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Research Articles

The use of design of experiments to develop hot melt extrudates for extended release of diclofenac sodium

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Pages 187-196 | Received 31 May 2019, Accepted 21 Oct 2019, Published online: 08 Nov 2019

References

  • Aljaberi A, Chatterji A, Dong Z, Shah NH, Malick W, Singhal D, Sandhu HK. 2013. Understanding and optimizing the dual excipient functionality of sodium lauryl sulfate in tablet formulation of poorly water soluble drug: wetting and lubrication. Pharm Dev Technol. 18(2):490–503.
  • Alshafiee M, Aljammal MK, Markl D, Ward A, Walton K, Blunt L, Korde S, Pagire SK, Kelly AL, Paradkar A, et al. 2019. Hot-melt extrusion process impact on polymer choice of glyburide solid dispersions: the effect of wettability and dissolution. Int J Pharm. 559:245–254.
  • Brabander C, van den Mooter G, Vervaet C, Remon JP. 2002. Characterization of ibuprofen as a nontraditional plasticizer of ethyl cellulose. J Pharm Sci. 91(7):1678–1685.
  • Bruce LD, Shah NH, Malick AW, Infeld MH, McGinity JW. 2005. Properties of hot-melt extruded tablet formulations for the colonic delivery of 5-aminosalicylic acid. Eur J Pharm Sci. 59(1):85–97.
  • Censi R, Gigliobianco MR, Casadidio C, Di Martino P. 2018. Hot melt extrusion: highlighting physicochemical factors to be investigated while designing and optimizing a hot melt extrusion process. Pharmaceutics. 10(3):89–125.
  • Crowley MM, Schroeder B, Fredersdorf A, Obara S, Talarico M, Kucera S, McGinity JW. 2004. Physicochemical properties and mechanism of drug release from ethyl cellulose matrix tablets prepared by direct compression and hot-melt extrusion. Int J Pharm. 269(2):509–522.
  • Desai D, Sandhu H, Shah N, Malick W, Zia H, Phuapradit W, Vaka SRK. 2018. Selection of solid-state plasticizers as processing aids for hot-melt extrusion. J Pharm Sci. 107(1):372–379.
  • Follonier N, Doelker E, Cole ET. 1995. Various ways of modulating the release of diltiazem hydrochloride from hot-melt extruded sustained release pellets prepared using polymeric materials. J Control Release. 36(3):243–250.
  • Frohoff-Hulsmann MA, Schmitz A, Lippold BC. 1999. Aqueous ethyl cellulose dispersions containing plasticizers of different water solubility and hydroxypropyl methylcellulose as coating material for diffusion pellets I. Drug release rates from coated pellets. Int J Pharm. 177(1):69–82.
  • Gutierrez-Rocca JC, Mcginity JW. 1993. Influence of aging on the physical-mechanical properties of acrylic resin films cast from aqueous dispersions and organic solutions. Drug Dev Ind Pharm. 19(3):315–332.
  • Hengsawas Surasarang S, Keen JM, Huang S, Zhang F, McGinity JW, Williams RO. 3rd. 2017. Hot melt extrusion versus spray drying: hot melt extrusion degrades albendazole. Drug Dev Ind Pharm. 3(5):797–811.
  • Islam MT, Maniruzzaman M, Halsey SA, Chowdhry BZ, Douroumis D. 2014. Development of sustained-release formulations processed by hot-melt extrusion by using a quality-by-design approach. Drug Deliv and Transl Res. 4(4):377.
  • Kate L, Gokarna V, Borhade V, Prabhu P, Deshpande V, Pathak S, Sharma S, Patravale V. 2016. Bioavailability enhancement of atovaquone using hot melt extrusion technology. Eur J Pharm Sci. 86:103–114.
  • Liechty WB, Kryscio DR, Slaughter BV, Peppas NA. 2010. Polymers for drug delivery systems. Annu Rev Chem Biomol Eng. 1(1):149–173.
  • Mansour HM, Sohn M, Al-Ghananeem A, Deluca PP. 2010. Materials for pharmaceutical dosage forms: molecular pharmaceutics and controlled release drug delivery aspects. IJMS. 11(9):3298–3322.
  • Maru SM, de Matas M, Kelly A, Paradkar A. 2011. Characterization of thermal and rheological properties of zidovudine, lamivudine and plasticizer blends with ethyl cellulose to assess their suitability for hot melt extrusion. Eur J Pharm Sci. 44(4):471–478.
  • Moradiya HG, Nokhodchi A, Bradley MS, Farnish R, Douroumis D. 2016. Increased dissolution rates of carbamazepine-gluconolactone binary blends processed by hot melt extrusion. Pharm Dev Technol. 21(4):445–452.
  • Nokhodchi A, Raja S, Patel P, Asare-Addo K. 2012. The role of oral controlled release matrix tablets in drug delivery systems. Bioimpacts. 2(4):175–187.
  • Patil H, Tiwari RV, Repka MA. 2016. Hot-melt extrusion: from theory to application in pharmaceutical formulation. AAPS PharmSciTech. 17(1):20–42.
  • Rekhi GS, Jambhekar SS. 1995. Ethylcellulose – a polymer review. Drug Dev Ind Pharm. 21(1):61–77.
  • Repka MA, Bandari S, Kallakunta VR, Vo AQ, McFall H, Pimparade MB, Bhagurkar AM. 2018. Melt extrusion with poorly soluble drugs – an integrated review. Int J Pharm. 535(1–2):68–85.
  • Sarode AL, Sandhu H, Shah N, Malick W, Zia H. 2013. Hot melt extrusion (HME) for amorphous solid dispersions: predictive tools for processing and impact of drug-polymer interactions on supersaturation. Eur J Pharm Sci. 48(3):371–384.
  • Skultety PF, Sims SM. 1987. Evaluation of the loss of propylene glycol during aqueous film coating. Drug Dev Ind Pharm. 13(12):2209–2219.
  • Tate S, Chiba S, Tani K. 1996. Melt viscosity reduction of poly(ethylene terephthalate) by solvent impregnation. Polymer. 37(19):4421–4424.
  • Tiwari RV, Patil H, Repka MA. 2016. Contribution of hot-melt extrusion technology to advance drug delivery in the 21st century. Expert Opin Drug Deliv. 13(3):451–464.
  • Tominaga K, Langevin B, Orton E. 2015. Recent innovations in pharmaceutical hot melt extrusion. Am Pharm Review. 18(6):1–4.
  • Vo AQ, Feng X, Morott JT, Pimparade MB, Tiwari RV, Zhang F, Repka MA. 2016. A novel floating controlled release drug delivery system prepared by hot-melt extrusion. Eur J Pharm Biopharm. 98:108–121.
  • Zhang D, Lee YC, Shabani Z, Frankenfeld Lamm C, Zhu W, Li Y, Templeton A. 2018. Processing impact on performance of solid dispersions. Pharmaceutics. 10(3):142–155.
  • Zhang F, McGinity JW. 1999. Properties of sustained-release tablets prepared by hot-melt extrusion. Pharm Dev Technol. 4(2):241–250.

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