Publication Cover
Synthetic Communications
An International Journal for Rapid Communication of Synthetic Organic Chemistry
Volume 34, 2004 - Issue 4
264
Views
5
CrossRef citations to date
0
Altmetric
Original Articles

5‐Amino‐2H‐pyran‐3(6H)‐one, 1, a Convenient Intermediate in the Synthesis of Pyran Containing 1,4‐Dihydropyridines

, , &
Pages 557-565 | Received 07 Aug 2003, Published online: 16 Aug 2006

References

  • Frank , C. A. , Forst , J. M. , Grant , T. , Harris , R. J. , Kau , S. T. , Li , J. H. , Ohnmacht , C. J. , Smith , R. W. , Trainor , D. A. and Trivedi , S. 1993 . Dihydropyridine KATP potassium channel openers . Bioorg. Med. Chem. Lett. , 3 ( 12 ) : 2725 – 2726 .
  • Trivedi , S. , Potter‐Lee , L. , McConville , M. W. , Li , J. H. , Ohnmacht , C. J. , Trainor , D. A. and Kau , S. T. 1995 . K‐channel opening activity of dihydropyridine ZM244085: effect on 86Rb efflux and 3H‐P1075 binding in urinary bladder smooth muscle . Res. Commun. Mol. Pathol. Pharmacol. , 88 ( 2 ) : 137 – 151 . [PUBMED] [INFOTRIEVE] [CSA]
  • Carroll , W. A. , Agrios , K. A. , Altenbach , R. J. , Drizin , I. and Kort , M. E. Pyrano, Piperidino, and Thiopyrano Compounds and Methods of Use . US Patent US 6,191,140 B1 . February 20, 2001 .
  • Terasawa , T. and Okada , T. 1977 . Novel heterocyclic synthons. Synthesis and properties of thia‐ and oxacyclohexane‐3,5‐diones . J. Org. Chem. , 42 ( 7 ) : 1163 – 1169 .
  • Morgan , M. A. and Van Heyningen , E. 1957 . 2H‐Pyran‐3,5(4H,6H)‐diones . J. Am. Chem. Soc. , 79 ( 2 ) : 422 – 424 .
  • Ziegler , F. E. and Bennett , G. B. 1973 . Claisen rearrangement in indole alkaloid synthesis. Total synthesis of (±)‐tabersonine . J. Am. Chem. Soc. , 95 ( 22 ) : 7458 – 7464 . [PUBMED] [INFOTRIEVE]
  • Li , W. , Wayne , G. S. , Lallaman , J. E. , Wittenberger , S. J. and King , S. A. Scalable synthesis of pyran-3,5-dione . 222nd ACS National Meeting . August 26–30 2001 , Chicago, IL, United States. Abstracts of Papers , Washington, DC : American Chemical Society . ORGN‐285
  • Baraldi , P. G. , Simoni , D. and Manfredini , S. 1983 . An improved preparation of enaminones from 1,3‐diketones and ammonium acetate or amine acetates . Synthesis , : 902 – 903 . [CROSSREF]
  • Huang , Y. and Hartmann , R. W. 1998 . The improved preparation of 7,8‐dihydroquinolin‐5(6H)‐one and 6,7‐dihydro‐5H‐1‐pyrindin‐5‐one . Synth. Commun. , 28 ( 7 ) : 1197 – 1200 .
  • Zymalkowski , F. and Rimek , H. 1961 . New synthesis of benzoyltetrahydroquinoline . Arch. Pharm. , 294 : 759 – 765 .
  • Kikani , B. B. , Mckee , J. R. and Zanger , M. 1991 . An efficient synthesis of 3‐aminocyclopent‐2‐en‐1‐one . Synthesis , : 176 [CROSSREF]
  • Ohnmacht , C. J. Acridine Derivatives as Therapeutic Agent . European Patent EP0539153 . April 23, 1997 .
  • Altenbach , R. J. , Kalvoda , L. and Carroll , W. A. 2004 . A convenient multigram scale synthesis of tetrahydrothiophene‐3‐one‐1,1‐dioxide . Synth. Commun. , 34 ( 4 ) : 541 – 548 .
  • Nakagawa , S. , Naito , T. and Kawaguchi , H. 1979 . Structures of BU‐2313 A and B, new antianaerobic antibiotics and syntheses of their analogs . Heterocycles , 13 ( Spec. Issue ) : 477 – 495 .
  • Fehnel , E. A. and Paul , A. P. 1955 . Thiapyran derivatives. V. The monosulfinyl and monosulfonyl analogs of phloroglucinol . J. Am. Chem. Soc. , 77 ( 16 ) : 4241 – 4244 .

Reprints and Corporate Permissions

Please note: Selecting permissions does not provide access to the full text of the article, please see our help page How do I view content?

To request a reprint or corporate permissions for this article, please click on the relevant link below:

Academic Permissions

Please note: Selecting permissions does not provide access to the full text of the article, please see our help page How do I view content?

Obtain permissions instantly via Rightslink by clicking on the button below:

If you are unable to obtain permissions via Rightslink, please complete and submit this Permissions form. For more information, please visit our Permissions help page.