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Articles

Polymeric drug based on acrylates for biological applications: synthesis, characterization, antimicrobial, and drug release study

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Pages 753-761 | Received 22 Dec 2013, Accepted 17 Apr 2014, Published online: 21 May 2014

References

  • Vogl O, Tirrell D. Functional polymers with biologically active groups. J. Macromol. Sci. Chem. 1979;13:415–439.10.1080/00222337908068110
  • Ayfer B, Dizman B, Elasri MO, Mathias LJ, Avci D. Synthesis and antibacterial activities of new quaternary ammonium monomers. Des. Monomers Polym. 2005;8:437–451.10.1163/1568555054937935
  • Ballesteros JF, Sanz MJ, Ubeda A, Miranda MA, Iborra S. Synthesis and pharmacological evaluation of 2′-hydroxychalcones and flavones as inhibitors of inflammatory mediators generation. J. Med. Chem. 1995;38:2794–2797.10.1021/jm00014a032
  • Viana GS, Bandeira MA, Matos F. Analgesic and antiinflammatory effects of chalcones isolated from Myracrodruon urundeuva allemão. J. Phytomedicine. 2003;10:189–195.10.1078/094471103321659924
  • Mukarami S, Muramatsu M, Aihara H, Otomo S. Oleic acid as an inhibitor of gastric H+, K(+)-ATPase. Biochem. Pharmacol. 1991;42:337–350. Retrieved from http://www.ncbi.nlm.nih.gov/pubmed/1646470.
  • Barfod L, Kemp K, Hansen M, Kharazmi A. Chalcones from Chinese liquorice inhibit proliferation of T cells and production of cytokines' International Immunopharmacology. Int. Immunopharmacol. 2002;2:545–555.10.1016/S1567-5769(01)00202-8
  • Liu M, Wilairat P, Go M-L. Antimalarial alkoxylated and hydroxylated chalcones [corrected]: structure-activity relationship analysis. J. Med. Chem. 2001;44:4443–4452.10.1021/jm0101747
  • Nielsen SF, Chen M, Theander TG, Kharazmi A, Brøgger Christensen SB. Synthesis of antiparasitic licorice chalcones. Bioorg. Med. Chem. Lett. 1995;5:449–452.10.1016/0960-894X(95)00053-V
  • Vogel S, Barbic M, Jürgenliemk G, Heilmann J. Synthesis, cytotoxicity, anti-oxidative and anti-inflammatory activity of chalcones and influence of A-ring modifications on the pharmacological effect. Eur. J. Med. Chem. 2010;45:2206–2213. Retrieved from http://www.ncbi.nlm.nih.gov/pubmed/20153559.10.1016/j.ejmech.2010.01.060
  • Zhao LM, Jin HS, Sun LP, Piao HR, Quan ZS. Synthesis and evaluation of antiplatelet activity of trihydroxychalcone derivatives. Bioorg. Med. Chem. Lett. 2005;15:5027–5029.10.1016/j.bmcl.2005.08.039
  • Nowakowska Z, Kędzia B, Schroeder G. Synthesis, physicochemical properties and antimicrobial evaluation of new (E)-chalcones. Eur. J. Med. Chem. 2008;43:707–713.10.1016/j.ejmech.2007.05.006
  • Nagaini Z, Fadzillah H, Hussain H, Kamaruddin K. Synthesis and antimicrobial studies of (E)-3-(4-Alkyloxyphenyl)-1-(2-hydroxyphenyl)prop-2-ene-1-one,(E)-3-(4-Alkyloxyphenyl)-1-(4-hydroxyphenyl)prop-2-ene-1-one and their analogues. World J. Chem. 2009;4:9–14.
  • Swamy PMG, Agasimundin YS. Synthesis and antimicrobial activity of some novel chalcones containing 3-hydroxy benzofuran. Acta Pharm. Sciencia. 2008;50:197–202.
  • Mayekar AN. Int. J. Chem. Synthesis, characterization and antimicrobial study of some new cyclohexenone derivatives. 2010;2:114–123.
