547
Views
60
CrossRef citations to date
0
Altmetric
Research Article

A Critical Review of Gastric Retentive Controlled Drug Delivery

Pages 1-10 | Received 21 Apr 2006, Accepted 23 Jun 2006, Published online: 07 Oct 2008

REFERENCES

  • Moës A.J. Gastroretentive dosage forms. Crit. Rev. Ther. Drug Carrier Syst. 1993; 10: 143–195
  • Deshpande A.A., Rhodes C.T., Shah N.H., Malick A.W. Controlled-release drug delivery systems for prolonged gastric residence: an overview. Drug Dev. Ind. Pharm. 1996; 22(6)531–539
  • Hwang S.-J., Park H., Park K. Gastric retentive drug-delivery systems. Crit. Rev. Ther. Drug Carrier Syst. 1998; 15(3)243–284
  • Singh B.N., Kim K.H. Floating drug delivery systems: An approach to oral controlled drug delivery via gastric retention. J. Control. Release 2000; 63: 235–259
  • Fell J.T., Whitehead L., Collett J.H. Prolonged gastric retention using floating dosage forms. Pharm. Tech. March, 2000, 82, 84, 86, 88, 90
  • Soppimath K.S., Kulkarni A.R., Rudzinski W.E., Aminabhavi T.M. Microspheres as floating drug-delivery systems to increase gastric retention of drugs. Drug Met. Rev. 2001; 33: 149–160
  • Gutierrez-Rocca J., Omidian H., Shah K. Progress in gastroretentive drug delivery systems. Business Briefing: Pharmatech. 2003; 152–156
  • Hou S.Y.E., Cowles V.E., Berner B. Gastric retentive dosage forms: a review. Crit. Rev. Ther. Drug Carrier Syst. 2003; 20: 461–497
  • Klausner E.A., Lavy E., Friedman M., Hoffman A. Expandable gastroretentive dosage forms. J. Control. Release 2003; 90(2)143–162
  • Moës A.J. Gastric retention systems for oral drug delivery. Business Briefing: Pharmatech. 2003; 157–159
  • Talukder R., Fasshihi R. Gastroretentive delivery systems: A mini review. Drug Dev. Ind. Pharm. 2004; 30: 1019–1028
  • Hoffman A., Stepensky D., Lavy E., Eyal S., Klausner E., Friedman M. Pharmacokinetic and pharmacodynamic aspects of gastroretentive dosage forms. Int. J. Pharm. 2004; 277(1–2)141–153
  • Chowdary K.P.R., Rao Y.S. Mucoadhesive microspheres and microcapsules: Current status. Ind. J. Pharm. Sci. 2005; 67: 141–150
  • Rocca J.G., Omidian H., Shah K.U. Commercial status of gastric retention technologies. Drug Del. Tech. 2005; 50–58
  • Bardonnet P.L., Faivre V., Pugh W.J., Piffaretti J.C., Falson F. Gastroretentive dosage forms: Overview and special case of Helicobacter pylori. J. Control. Release 2006; 111(1–2)1–18
  • Streubel A., Siepmann J., Bodmeier R. Gastroretentive drug delivery systems. Expert Opin. Drug Deliv. 2006; 3(2)217–233
  • Fix J.A., Cargill R., Engle K. Controlled gastric emptying. III. Gastric residence time of a nondisintegrating geometric shape in human volunteers. Pharm. Res. 1993; 10: 1087–1089
  • Coupe A.J., Davis S.S., Evans D.F., Wilding I.R. Correlation of the gastric emptying of nondisintegrating tablets with gastrointestinal motility. Pharm. Res. 1991; 8(10)1281–1285
  • Itoh T., Higuchi T., Gardner C.R., Caldwell L. Effect of particle size and food on gastric residence time of non-disintegrating solids in beagle dogs. J. Pharm. Pharmacol. 1986; 38(11)801–806
  • Kaniwa N., Aoyagi N., Ogata H., Ejima A. Gastric emptying rates of drug preparations. I. Effects of size of dosage forms, food and species on gastric emptying rates. J. Pharm.-Dyn. 1988; 11(8)563–570
