Bibliography
- NORMAN P: Developing anti- inflammatory drugs for the treatment of COPD. Inflamm. Res. in press.
- •Up-to-date review of approaches to the treatment of COPD.
- STOCKLEY RA: Proteases and antiproteases. Novartis Found Symp (2001) 234:189–199.
- ••Excellent description of this key hypothesis.
- BERNSTEIN PR, EDWARDS PD, WILLIAMS JC: Inhibitors of human leukocyte elastase. Prog. Med. Chem. (1994) 31:59–120.
- ••Excellent review of earlier chemical approaches to this target.
- TREMBLAY GM, JANELLE ME BOURBONNAIS Y: Anti-inflammatory activity of neutrophil elastase inhibitors. Cum Opin. Investig. Drugs (2003) 4:556–565.
- •Recent review of what has been an intensively targeted area.
- OHBAYASHI H: Neutrophil elastase inhibitors as treatment for COPD. Expert Opin. Investig. Drugs (2002) 11:965–980.
Websites
- www.etiologics.com/docs/etiobayer.pdf Etiologics Ltd, Press release 16 June 2003.
- http://www.etiologics.com/therapeutic-respiratory/respipe.htm Etiologics Ltd, Illustrative syntheses of the claimed elastase inhibitors.