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Original Articles

Synthesis, Antimicrobial Evaluation of 4-[(arylimino) methyl-5-(4-[(aryl) methylidene] amino) Phenyl)-4H-1, 2, 4-triazole-3-thiol Derivatives

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Pages 470-477 | Received 23 Apr 2016, Accepted 14 Jul 2016, Published online: 06 Oct 2016

References

  • Miniyar, P.B., Barmade, M.A., Mahajan, A.A. (2015). Synthesis and biological evaluation of 1-(5-(2-chloroquinolin-3-yl)-3-phenyl-1H-pyrazol-1-yl) ethanone derivatives as potential antimicrobial agents. J. Saudi. Chem. Soc., 19: 655–660. doi: 10.1016/j.jscs.2013.12.004
  • Kulandaivelu, U., Padmini, V.G., Suneetha, K., Shireesha, B., Vidyasagar, J.V., Rao, T.R., Jayaveera, K.N., Basu, A., Jayaprakash, V. (2011). Synthesis, antimicrobial and anticancer activity of new thiosemicarbazones derivatives. Arch. Pharm., 344(2): 84–90. doi: 10.1002/ardp.201000201
  • Brown, R.C.D. (1998). Recent developments in solid phase organic synthesis. J. Chem. Soc. Perkin. Trans.,1: 3293–3320. doi: 10.1039/a805801f
  • Shridhar, M., Arun, M.I., Shrikrishna, I., Akhila, D.S., Hoong, K.F. (2013). Synthesis, characterization and antibacterial activity of some new pyrazole based Schiff bases. Arabian J. Chem., 6: 335–340. doi: 10.1016/j.arabjc.2011.10.009
  • Seyhan, E., Sultan, N., Rukiye, B. (1998). Synthesis and antimicrobial activity of N-[(α-methyl)-benzylidene]-(3-substituted-1,2,4-triazol-5-yl-thio)acetohydrazides.II Farmaco, 3(12): 773–776.
  • Datoussaid, Y., Othman, A.A., Kirsch, G.S. (2012). Synthesis and antibacterial activity of some 5,5’-(1,4-phenylene)-bis-1,3,4-oxadiazole and bis-1,2,4-triazole derivatives as precursors of new s-nucleosides. Afr. J .Chem., 65: 30–35.
  • Aamer, S., Amara, M. (2015). Novel isochroman-triazoles and thiadiazole hybrids: Design, synthesis and antimicrobial activity. J. Saudi. Chem. Soc., Accepted.
  • Ma, Y., Liu, R., Gong, X., Li, Z., Huang, Q., Wang, H., Song, G. (2006). Synthesis and herbicidal activity of N,N-diethyl-3-(arylselenonyl)-1H-1,2,4-triazole-1-carboxamide. J. Agric Food Chem., 54(20): 7724–7728. doi: 10.1021/jf0609328
  • Tarzia, G., Ocelli, E., Toja, E., Barone, D., Corsico, N., Gallico, L., Luzzani, F. (1988). 6-(al-kylamino) -3-aryl-1,2,4-triazolo[3,4-a] phthalazines. A new class of benzodiazepine receptor ligands. J., Med. Chem., 31(6): 1115–1123. doi: 10.1021/jm00401a010
  • Pattan, S., Gadhave, P., Tambe, V., Dengale, S., Thakur, D., Hiremath, S.V., Shete, R.V., Deotarse, P. (2012). Synthesis and evaluation of some novel 1,2,4-triazole derivatives for antimicrobial, antitubercular and anti-inflammatory activities. Ind. J. Chem.,41B: 297–301.
  • Husain, A., Rashid, M., Mishra, R., Parveen, S., Shin, D., Kumar, D. (2012). Benzimidazole bearing oxadiazole and triazolo-thiadiazoles nucleus: design and synthesis as anticancer agents. Bioorg. Med. Chem. Lett., 22: 5438–5444. doi: 10.1016/j.bmcl.2012.07.038
  • Shah, M.H., Hasalkar, M.Y., Patki, V.M., Deliwala, C.V., Sheth, U.K.(1969). New 1,2,4 (H)-triazole derivatives as diuretic agents J. Pharm. Sci., 58: 1398–1401. doi: 10.1002/jps.2600581123
  • Hunashal, R.D., Ronad, P.M., Maddi, V.S., Satyanarayana, D., Kamadod, M.A. (2014). Synthesis,anti-inflammatory and analgesic activity of 2-[4-(substituted benzylideneamino)-5-(substituted phenoxymethyl)-4H-1,2,4-triazol-3-ylthio] acetic acid derivatives. Arabian J. Chem., 7: 1070–1078. doi: 10.1016/j.arabjc.2011.01.003
  • Franciele, D., Marcelo, Gde, G., André Tiago, R.G., Natália, S., Diego, A., Cristiano, R.J., Lucielli, S.(2013). Involvement of the dopaminergic and serotonergic systems in the antidepressant-like effect caused by 4-phenyl-1-(phenylselanylmethyl)-1,2,3-triazole. Life Sci., 93: 393–400. doi: 10.1016/j.lfs.2013.07.024
  • Bhanojirao, M.E., Rajurkar, V.G. (2009). Synthesis and biological evaluation of 5-pyridine-4-(arylidine amino)-3-mercapto-4(H)-1,2,4-triazoles. Asian. J. Chem., 21(6): 4733–4736.
  • Rajurkar, V.G., Gadekar, K., Deshmukh, V.K. (2014). Synthesis, characterization and study of some n-substituted aryl-2-({4-[(substituted aryl carbamoyl) methyl]-5-(pyridin-4-yl)-4H-1, 2,4-triazol-3-yl} sulfanyl) acetamide. Iranian J. Pharma. Sci., 10(2): 21–34.
  • Rajurkar, V.G., Lambe, S.V., Deshmukh, V.K.(2015) Synthesis of some N-(4-(aryl)-2-thioxo-1,3-thiazol-3(2H)-yl)pyridine-4-carboxamide as antimicrobial and anti-inflammatory agents. Med. Chem., 5:6. http://dx.doi.org/10.4172/2161-0444.1000276. doi: 10.4172/2161-0444.1000276
  • Rajurkar, V.G., Pund, A.R. (2014). Novel linezolid like analogues: synthesis, characterization and biological evaluation. Iranian J. Pharma Sci., 10(2): 69–78.
  • Rajurkar, V.G., Gaikwad, S.S., Devdhe, S.J., Angadi, S. (2014). Synthesis and biological evaluation of novel 4-[4-(1H-benzimidazol-2ylmethoxy) phenyl]-6-(substituted phenyl) pyrimidin-2-amine as potent antimicrobial agents. Inter. J. Pharma Res. Scho., 3(1): 872–882.
  • Rajurkar, V.G., Patil, R.B., Bhanojirao, M.E., Pattan, S.R. (2012). Synthesis, characterization and antimicrobial, antifungal and antitubercular activity of some 3,5-substituted isoxazoles, 4-[(3, 5-substituted,1H-pyrazol-1-yl) carbonyl] pyridines and 4, 6-substituted pyrimidin-2-amines. International J. Adv. In Phar, Bio. and Chem., 1(1): 1–6.

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