  • 21. Nause, R., Li, F., Sagawa, K. Modeling and prediction of upper GI transit times for non-disintegrating oral dosage forms, Manuscript in preparation.
  • Davis S.S., Hardy J.G., Fara J.W. Transit of pharmaceutical dosage forms through the small intestine. Gut 1986; 27(8)886–892
  • Ewe K., Press A.G., Bollen S., Schuhn I. Gastric emptying of indigestigle tablets in relation to composition and time of ingestion of meals studied by metal detector. Dig. Dis. Sci. 1991; 36(2)146–152
  • Steed K.P., Hooper G., Monti N., Strolin Benedetti M., Fornasini G., Wilding I.R. The use of pharmacoscintigraphy to focus the development strategy for a novel 5-ASA colon targeting system (“TIME CLOCK” system). J. Control. Release 1997; 49(2,3)115–122
  • Khosla R., Davis S.S. The effect of polycarbophil on the gastric emptying of pellets. J. Pharm. Pharmacol. 1987; 39: 47–49
  • Harris D., Fell J.T., Sharma H.L., Taylor D.C. Gastrointestinal transit of potential bioadhesive formulations in man: A scintigraphic study. J. Control. Release 1990; 12: 45–53
  • Jackson S.J., Bush D., Perkins A.C. Comparative scintigraphic assessment of the intragastric distribution and residence of cholestyramine, Carbopol 934P and sucralfate. Int. J. Pharm. 2001; 212: 55–62
  • Säkkinen M., Tuononen T., Jürjenson H., Veski P., Marvola M. Evaluation of microcrystalline chitosans for gastro-retentive drug delivery. Eur. J. Pharm. Sci. 2003; 19: 345–353
  • Säkkinen M., Marvola J., Kanerva H., Lindevall K., Lipponen M., Kekki T., Ahonen A., Marvola M. Gamma scintigraphic evaluation of the fate of microcrystalline chitosan granules in human stomach. Eur. J. Pharm. Biopharm. 2004; 57: 133–143
  • Ch'ng H. S., Park H., Kelly P., Robinson J.R. Bioadhesive polymers as platforms for oral controlled drug delivery. II. Synthesis and evaluation of some swelling, water-insoluble bioadhesive polymers. J. Pharm. Sci. 1985; 74(4)399–405
  • Lehr C.M., Bouwstra J.A., Schacht E.H., Junginger H.E. In vitro evaluation of mucoadhesive properties of chitosan and some other natural polymers. Int. J. Pharm. 1992; 78: 43–48
  • He P., Davis S.S., Illum L. In vitro evaluation of the mucoadhesive properties of chitosan microspheres. Int. J. Pharm. 1998; 166: 75–88
  • Gåserød O., Jolliffe A.G., Hampson F.C., Dettmar P.W., Skjåk-Braek G. The enhancement of the bioadhesive properties of calcium alginate gel beads by coating with chitosan. Int. J. Pharm. 1998; 175: 237–246
  • Slovin E.M., Robinson J.R. Bioadhesives in ocular drug delivery. Biopharm. Ocul. Drug Deliv. 1993; 145–157
  • Signorin J., Aguinaldo E.R., Reilly W.J. Nasal mucoadhesive characteristics of co-processed MCC CMC-Avicel RC-591. Proc. Intern. Symp. Control. Release Bioact. Mat. 1998; 25: 758–759
  • Ugwoke M.I., Exaud S., Van Den Mooter G., Verbeke N., Kinget R. Bioavailability of apomorphine following intranasal administration of mucoadhesive drug delivery systems in rabbits. Eur. J. Pharm. Sci. 1999; 9: 213–219
  • Ugwoke M.I., Verbeke N., Kinget R. The biopharmaceutical aspects of nasal mucoadhesive drug delivery. J. Pharm. Pharmacol. 2001; 53: 3–22
  • Jain S.K., Chourasia M.K., Jain A.K., Jain R.K., Shrivastava A.K. Development and characterization of mucoadhesive microspheres bearing salbutamol for nasal delivery. Drug Deliv. 2004; 11(2)113–122
