous materials. 2nd ed. New York (NY): Wiley.
  • Koyanagi Y, Miles S, Mitsuyasu RT, Merrill JE, Vinters HV, Chen IS. 1987. Dual infection of the central nervous system by AIDS viruses with distinct cellular tropisms. Science. 236:819–822.
  • Leuner C, Dressman J. 2000. Improving drug solubility for oral delivery using solid dispersions. Eur J Pharm Biopharm. 50: 47–60.
  • Liversidge GG, Cundy KC. 1995. Particle size reduction for improvement of oral bioavailability of hydrophobic drugs: I. Absolute oral bioavailability of nanocrystalline danazol in beagle dogs. Int J Pharm. 125:91–97.
  • Mosharraf M, Nystrom C. 1995. The effect of particle size and shape on the surface specific dissolution rate of microsized practically insoluble drugs. Int J Pharm. 122:35–47.
  • Muller RH, Keck CM. 2004. Challenges and solutions for the delivery of biotech drugs – a review of drug nanocrystal technology and lipid nanoparticles. J Biotechnol. 113:151–170.
  • Patel DJ, Patel JK, Pandya VM. 2010. Improvement in the dissolution of poorly water soluble drug using media milling technique. Thai J Pharm Sci. 34:155–164.
  • Patel GV, Patel VB, Pathak A, Rajput SJ. 2013. Nanosuspension of efavirenz for improved oral bioavailability: formulation optimization, in vitro, in situ and in vivo evaluation. Drug Dev Ind Pharm. 40(1):80–91.
  • Rabinow BE. 2004. Nanosuspensions in drug delivery. Nat Rev Drug Discov. 3:785–796.
  • Raza K, Kumar P, Ratan S, Malik R, Arora S. 2014. Polymorphism: the phenomenon affecting the performance of drugs. SOJPPS. 1:1–10.
  • Rebuffi L, Plaisier JR, Abdellatief M, Lausi A, Scardi P. 2014. MCX: a synchrotron radiation beamline form X-ray diffraction line profile analysis. Z Anorg Allg Chem. 640:3100–3106.
  • Reddy NP, Padmavathi Y, Mounika P, Anjali A. 2015. FTIR spectroscopy for estimation of efavirenz in raw material and tablet dosage form. Int Curr Pharm J. 4:390–395.
  • Rosa A, Chande A, Ziglio S, De Sanctis V, Bertorelli R, Goh SL, McCauley SM, Nowosielska A, Antonarakis SE, Luban J, et al. 2015. HIV-1 Nef promotes infection by excluding SERINC5 from virion incorporation. Nature. 526:121–127.
  • Saleem IY, Smyth HDC. 2010. Micronization of a Soft Material: Air-Jet and Micro-Ball Milling. AAPS PharmSciTech. 11:1642–1649.
  • Santos Alves LD, Felts de La Roca Soares M, Tavares de Albuquerque C, Rodrigues da Silva E, Couto Carneiro Vieira A, Ferreira Fontes DA, Bezerra Melo Figueirêdo C, Soares Sobrinho JL, Rolim Neto PJ. 2014. Solid dispersion of efavirenz in PVP K-30 by conventional solvent and kneading methods. Carbohyd Polym. 104:166–174.
  • Sun J, Wang F, Sui Y, She Z, Zhai W, Wang C, Deng Y. 2012. Effect of particle size on solubility, dissolution rate, and oral bioavailability: evaluation using coenzyme Q10 as naked nanocrystals. Int J Nanomedicine. 7:5733–5744.

Reprints and Corporate Permissions

Please note: Selecting permissions does not provide access to the full text of the article, please see our help page How do I view content?

To request a reprint or corporate permissions for this article, please click on the relevant link below:

Academic Permissions

Please note: Selecting permissions does not provide access to the full text of the article, please see our help page How do I view content?

Obtain permissions instantly via Rightslink by clicking on the button below:

If you are unable to obtain permissions via Rightslink, please complete and submit this Permissions form. For more information, please visit our Permissions help page.