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Original Articles

Synthesis of Some New 1,3/ or 1,4-Bis(Glucopyranosyl-1,2,4-Triazol-5-Ylthio)Propanes/ or Butanes as Potential Antimicrobial Agents

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Pages 1353-1372 | Accepted 11 May 2005, Published online: 31 Aug 2006

References

  • Jones , D . H .; Slack , R .; Squires , S .; Wooldridge , K . R.H . Antiviral chemotherapy. I. The activity of pyridine and quinoline derivatives against neurovaccina in mice . J. Med. Chem . 1965 , 8 , 676 – 680 . [CSA]
  • Goswami , B . N .; Kataky , J . C.S .; Baruah , J . N . Synthesis and antibacterial activity of 1-(2,4-dichlorobenzoyl)-4-substituted thiosemicarbazides, 1,2,4-triazoles and their methyl derivatives . J. Heterocycl. Chem . 1984 , 21 , 1225 – 1229 . [CSA]
  • Holla , B . S .; Kalluraya , B .; Sridhar , K . R . Synthesis of 4-(5-nitro-2-furfurylidene)amino-3-mercapto-5-(substituted)-1,2,4-triazoles as possible antibacterial agents . Curr. Sci . 1987 , 56 , 236 – 238 . [CSA]
  • Abdou , N . A .; Amin , F . M . Synthesis and biological activity of certain 5-mercapto-3-(3-pyridyl)-4H-1,2,4-triazole derivatives . Mansoura J. Pharm. Sci . 1990 , 6 , 25 – 29 . [CSA]
  • Mishra , R . K .; Tewari , R . K .; Srivastava , S . K .; Bahel , S . C . Synthesis and antifungal activity of some 1,4-disubstitued-thiosemicarbazides, 2,5-disubstituted-1,3,4-thiadiazoles and 3,4-disubstituted-5-mercapto-1,2,4-triazoles . J. Indian Chem. Soc . 1991 , 68 , 110 – 112 . [CSA]
  • Unangst , P . C .; Shurum , G . P .; Connor , D . T .; Dyer , R . D .; Schrier , D . J . Novel 1,2,4-oxadiazoles and 1,2,4-thiadiazoles as dual 5-lipoxygenase and cyclooxygenase inhibitors . J. Med. Chem . 1992 , 35 , 3691 – 3698 . [PUBMED] [INFOTRIEVE] [CSA] [CROSSREF]
  • Mullican , M . D .; Wilson , M . W .; Connor , D . T .; Kostlan , C . R .; Schrier , D . J .; Dyer , R . D . Design of 5-(3,5-di-tert-butyl-4-hydroxyphenyl)-1,3,4-thiadiazoles, -1,3,4-oxadiazoles, and -1,2,4-triazoles as orally active, nonulcerogenic antiinflammatory agents . J. Med. Chem . 1993 , 36 , 1090 – 1099 . [PUBMED] [INFOTRIEVE] [CSA] [CROSSREF]
  • Sugden , J . K .; Yoloye , T . O . Medicinal applications of indole derivatives . Pharm. Acta Helv . 1978 , 53 , 65 – 92 . [PUBMED] [INFOTRIEVE] [CSA]
  • Shams El-Dine , Sh . A .; Hazzaa , A . A.B . Synthesis of compounds with potential fungicidal activity . Pharmazie 1974 , 29 , 761 – 763 . [PUBMED] [INFOTRIEVE] [CSA]
  • Misato , T .; Ko , K .; Honma , Y .; Konno , K .; Taniyama , E . 1,3,4-Thiadiazole derivatives as fungicides . Chem. Abstr . 1977 , 87 , 147054a . [CSA]
  • Cansiz , A .; Servi , S .; Koparir , M .; Altintas , M .; Digrak , M . J. Chem. Soc. Pak . 2001 , 23 , 237 – 239 . [CSA]
  • Stillings , M . R .; Welbourn , A . P .; Walter , D . S . Substituted 1,3,4-thiadiazoles with anticonvulsant activity. 2. Aminoalkyl derivatives . J. Med. Chem . 1986 , 29 , 2280 – 2284 . [PUBMED] [INFOTRIEVE] [CSA] [CROSSREF]
  • Kane , J . M .; Dudley , M . W .; Sorensen , S . M .; Miller , F . P . 2,4-Dihydro-3H-1,2,4-triazole-3-thiones as potential antidepressant agents . J. Med. Chem . 1988 , 31 , 1253 – 1258 . [PUBMED] [INFOTRIEVE] [CSA] [CROSSREF]
  • Witkowski , J . T .; Robins , R . K .; Sidwell , R . W .; Simon , L . N . Design, synthesis, and broad spectrum antiviral activity of 1-β-d-ribofuranosyl-1,2,4-triazole-3-carboxamide and related nucleosides . J. Med. Chem . 1972 , 15 , 1150 – 1154 . [PUBMED] [INFOTRIEVE] [CSA] [CROSSREF]
  • The Pharmacology of Ribavirin ; Smith , R . A ., Kirkpatrick , W ., Eds.; Academic Press : London , 1980 ; 133 – 156 .