  • Edsman K., Haegerstroem H. Pharmaceutical applications of mucoadhesion for the non-oral routes. J. Pharm. Pharmacol. 2005; 57: 3–22
  • Ingani H.M., Timmermans J., Moës A. Conception and in vivo investigation of peroral sustained release floating dosage forms with enhanced gastrointestinal transit. J. Int. Pharm. 1987; 35: 157–164
  • Mazer N., Abisch E., Gfeller J.-C., Laplanche R., Bauerfeind P., Cucala M., Lukachich M., Blum A. Intragastric behavior and absorption kinetics of a normal and “floating” modified-release capsule of isradipine under fasted and fed conditions. J. Pharm. Sci. 1988; 77: 647–657
  • Washington N., Wilson C.G., Greaves J.L., Danneskiold-Samsøe P. An investigation into the floating behaviour of a pectin-containing anti-reflux formulation (FF5005) by means of gamma scintigraphy, Scand. J. Gastroenterol. 1988; 23: 920–924
  • Timmermans J., Van Gansbeke B., Moës A.J. Assessing by gamma scintigraphy the in vivo buoyancy of dosage forms having known size and floating force profiles as a function of time. Congr. Int. Technol. Pharm. 5th. 1989; 1: 42–51
  • Timmermans J., Moës A.J. Factors controlling the buoyancy and gastric retention capabilities of floating matrix capsules: New data for reconsidering the controversy. J. Pharm. Sci. 1994; 83(1)18–24
  • Babu V.B.M., Khar R.K. In vitro and in vivo studies of sustained-release floating dosage forms containing salbutamol sulfate. Pharmazie 1990; 45: 268–270
  • Phuapradit W., Bolton S. The influence of tablet density on the human oral absorption of sustained release acetaminophen tablets. Drug Dev. Ind. Pharm. 1991; 17: 1097–1107
  • Xu W.L., Tu X.D., Lu Z.D. Development of gentamicin sulfate sustained-release tablet floating in stomach. Yaoxue Xuebao 1991; 26(7)541–545
  • Agyilirah G.A., Green M., DuCret R., Banker G.S. Evaluation of the gastric retention properties of a crosslinked polymer coated tablet versus those of a nondisintegrating tablet. Int. J. Pharm. 1991; 75(2–3)241–247
  • Hilton A.K., Deasy P.B. In vitro and in vivo evaluation of an oral sustained-release floating dosage form of amoxicillin trihydrate. Int. J. Pharm. 1992; 86: 79–88
  • Oth M., Franz M., Timmermans J., Möes A. The bilayer floating capsule: A stomach-directed drug delivery system for misoprostol. Pharm. Res. 1992; 9: 298–302
  • Desai S., Bolton S. A floating controlled-release drug delivery system: In vitro-in vivo evaluation. Pharm. Res. 1993; 10: 1321
  • Özdemir N., Ordu S., Özkan Y. Studies of floating dosage forms of furosemide: in vitro and in vivo evaluations of bilayer tablet formulations. Drug Dev. Ind. Pharm. 2000; 26: 857–866
  • Gabr K.E., Borg T.M. Formulation and evaluation of buffered floating furosemide delivery systems. S.T.P. Pharm. Sci. 2000; 10: 181–186
  • Chavanpatil M., Jain P., Chaudhari S., Shear R., Vavia P. Development of sustained release gastroretentive drug delivery system for ofloxain: in vitro and in vivo evaluation. Int. J. Pharm. 2005; 304: 178–184
  • Bechgaard H. Distribution of different types of dosage forms in the gastrointestinal tract. Top. Pharm. Sci. 1983; 217–228
  • Bechgaard H., Christensen F.N., Davis S.S., Hardy J.G., Taylor M.J., Whalley D.R., Wilson C.G. Gastrointestinal transit of pellet systems in ileostomy subjects and the effect of density. J. Pharm. Pharmacol. 1985; 37: 718–721
