Publication Cover
Synthetic Communications
An International Journal for Rapid Communication of Synthetic Organic Chemistry
Volume 33, 2003 - Issue 12
520
Views
22
CrossRef citations to date
0
Altmetric
Original Articles

Cannabinoid CB1 Receptor Chemical Affinity Probes: Methods Suitable for Preparation of Isopropyl [11,12-3H]Dodecylfluorophosphonate and [11,12-3H]Dodecanesulfonyl Fluoride

, &
Pages 2151-2159 | Received 28 Oct 2002, Published online: 17 Aug 2006

References

  • Devane , W.A. , Hanuš , L. , Breuer , A. , Pertwee , R.G. , Stevenson , L.A. , Griffin , G. , Gibson , D. , Mandelbaum , A. , Etinger , A. and Mechoulam , R. 1992 . Isolation and structure of a brain constituent that binds to the cannabinoid receptor . Science , 258 : 1946 – 1949 .
  • Cravatt , B.F. , Prospero-Garcia , O. , Siuzdak , G. , Gilula , N.B. , Hendriksen , S.J. , Boger , D.L. and Lerner , R.A. 1995 . Chemical characterization of a family of brain lipids that induce sleep . Science , 268 : 1506 – 1509 .
  • Martin , B.R. , Beletskaya , I. , Patrick , G. , Jefferson , R. , Winckler , R. , Deutsch , D.G. , Di Marzo , V. , Dasse , O. , Mahadevan , A. and Razdan , R.K. 2000 . Cannabinoid properties of methylfluorophosphonate analogs . J. Pharmacol. Exp. Ther. , 294 : 1209 – 1218 .
  • Deutsch , D.G. , Lin , S. , Hill , W.A.G. , Morse , K.L. , Salehani , D. , Arreaza , G. , Omeir , R.L. and Makriyannis , A. 1997 . Fatty acid sulfonyl fluorides inhibit anandamide metabolism and bind to the cannabinoid receptor . Biochem. Biophys. Res. Commun. , 231 : 217 – 221 .
  • Patricelli , M.P. , Lovato , M.A. and Cravatt , B.F. 1999 . Chemical and mutagenic investigations of fatty acid amide hydrolase: evidence for a family of serine hydrolases with distinct catalytic properties . Biochemistry , 38 : 9804 – 9812 .
  • Zhang , N. , Morimoto , H. , Williams , P.G. and Casida , J.E. 2000 . Synthesis of high specific activity [ethyl-1,2-3H]-labeled chlorpyrifos oxon and diazoxon . J. Labelled Compds. Radiopharm. , 43 : 1275 – 1282 .
  • Quistad , G.B. , Nomura , D.K. , Sparks , S.E. , Segall , Y. and Casida , J.E. 2002 . Cannabinoid CB1 receptor as a target for chlorpyrifos oxon and other organophosphorus pesticides . Toxicol. Lett. , 135 : 89 – 93 .
  • Quistad , G.B. , Sparks , S.E. and Casida , J.E. 2001 . Fatty acid amide hydrolase inhibition by neurotoxic organophosphorus pesticides . Toxicol. Appl. Pharmacol. , 173 : 48 – 55 .
  • Quistad , G.B. , Sparks , S.E. , Segall , Y. , Nomura , D.K. and Casida , J.E. 2002 . Selective inhibitors of fatty acid amide hydrolase relative to neuropathy target esterase and acetylcholinesterase: toxicological implications . Toxicol. Appl. Pharmacol. , 179 : 57 – 63 .
  • Sparks , S.E. , Quistad , G.B. and Casida , J.E. 1999 . Organophosphorus pesticide-induced butyrylcholinesterase inhibition and potentiation of succinylcholine toxicity in mice . J. Biochem. Mol. Toxicol. , 13 : 113 – 118 .
  • Capodicasa , E. , Scapellato , M.L. , Moretto , A. , Caroldi , S. and Lotti , M. 1991 . Chlorpyrifos-induced delayed polyneuropathy . Arch. Toxicol. , 65 : 150 – 155 .
  • Segall , Y. , Quistad , G.B. , Sparks , S.E. , Nomura , D.K. and Casida , J.E. Unpublished Results
  • Dalla Cort , A. , Mandolini , L. and Masci , B. 1983 . Ring closure reactions. 21. Intramolecular β-elimination competing with ring formation from o-(ω-bromoalkoxy)phenoxides over a wide range of ring sizes . J. Org. Chem. , 48 : 3979 – 3982 .
  • Cid , M.M. 1996 . Synthesis of 4-substituted-1,4-dihydropyridines . Tetrahedron Lett. , 37 : 6033 – 6036 .
  • Wu , S.-Y. , Yoshida , M. and Casida , J.E. 1994 . 2-Octyl-4H-1,3,2-benzodioxaphosphorin 2-oxide labeled with tritium in the octyl and aryl moieties . J. Labelled Compds. Radiopharm. , 34 : 921 – 927 .
  • Hur , J.H. , Wu , S.-Y. and Casida , J.E. 1992 . Oxidative chemistry and toxicology of S, S, S-tributyl phosphorotrithioate (DEF Defoliant) . J. Agric. Food Chem. , 40 : 1703 – 1709 .

Reprints and Corporate Permissions

Please note: Selecting permissions does not provide access to the full text of the article, please see our help page How do I view content?

To request a reprint or corporate permissions for this article, please click on the relevant link below:

Academic Permissions

Please note: Selecting permissions does not provide access to the full text of the article, please see our help page How do I view content?

Obtain permissions instantly via Rightslink by clicking on the button below:

If you are unable to obtain permissions via Rightslink, please complete and submit this Permissions form. For more information, please visit our Permissions help page.