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Journal of Enzyme Inhibition and Medicinal Chemistry Volume 17, 2002 - Issue 3
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Research Article

N -substituted 4-(4-carboxyphenoxy)benzamides. Synthesis and Evaluation as Inhibitors of Steroid-5α-reductase Type 1 and 2

Franck Picard 8.5 Pharmaceutical and Medicinal Chemistry, Saarland University, P.O. Box 15 11 50, D-66041 Saarbrücken, Germany
&
Rolf W. Hartmann 8.5 Pharmaceutical and Medicinal Chemistry, Saarland University, P.O. Box 15 11 50, D-66041 Saarbrücken, Germany
Pages 187-196 | Published online: 30 Sep 2008

  • Picard, F., Schulz, T. and Hartmann, R.W. (2002) Bioorg. Med. Chem. 10, 437-448.
  • Keetch, D.W. and Andriole, G.L. (1995) Am. J. Roentgenology 164, 11-15.
  • Kenny, B., Ballard, S., Blagg, J. and Fox, D. (1997) J. Med. Chem. 40, 1293-1315.
  • Ziada, A., Rosenblum, M. and Crawford, E.D. (1999) Urology 53, 1-6.
  • Lepor, H., Williford, W.O., Barry, M.J., Brawer, M.K., Dixon, C.M., Gormley, G., Haakenson, C, Machi, M., Narayan, P. and Padley, R.J. (1996) N. Engl. J. Med. 335, 533-539.
  • Baston, E., Palusczak, A. and Hartmann, R.W. (2000) Eur. J. Med. Chem. 35, 931-940.
  • Hartmann, R.W. and Reichert, M. (2000) Arch. Pharm. Pharm. Med. Chem. 333, 145-153.
  • Picard, F., Baston, E., Reichert, W. and Hartmann, R.W. (2000) Bioorg. Med. Chem. 8, 1479-1487.
  • Baston, E. and Hartmann, R.W. (1999) Bioorg. Med. Chem. Lett. 9, 1601-1606.
  • Hartmann, R.W., Reichert, M. and Göhring, S. (1994) Eur. J. Med. Chem. 29, 807-817.
  • Lesuisse, D., Gourvest, J.F., Albert, E., Doucet, B., Hartmann, C., Lefrançois, J.M., Tessier, S., Trie, B. and Teutsch, G. (2001) Bioorg. Med. Chem. Lett. 11, 1713-1716.
  • Igarashi, S., Inami, H., Hara, H., Fujii, M., Koutoku, H., Oritani, H. and Mase, T. (2000) Chem. Pharm. Bull. 48, 382-388.
  • McNulty, A.M., Audia, J.E., Bemis, K.G., Goode, R.L., Rocco, V.P and Neubauer, B.L. (2000) J. Steroid Biochem. Mol. Biol. 72, 13-21.
  • Holt, D.A., Yamashita, D.S., Konialian-Beck, A.L., Luengo, J.I., Abell, A.D., Bergsam, D.J., Brandt, M. and Levy, M.A. (1995) J. Med. Chem. 38, 13-15.
  • Igarashi, S., Kimura, T., Naito, R., Hara, H., Fujii, M., Koutoku, H., Oritani, H. and Mase, T. (1999) Chem. Pharm. Bull. 47, 1073-1080.
  • Picard, F., Barassin, S., Mokhtarian, A. and Hartmann, R.W. (2002) J. Med. Chem., in press.
  • Dann, O., Ruff, J., Wolf, H.P. and Grießmeier, H. (1984) Liebigs Ann. Chem., 409-425.
  • Liang, T., Cascieri, M.A., Cheung, A.H., Reynolds, G.F. and Rasmusson, G.H. (1985) Endocrinology 117, 571-579.
  • Delos, S., Iehle, C., Martin, P.M. and Raynaud, J.P (1994) J. Steroid Biochem. Mol. Biol. 48, 347-352.
  • Kaefer, M., Audia, J.E., Bruchovsky, N., Goode, R.L., Hsiao, K.C., Leibovitch, I.Y., Krushinski, J.H., Lee, C., Steidle, C.P, Sutkowski, D.M. and Neubauer, B.L. (1996) J. Steroid Biochem. Mol. Biol. 58, 195-205.
  • Reichert, W., Jose, J. and Hartmann, R.W. (2000) Arch. Pharm. Pharm. Med. Chem. 333, 201-204.
  • Cook, S.J., Rawlings, N.C. and Kennedy, R.l. (1982) Steroids 40, 369-380.
  • Mukaiyama, T. (1979) Angew: Chem. 91, 798-812.
  • Dalcanale, E. and Montanari, F. (1986) J. Org. Chem. 51, 567-569.
  • Bartsch, G., Rittmaster, R.S. and Klocker, H. (2000) Eur. Urol. 37, 367-380.
  • Graul, A., Silvestre, J. and Castaner, J. (1999) Drugs Fut. 24, 246-253.
  • Frye, S.V., Haffner, C.D., Maloney, R.J., Dorsey, G.F., Noe, R.A., Hiner, R.N., Cribbs, C.M., Batchelor, K.W., Bramson, H.N., Stuart, J.D., Schweiker, S.L., Van Arnold, J., Croom, D.K., Bickett, M., Moss, M.L., Tian, G., Unwalla, R.J., Lee, F.W., Tippin, T.K., James, M.K., Grizzle, M.K. and Long, J.E. (1995) J. Med. Chem. 38, 2621-2627.
  • Frye, S.V., Haffner, C.D., Maloney, PR., Mook, Jr, R.A., Dorsey, Jr, G.F., Hiner, R.N., Batchelor, K.W., Bramson, H.N., Stuart, J.D., Schweiker, S.L., Van Arnold, J., Bickett, D.M., Moss, M.L., Tian, G., Unwalla, R.J., Lee, F.W., Tippin, T.K., James, M.K., Grizzle, M.K., Long, J.E. and Schuster, S.V. (1993) J. Med. Chem. 36, 4313-4315.
  • Igarashi, S., Inami, H., Hara, H., Fujii, M., Koutoku, H., Oritani, H. and Mase, T. (2000) Chem. Pharm. Bull. 48, 382-388.
  • McNulty, A.M., Audia, J.E., Bemis, K.G., Goode, R.L., Rocco, V.P. and Neubauer, B.L. (2000) J. Steroid Biochem. Mol. Biol. 72, 13-21.
  • Hirosumi, J., Nakayama, O., Chida, N., Inami, M., Fagan, T., Sawada, K., Shigematsu, S., Kojo, H., Notsu, Y. and Okuhara, M. (1995) J. Steroid Biochem. Mol. Biol. 52, 365-373.
  • Hirosumi, J., Nakayama, O., Fagan, T., Sawada, K., Chida, N., Inami, M., Takahashi, S., Shigematsu, S., Kojo, H., Notsu, Y. and Okuhara, M. (1995) J. Steroid Biochem. Mol. Biol. 52, 357-363.

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