  • Lippold B.C., Günther J. In-vivo Prüfung einer multipartikulären Retard-Schwimmarzneiform. Eur. J. Pharm. Biopharm. 1991; 37: 254–261
  • Kawashima Y., Niwa T., Takeuchi H., Hino T., Ito Y. Preparation of multiple unit hollow microspheres (microballoons) with acrylic resin containing tranilast and their drug release characteristics (in vitro) and floating behavior (in vivo). J. Control. Release 1991; 16: 279–190
  • Atyabi F., Sharma H.L., Mohammad H.A.H., Fell J.T. In vivo evaluation of a novel gastric retentive formulation based on ion exchange resins. J. Control. Release 1996; 42: 105–113
  • Iannuccelli V., Coppi G., Cameroni R. Intragastric behaviour of a multiple-unit dosage form. Proc. Intl. Symp. Control. Release Bioact. Mater. 1997; 24: 403–404
  • Iannuccelli V., Coppi G., Sansone R., Ferolla G. Air compartment multiple-unit system for prolonged gastric residence. II. In vivo evaluation. Int. J. Pharm. 1998; 174: 55–62
  • Whitehead L., Fell J.T., Collett J.H., Sharma H.L., Smith A.-M. Floating dosage forms: an in vivo study demonstrating prolonged gastric retention. J. Control. Release 1998; 55: 3–12
  • Sawicki W. Pharmacokinetics of verapamil and norverapamil from controlled release floating pellets in humans. Eur. J. Pharm. Biopharm. 2002; 53: 29–35
  • hrrp://www.aapspharmscitech.org, Shimpi, S., Chauhan, B., Mahadik, K.R., Paradkar, A. Preparation and evaluation of diltiazem hydrochloride-gelucire 43/01 floating granules prepared by melt granulation. AAPS PharmSciTech 2004, 5, article 43
  • Munk J., Gannaway R., Hoare M., Johnson A. H.L. DuthieGastroinestinal Motility in Health and Disease, . MTP, Lancaster 1978; 349–359
  • Channer K.S., Virjee J.P. The effect of size and shape of tablets on the esophageal transit. J. Clin. Pharmacol. 1986; 26: 141–146
  • Gusler G., Gorsline J., Levy G., Zhang S.Z., Weston I.E., Naret D., Berner B. Pharmacokinetics of metformin gastric-retentive tablets in healthy volunteers. J. Clin. Pharmacol. 2001; 41: 655–661
  • Gusler G., Berner B. Metformin (GRTM) gastric retentive tablets: GI transit and pharmacokinetics in healthy volunteers. Millenial World Congress of Pharm. Sci, San Francisco 2000; 2–5019
  • Klausner E.A., Lavy E., Barta M., Cserepes E., Friedman M., Hoffman A. Novel gastroretentive dosage forms: Evaluation of gastroretentivity and its effect on levodopa absorption in humans. Pharm. Res. 2003; 20: 1466–1473
  • Cargill R., Caldwell L.J., Engle K., Fix J.A., Porter P.A., Gardner C.R. Controlled gastric emptying. I. Effects of physical properties on gastric residence times of nondisintegrating geometric shapes in beagle dogs. Pharm. Res. 1988; 5: 533–536

Reprints and Corporate Permissions

Please note: Selecting permissions does not provide access to the full text of the article, please see our help page How do I view content?

To request a reprint or corporate permissions for this article, please click on the relevant link below:

Academic Permissions

Please note: Selecting permissions does not provide access to the full text of the article, please see our help page How do I view content?

Obtain permissions instantly via Rightslink by clicking on the button below:

If you are unable to obtain permissions via Rightslink, please complete and submit this Permissions form. For more information, please visit our Permissions help page.