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Journal of Enzyme Inhibition and Medicinal Chemistry Volume 35, 2020 - Issue 1
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Research Paper

Further validation of strecker-type α-aminonitriles as a new class of potent human carbonic anhydrase II inhibitors: hit expansion within the public domain using differential scanning fluorimetry leads to chemotype refinement

Mikhail Krasavina Saint Petersburg State University, Saint Petersburg, Russian FederationCorrespondence[email protected]
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,
Stanislav Kalinina Saint Petersburg State University, Saint Petersburg, Russian FederationView further author information
,
Sergey Zozulyab Enamine Ltd, Kyiv, Ukraine;c Taras Shevchenko National University, Kyiv, UkraineView further author information
,
Anastasia Griniukovab Enamine Ltd, Kyiv, UkraineView further author information
,
Petro Boryskob Enamine Ltd, Kyiv, UkraineView further author information
,
Andrea Angelid Neurofarba Department, Universita degli Studi di Firenze, Florence, ItalyORCID Iconhttps://orcid.org/0000-0002-1470-7192View further author information
ORCID Icon &
Claudiu T. Supurand Neurofarba Department, Universita degli Studi di Firenze, Florence, ItalyCorrespondence[email protected]
ORCID Iconhttps://orcid.org/0000-0003-4262-0323View further author information
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Pages 165-171 | Received 16 Oct 2019, Accepted 11 Nov 2019, Published online: 22 Nov 2019

References

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