  • de Carvalho Tavares LC, Johann S, Maria de Almeida Alves TMA, Guerra JC, Maria de Souza-Fagundes EMS, Cisalpino PS, Bortoluzzi AJ, Caramori GF, de Mattos Piccoli RMC, Braibante HTS, Braibante MEF, Pizzolatti MG, Pizzolatti G. Quinolinyl and quinolinyl N-oxide chalcones: synthesis, antifungal and cytotoxic activities. Eur. J. Med. Chem. 2011;46:4448–4456.10.1016/j.ejmech.2011.07.019
  • Nakagawa-Goto KN, Lee KH. Anti-AIDS agents 68. The first total synthesis of a unique potent anti-HIV chalcone from genus Desmos. Tetrahedron Lett. 2006;47:8263–8266.10.1016/j.tetlet.2006.09.110
  • Arun A, Reddy BSR. In vitro drug release studies of 2-hydroxyethyl acrylate or 2-hydroxypropyl methacrylate-4-{(1E,4E)-5-[4-(acryloyloxy)phenyl]-3-oxopenta-1,4-dienyl}phenyl acrylate copolymer beads. J. Bioact. Compat. Polym. 2003;18:219–300.10.1177/0883911503035385
  • Esquivel-Guzmán JA, Zaragoza-Galán G, Ortíz-Palacios J, Rivera E. Synthesis and characterization of novel polymers bearing fluorescein units: thermal and optical properties. Des. Monomers Polym. 2012;15:561–574.10.1080/1385772X.2012.688339
  • Vijayanand PS, Kato S, Koyama M, Satokawa S, Kojima T. Co-polymerization of 4-biphenyl methacrylate with methyl methacrylate: synthesis, characterization and determination of monomer reactivity ratios. Des. Monomers Polym. 2007;10:375–388. Retrieved from http://www.jiscjournalarchives.ac.uk/openurl.html?ref=brill/1385772X/pdf/1385772x_v10n4_20070814_s7.pdf.
  • Bolard J, Legrand P, Heitz F, Cybulska B. One-sided action of amphotericin B on cholesterol-containing membranes is determined by its self-association in the medium. Biochemistry. 1991;30:5707–5715.10.1021/bi00237a011
  • Arun A, Reddy BSR. In vitro drug release studies from the polymeric hydrogels based on HEA and HPMA using 4-{(E)-[(3Z)-3-(4-(acryloyloxy)benzylidene)-2-hexylidene]methyl}phenyl acrylate as a crosslinker. Biomaterials. 2005;26:1185–1193. Retrieved from http://www.sciencedirect.com/science/article/pii/S0142961204003680.
  • Sharkawi T, Leyni-Barbaz D, Chikh N, McMullen JN. Evaluation of the in vitro drug release from resorbable biocompatible coatings for vascular stents. J. Bioact. Compat. Polym. 2005;20:153–168.10.1177/0883911505051661
  • Gallardo A, Parejo C, San Román J. NSAIDs bound to methacrylic carriers: microstructural characterization and in vitro release analysis. J. Controlled Release. 2001;71:127–140.10.1016/S0168-3659(01)00212-7
  • Elvira C, Gallardo A, Lacriox N, Schacht E, Sanroman J. Incorporation of salicylic acid derivatives to hydrophilic copolymer systems with biomedical applications. J. Mater. Sci. Mater. Med. 2001;12:535–542.
  • Davaran S, Hanaee J, Khosravi A. Release of 5-amino salicylic acid from acrylic type polymeric prodrugs designed for colon-specific drug delivery. J. Controlled Release. 1999;58:279–287.10.1016/S0168-3659(98)00167-9
  • McCormick CL. Controlled activity polymers with pendent metribuzin: effect of structure on hydrolytic release. Ann. N.Y. Acad. Sci. 1985;446:76–92.10.1111/nyas.1985.446.issue-1

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