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Original Articles

Synthesis and in Vitro Anti-Tumor Activity of A New Class of Acyclic Thioglycosides

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Pages 463-474 | Received 01 Jul 2014, Accepted 31 Jan 2015, Published online: 09 Jul 2015

REFERENCES

  • Elgemeie, G.H.; Elghandour, A.H.; Elzanate, A.M.; Ahmed, S.A. Synthesis of some novel α-cyanoketene S,S-acetals and their use in Heterocyclic synthesis. J. Chem. Soc. Perkin Trans. I. 1997, 3285.
  • Elgemeie, G.H.; Hussein, M.M.; Al-Khursani, S.A. A total synthesis of a new class of biazine thioglycosides. J. Carbohydr. Chem. 2004, 23, 465.
  • Elgemeie, G.H. Thioguanine, mercaptopurine, their analogs, and nucleosides as antimetabolites. Current Pharmaceutical Design. 2003, 9, 2627.
  • Elgemeie, G.H.; Hussain, B.A. A convenient synthesis of 5-deaza nonclassical antifolates: reaction of cyanothioacetamide with sodium salts of 2-(hydroxymethylene)-1-cycloalkanones. Tetrahedron 1994, 50, 199.
  • Elgemeie, G.H.; Zaghary, W.A.; Amin, K.M.; Nasr, T.M. First synthesis of thienopyrazole thioglycosides. J. Carbohydr. Chem. 2008, 27, 345.
  • Abu-Zaied, M.A.; El-Telbani, E.M.; Elgemeie, G.H.; Nawwar, G.A. Synthesis and in vitro anti-tumor activity of new oxadiazole thioglycosides. Eur. J. Med. Chem. 2011, 46, 229.
  • Elgemeie, G.H.; Mahdy, E.M.; Elgawish, M.A.; Ahmed, M.M.; Shousha, W.G.; Eldin, M.E. A new class of antimetabolites: pyridine thioglycosides as potential anticancer agents. Z. Naturforsch. 2010, 65c, 577.
  • Scala, S.; Akhmed, N.; Rao, U.S.; PaullLan, K.L.; Dickstein, B.; Lee, J.; Elgemeie, G.H.; Stein, W.D.; Bates, S.E. P-Glycoprotein substrates and antagonists cluster into two distinct groups. Mol. Pharmacol. 1997, 51, 1024.
  • Xia, Y.; Fan, C.D.; Zhao, B.X.; Zhao, J.; Shin, D.S.; Miao, J.Y. Synthesis and structure–activity relationships of novel 1-arylmethyl-3-aryl-1H-pyrazole-5-carbohydrazide hydrazone derivatives as potential agents against A549 lung cancer cells. Eur. J. Med. Chem. 2008, 43, 2347.
  • Zheng, C.; Xu, L.; Sun, L.; Miao, J.; Piao, H. Synthesis and antibacterial activity of novel 1,3-diphenyl-1H-pyrazoles functionalized with phenylalanine-derived rhodanines. Eur. J. Med. Chem. 2012, 58, 112.

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