  • In Vitro and In Vivo Inhibition of DNA Viruses by Ribavirin ; Sidwell , R . W ., Eds.; Academic Press : Orlando, FL , 1984 ; 19 – 32 .
  • Clinical Applications of Ribavirin ; Smith , R . A ., Knight , V ., Smith , J . A.D ., Eds.; Academic Press : Orlando, FL , 1984 ; 222 .
  • Ibrahim , Y . A .; Behbeheni , H .; Khalil , N . S . Efficient route to 20–32 membered macrocyclic crown diamides via ring closing metathesis . Tetrahedron 2004 , 60 , 8429 – 8436 , and references cited therein. [CSA] [CROSSREF]
  • Drug Design ; Ariens , E . J ., Ed.; Academic Press : New York , 1971 ; 2 – 4 .
  • Khalil , N . S.A.M .; Mansour , A . K .; Eid , M . M . Synthesis of some novel 6-benzyl(or substituted benzyl)-2-β-d-glucopyranosyl-1,2,4-triazolo[4,3-b][1,2,4]triazines as potential antimicrobial chemotherapeutics . Nucleosides Nucleotides Nucleic Acids 2004 , 23 , 1889 – 1910 . [PUBMED] [INFOTRIEVE] [CSA] [CROSSREF]
  • Khalil , N . S.A.M . Synthesis of some novel N-ribosyl-1,2,4-triazin-6(1H)- ones or thiones as potential antibacterial and antifungal chemotherapeutics . Nucleosides Nucleotides Nucleic Acids 2005 , 24 , 111 – 120 . [PUBMED] [INFOTRIEVE] [CSA]
  • Khalil , N . S.A.M . Synthesis of novel α-l-arabinopyranosides of monocyclic β-lactams with potential antimicrobial activity . Nucleosides Nucleotides Nucleic Acids 2005 , in press . [CSA]
  • Mansour , A . K .; Eid , M . M .; Khalil , N . S.A.M . Selective synthesis and reactions of 6-substituted-2-β-galactosyl-1,2,4-triazines of potential anticancer activity . Nucleosides Nucleotides Nucleic Acids 2003 , 22 , 21 – 44 . [PUBMED] [INFOTRIEVE] [CSA] [CROSSREF]
  • Mansour , A . K .; Eid , M . M .; Khalil , N . S.A.M . Synthesis of some new 2-α-l-arabinopyranosyl-1,2,4-triazines as potential antitumor chemotherapeutics . Nucleosides Nucleotides Nucleic Acids 2003 , 22 , 1805 – 1823 . [PUBMED] [INFOTRIEVE] [CSA] [CROSSREF]
  • Mansour , A . K .; Eid , M . M .; Khalil , N . S.A.M . Synthesis of some N-galactosides of 3-aryl-5-benzyl(or substituted benzyl)-1,2,4-triazin-6(1H)- ones or thiones of expected biological activity . Nucleosides Nucleotides Nucleic Acids 2003 , 22 , 1825 – 1833 . [PUBMED] [INFOTRIEVE] [CSA] [CROSSREF]
  • Mansour , A . K .; Eid , M . M .; Khalil , N . S.A.M . Synthesis and reactions of some new heterocyclic carbohydrazides and related compounds as potential anticancer agents . Molecules 2003 , 8 , 744 – 755 . [CSA]
  • Mansour , A . K .; Ibrahim , Y . A .; Khalil , N . S.A.M . Selective synthesis and structure of 6-arylvinyl-2- and 4-glucosyl-1,2,4-triazines of expected interesting biological activity . Nucleosides Nucleotides 1999 , 18 , 2265 – 2283 . [CSA]
  • Ibrahim , Y . A .; Abbas , A . A .; Elwahy , A . H.M . Selective synthesis and structure of 2-N- and 3-S-glucosyl-1,2,4-triazoles of potential biological interest . Carbohydr. Lett . 1999 , 35 , 331 – 338 . [CSA]
  • Cleve , G .; Hoyer , G . A .; Schulz , G .; Vorbrueggen , H . Synthesis of nucleosides. VIII. NMR and CD spectra of pyrimidine nucleosides and their 2-thio analogs . Chem. Ber . 1973 , 106 , 3062 – 3072 . [CSA]
  • Ahmed , A . A.M . Synthesis and reactions of some new bis(heterocycles) and hetero macrocycles using versatile starting materials . M.Sc. Thesis ; Faculty of Science, Department of Chemistry, Cairo University : Giza, , Egypt , 2004 .
  • Vogel's Textbook of Practical Organic Chemistry, , 4th Ed .; Furniss , B . S ., Hannaford , A . J ., Rogers , V ., Smith , P . W.G ., Tatchell , A . R ., Eds.; Longman Group Limited : Harlow, , UK , 1978 ; 457 .

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